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Search Result

Search Results for " blocker "

Targets

Others

611

Compounds

21

Natural Products

4

Libraries

Cat No. Product Name Synonyms Targets
T11063 DMT1 blocker 1 Others
DMT1 blocker 1 is a blocker of divalent metal transporter 1 (DMT1) with IC50 of 0.64 μM, which is expected to block the absorption of iron by intestinal cells in vivo.
T11064 DMT1 blocker 2 Others
DMT1 blocker 2, compound 12f, is a direct inhibitor of divalent metal transporter 1 (DMT1) with an IC50 hydrogen peroxide value of 0.83, which is expected to block iron uptake by intestinal epithelial cells in vivo.
T12504 (+)-KCC2 blocker 1 Potassium Channel
(+)-KCC2 blocker 1 is a selective blocker of KCC2 (IC50 = 0.4 μM).
T10690 Cav 2.2 blocker 1 Calcium Channel
Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
T72170 NaV1.2/1.6 channel blocker-1 Sodium Channel
NaV1.2/1.6 channel blocker-1 is a potent NaV1.2/1.6 channel blocker with inhibitory effects on rNaV1.6 and hNaV1.2.NaV1.2 channel blocker-1 can be used in the study of generalised epilepsy and movement disorders.
T39717 VGSC blocker-1
VGSC blocker-1 is a powerful small molecule that serves as a blocker for the neonatal isoform of the VGSC subtype known as Nav1.5 (nNav1.5). It effectively blocks INa peak currents by 34.9% at a concentration of 1 μM, an...
T28132 NaV1.7 Blocker-801
NaV1.7 Blocker-801 is a potent NaV1.7 blocker.
T11927 M2 ion channel blocker Others
M2 ion channel blocker ,Antiviral agent, is capable of inhibiting and blocking the activity of M2 ion channel.
T69387 NMO-IgG blocker A-01
NMO-IgG blocker A-01 is a idiotype-specific blocker of neuromyelitis opticaimmunoglobulin g (nmo-igg) binding to aquaporin-4 (aqp4)
T12153 N-type calcium channel blocker-1 Calcium Channel
N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.
T80930 TRPV2-selective blocker 1
TRPV2-selective blocker 1 (compound IV2-1) is a selective inhibitor of the TRPV2 channel, exhibiting an IC50 value of 6.3 μM. It specifically targets the TRPV2 channel without impacting related TRPV1, TRPV3, or TRPV4 cha...
T62586 Cav 2.2/3.2 blocker 1
Cav 2.2/3.2 blocker 1 (Compound 9e) is a neuronal calcium channel blocker that acts on Cav2.2 (IC50: 1.22 μM) and Cav3.2 (IC50: 80 μM). Can penetrate the central nervous system.
T26817 Bim-BLK-A Bim Blocker A,Compound A,Bim BLK A,BimBLKA
Bim-BLK-A efficiently blocks Bim-induced apoptosis after Bax is activated on the mitochondria. The cellular target of Bim-BLK-A was identified to be the succinate dehydrogenase subunit B (SDHB) protein of complex II of t...
T83705 BING TFA Blocker of Inter-membrane Stress Responses of Gram-negative Bacteria
BING, a antimicrobial peptide discovered in Japanese medaka fish (O. laptipes), originates from vacuolar protein sorting-associated protein 13D-like (Vps13D). It exhibits efficacy against a range of Gram-negative and Gra...
T15385 Glibornuride Potassium Channel
Glibornuride is an ATP-sensitive K+ channels (KATP channel) blocker ( pKi: 5.75). It is an antidiabetic agent.
T0440 Oxcarbazepine GP 47680 Apoptosis , Sodium Channel
Oxcarbazepine (GP 47680) is an Anti-epileptic Agent. The physiologic effect of oxcarbazepine is by means of Decreased Central Nervous System Disorganized Electrical Activity.
T21454 Nicardipine Cardene,Dagan,Antagonil,Flusemide Calcium Channel
Nicardipine (Cardene), a calcium channel blockers belonging to the dihydropyridine class, is a drug used to treat angina and high blood pressure.
T3574 Sematilide hydrochloride CK-1752A,CK-1752,Sematilide HCl Potassium Channel
Sematilide hydrochloride (CK-1752) is a class III antiarrhythmic. It is a selectively delayed rectifier K+ current (IKr) channel blocker. It inhibits rapidly activating Ik in guinea pig atrial myocytes, resulting in the ...
T8388 Vonoprazan TAK-438 (free base) Proton pump
Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer and reflux esophagitis
T0866 Propafenone Rythmol,Propafenonum Potassium Channel , MRP , Sodium Channel
Propafenone (Propafenonum) is only found in individuals that have used or taken this drug. It is an antiarrhythmia agent that is particularly effective in ventricular arrhythmias. It also has weak beta-blocking activity....
T7806 Licarbazepine ​10,11-hydroxy-10,11 Dihydrocarbamezer Others
Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial seizures and bipolar disorders.
T21254 Vonoprazan Fumarate TAK-438,TAK 438,Vonoprazan Fumurate,TAK438 Proton pump
Vonoprazan Fumarate (TAK438) , a novel potassium-competitive acid blocker, inhibits gastric acid secretion. Vonoprazan Fumarate (TAK438) inhibited H+,K+-ATPase activity in porcine gastric microsomes with IC50 value of 19...
T1215 Nicardipine hydrochloride RS-69216,Nicardipine HCl,YC-93 Hydrochloride Calcium Channel , Adrenergic Receptor , AChR , Autophagy
Nicardipine hydrochloride (YC-93 Hydrochloride) is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nicardipine (Nifedipine Family) blocks cal...
T0342 Carvedilol phosphate hemihydrate Carvedilol phosphate,BM 14190 (phosphate hemihydrate) VEGFR , Others , Potassium Channel , LDL , Integrin , Gap Junction Protein , NADPH , Adrenergic Receptor , Autophagy
Carvedilol phosphate hemihydrate (BM 14190 phosphate hemihydrate) is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intrinsic sympathom...
T1615 Irbesartan SR-47436,BMS-186295 Apoptosis , RAAS
Irbesartan (SR-47436) is an Angiotensin 2 Receptor Blocker. The mechanism of action of irbesartan is as an Angiotensin 2 Receptor Antagonist.
T3280 Clodronate disodium tetrahydrate clodronic acid disodium tetrahydrate,Disodium clodronate tetrahydrate,Clastoban,Clodronate disodium IL Receptor , TNF
Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.
T6666 Sevelamer Carbonate Others
Sevelamer carbonate is a non-absorbed phosphate binding crosslinked polymer, with the same polymeric structure as sevelamer hydrochloride, in which carbonate replaces chloride as the counterion.
T22330 Fenamic acid 2-Anilinobenzoic acid,Diphenylamine-2-carboxylic acid,2-(Phenylamino)benzoic acid,N-Phenylanthranilic acid Chloride channel
Fenamic acid (N-Phenylanthranilic acid) is a chloride channel blocker that causes renal papillary necrosis in rats. Fenamic acid serves as a parent structure for several nonsteroidal anti-inflammatory drugs (NSAIDs), inc...
T23301 (S)-(+)-Niguldipine hydrochloride Others
(S)-(+)-Niguldipine hydrochloride is a L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist.
T10813 Cilobradine hydrochloride DK-AH 269 HCN Channel
Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels.
T26689 AVE-0118 AVE 0118,AVE0118 Potassium Channel
AVE-0118 is a potassium channel blocker and suppresses persistent atrial fibrillation.
T29050 UK 66914 UK66914,UK-66914 Potassium Channel
UK 66914 is a K(+) channel blocker for the study of cardiac arrhythmias.
T79835 Aneratrigine hydrochloride Sodium Channel
Aneratrigine hydrochloride is a sodium channel protein type 9 subunit blocker that may be used for the prevention or treatment of sodium channel blocker-related diseases.
T3557 GAL-021 GAL 021 Potassium Channel
GAL-021 an intravenous BKCa-channel blocker.
T20341 DNDS CFTR
DNDS is a channel blocker of voltage-dependent cystic fibrosis transmembrane conductance regulator (CFTR).
T15143 DMP-543 XR-543 Others , Potassium Channel
DMP-543 (XR-543) is a potassium channel (KV7 channel) blocker that enhances the release of neurotransmitters.
T9709 TRPM8 antagonist 3 TRP/TRPV Channel
TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).
T60010 BTT-266 Calcium Channel
BTT-266 is a blocker of voltage-gated calcium channel for pain management.
T15174 DSP-2230 Sodium Channel
DSP-2230 is a selective blocker of Nav1.7/Nav1.8.
T17263 XEN907 Others
XEN907 is a novel spiro oxindole NaV1.7 blocker. XEN907 also inhibits hNaV1.7 (IC50: 3 nM).
T3703 ABT-639 ABT 639 Calcium Channel
ABT-639 is a potent and selective T-type calcium channel blocker.
T6577 Manidipine Iperten,Franidipine,Artedil Calcium Channel
Manidipine (Iperten), a calcium channel blocker, which is dihydropyridine type. It is utilized
T31716 Etidocaine Hydrochloride W-19053,Duranest,W19053,W 19053 Sodium Channel
Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel.
T31614 Elpetrigine GW-273293,JZP 4,JZP4,GW273293,JZP-4,GW 273293
Elpetrigine( GW 273293, JZP-4) is effective calcium and sodium channel blocker and is currently being evaluated in patients as an anticonvulsant and mood stabilizer.
T22745 DPO-1 Potassium Channel
DPO-1 is a blocker of IKur ultrarapid delayed rectifier potassium current and KV1.5 channels
T22675 Co 102862 V 102862 Others , Sodium Channel
Co 102862 is a voltage-gated sodium channel blocker. Co 102862 can be used for anticonvulsant studies.
T16514 PF 04531083 Others , Sodium Channel
PF 04531083 is a selective blocker of the NaV1.8 channel. PF 04531083 can be used for neuropathic and inflammatory pain studies.
T7811 Pilsicainide HCl SUN 1165 Sodium Channel
Pilsicainide HCl (SUN 1165) is a pure sodium channel blocker
T1422 Nilvadipine FK235,FR34235,ARC029 Calcium Channel
Nilvadipine (FK235), a calcium channel blocker (CCB), is utilized for treatment of hypertension.
T2519 Lercanidipine Masnidipine Calcium Channel
Lercanidipine (Masnidipine) is a calcium channel blocker of the dihydropyridine class.

Compounds

DMT1 blocker 1
T11063
Synonym:
Target: Others
DMT1 blocker 2
T11064
Synonym:
Target: Others
(+)-KCC2 blocker 1
T12504
Synonym:
Target: Potassium Channel
Cav 2.2 blocker 1
T10690
Synonym:
Target: Calcium Channel
NaV1.2/1.6 channel blocker-1
T72170
Synonym:
Target: Sodium Channel
VGSC blocker-1
T39717
Synonym:
Target:
NaV1.7 Blocker-801
T28132
Synonym:
Target:
M2 ion channel blocker
T11927
Synonym:
Target: Others
NMO-IgG blocker A-01
T69387
Synonym:
Target:
N-type calcium channel blocker-1
T12153
Synonym:
Target: Calcium Channel
TRPV2-selective blocker 1
T80930
Synonym:
Target:
Cav 2.2/3.2 blocker 1
T62586
Synonym:
Target:
Bim-BLK-A
T26817
Synonym: Bim Blocker A,Compound A,Bim BLK A,BimBLKA
Target:
BING TFA
T83705
Synonym: Blocker of Inter-membrane Stress Responses of Gram-negative Bacteria
Target:
Glibornuride
T15385
Synonym:
Target: Potassium Channel
Oxcarbazepine
T0440
Synonym: GP 47680
Target: Apoptosis, Sodium Channel
Nicardipine
T21454
Synonym: Cardene,Dagan,Antagonil,Flusemide
Target: Calcium Channel
Sematilide hydrochloride
T3574
Synonym: CK-1752A,CK-1752,Sematilide HCl
Target: Potassium Channel
Vonoprazan
T8388
Synonym: TAK-438 (free base)
Target: Proton pump
Propafenone
T0866
Synonym: Rythmol,Propafenonum
Target: Potassium Channel, MRP, Sodium Channel
Licarbazepine
T7806
Synonym: ​10,11-hydroxy-10,11 Dihydrocarbamezer
Target: Others
Vonoprazan Fumarate
T21254
Synonym: TAK-438,TAK 438,Vonoprazan Fumurate,TAK438
Target: Proton pump
Nicardipine hydrochloride
T1215
Synonym: RS-69216,Nicardipine HCl,YC-93 Hydrochloride
Target: Calcium Channel, Adrenergic Receptor, AChR, Autophagy
Carvedilol phosphate hemihydrate
T0342
Synonym: Carvedilol phosphate,BM 14190 (phosphate hemihydrate)
Target: VEGFR, Others, Potassium Channel, LDL, Integrin, Gap Junction Protein, NADPH, Adrenergic Receptor, Autophagy
Irbesartan
T1615
Synonym: SR-47436,BMS-186295
Target: Apoptosis, RAAS
Clodronate disodium tetrahydrate
T3280
Synonym: clodronic acid disodium tetrahydrate,Disodium clodronate tetrahydrate,Clastoban,Clodronate disodium
Target: IL Receptor, TNF
Sevelamer Carbonate
T6666
Synonym:
Target: Others
Fenamic acid
T22330
Synonym: 2-Anilinobenzoic acid,Diphenylamine-2-carboxylic acid,2-(Phenylamino)benzoic acid,N-Phenylanthranilic acid
Target: Chloride channel
(S)-(+)-Niguldipine hydrochloride
T23301
Synonym:
Target: Others
Cilobradine hydrochloride
T10813
Synonym: DK-AH 269
Target: HCN Channel
AVE-0118
T26689
Synonym: AVE 0118,AVE0118
Target: Potassium Channel
UK 66914
T29050
Synonym: UK66914,UK-66914
Target: Potassium Channel
Aneratrigine hydrochloride
T79835
Synonym:
Target: Sodium Channel
GAL-021
T3557
Synonym: GAL 021
Target: Potassium Channel
DNDS
T20341
Synonym:
Target: CFTR
DMP-543
T15143
Synonym: XR-543
Target: Others, Potassium Channel
TRPM8 antagonist 3
T9709
Synonym:
Target: TRP/TRPV Channel
BTT-266
T60010
Synonym:
Target: Calcium Channel
DSP-2230
T15174
Synonym:
Target: Sodium Channel
XEN907
T17263
Synonym:
Target: Others
ABT-639
T3703
Synonym: ABT 639
Target: Calcium Channel
Manidipine
T6577
Synonym: Iperten,Franidipine,Artedil
Target: Calcium Channel
Etidocaine Hydrochloride
T31716
Synonym: W-19053,Duranest,W19053,W 19053
Target: Sodium Channel
Elpetrigine
T31614
Synonym: GW-273293,JZP 4,JZP4,GW273293,JZP-4,GW 273293
Target:
DPO-1
T22745
Synonym:
Target: Potassium Channel
Co 102862
T22675
Synonym: V 102862
Target: Others, Sodium Channel
PF 04531083
T16514
Synonym:
Target: Others, Sodium Channel
Pilsicainide HCl
T7811
Synonym: SUN 1165
Target: Sodium Channel
Nilvadipine
T1422
Synonym: FK235,FR34235,ARC029
Target: Calcium Channel
Lercanidipine
T2519
Synonym: Masnidipine
Target: Calcium Channel
1 2 3 4 5 6 7 8 9 10 11 12 13
Cat No. Product Name Synonyms Targets
T3S0081 Oxypeucedanin (+-)-Oxypeucedanin,Oxypeucadanin Potassium Channel
1. Oxypeucedanin ((+-)-Oxypeucedanin) has novel anticancer effect, mediated via induction of G2-M cell cycle arrest and apoptosis in human prostate carcinoma DU145 cells. 2. Oxypeucedanin is a kind of open-channel blocke...
T0801 Tannic acid Gallotannic acid Potassium Channel , HER , CXCR
Tannic acid (Gallotannic acid) is a novel hERG channel blocker.
T3054 Daurisoline (R,R)-Daurisoline Others , Potassium Channel , Autophagy
Daurisoline ((R,R)-Daurisoline) is a hERG inhibitor. Daurisoline is also an autophagy blocker.
T23107 Ononetin 2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone TRP/TRPV Channel
Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).
T0792 (-)-Sparteine sulfate pentahydrate (-)-Sparteine Sulfate,Lupinidine sulfate pentahydrate,(-)-Sparteine sulfate salt,sulfate pentahydrate Sodium Channel
(-)-Sparteine sulfate pentahydrate ((-)-Sparteine Sulfate) is a class 1a antiarrhythmic agent and a sodium channel blocker. It can chelate the bivalents calcium and magnesium.
T6631 Quinine hydrochloride dihydrate Quinine HCl Dihydrate Potassium Channel , Parasite
Quinine hydrochloride dihydrate (Quinine HCl Dihydrate) is a white crystalline K+ channel blocker, used to treat malaria.
T6S0084 Tuberostemonine Tuberstemonine Parasite
1. Tuberostemonine (Tuberstemonine) exhibits relatively higher intestinal permeabilities. 2. Tuberostemonine acts in part as an open-channel blocker at the crayfish neuromuscular junction.
T16535 Picrotoxinin Chloride channel , GABA Receptor
Picrotoxinin is a blocker of chloride channel and a noncompetitive antagonist of GABAA with an IC50 of 1.15 μM for α1β2γ2L GABAA. Picrotoxinin shows convulsant properties.
T3S0807 Berbamine CaMK , NF-κB , Autophagy
Berbamine is a natural product extracted from Phellodendron amurense. It acts as a calcium channel blocker and possesses anti-tumor, immunomodulatory, and cardiovascular effects.
T7853 (+)-Sparteine Pachycarpine AChR
(+)-Sparteine (Pachycarpine) is a natural product extracted from scotch broom, is a sodium channel blocker and a class 1a antiarrhythmic agent
T8716 Physalin F Apoptosis
Physalin F is a natural blocker of CaV2.3 (R-type) and CaV2.2 (N-type) voltage-gated calcium channels.It is a secosteroid with potent anti-inflammatory and immunomodulatory activities. Physalin F induces apoptosis of PBM...
TMA2106 (-)-Sparteine P450
Sparteine is a class 1a antiarrhythmic agent, a sodium channel blocker. The deficient debrisoquine hydroxylation of Sparteine is due to the absence of P-450IID1 protein in the livers of poor metabolizers.
T27191 D-Mannuronic Acid
D-Mannuronic Acid is a blocker of the TLR2 and TLR4 downstream signaling pathway. D-Mannuronic Acid effectively inhibits mRNA expression of MyD88 and p65, major subunit of nuclear factor-kappaB.
T3029 Sparteine sulfate Depasan,Tocosimplex,Actospar Others , Sodium Channel
Sparteine sulfate (Tocosimplex) is a class 1a antiarrhythmic agent and a sodium channel blocker. It can chelate the bivalents calcium and magnesium.
T62265 (+)-Sparteine sulfate pentahydrate
(+)-sparteine (sulfate pentahydrate) is a ganglion blocker that competitively blocks nicotinic acetylcholine receptors in neurons.
T75722 Chlorotoxin TFA
Chlorotoxin TFA, a peptide derived from the Leiurus quinquestriatus scorpion venom, functions as a chloride channel blocker [1] and exhibits anti-cancer activity [2].
TN3636 Chlorahololide C Potassium Channel
Chlorahololide C is a potent and selective potassium channel blocker, it exerts potent and selective inhibition on the delayed rectifier (I(K)) K(+) current with the IC(50) value of 3.6 +/- 10.1 mu M.
T21266 Quinine sulfate
Quinidine is an antiarrhythmic agent. Quinidine is a potent, orally active, selective cytochrome P450db inhibitor. Quinidine is also a blocker of K + channel with an IC 50 of 19.9 μM. Quinidine has potential to be used ...
TN3587 Capillarisin MMP , ERK , IL Receptor , BCL , VEGFR , TNF , NOS , NF-κB , TLR , MAPK , COX , DNA/RNA Synthesis , Prostaglandin Receptor , JNK , STAT
Capillarisin is a novel blocker of STAT3 activation and thus may have a potential in negative regulation of growth, metastasis, and chemoresistance of tumor cells, it inhibits cancer cell growth of osteosarcoma cells by ...
TN5061 Stephanine Adrenergic Receptor , Antifection
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of 6.76. Stephanine shows significant antiplasmodial activitie...
T75697 1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone
1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone, a diacylglycerol acyltransferase inhibitor and angiotensin II receptor blocker, exhibits IC50 values of 20.1 μM and 34.1 μM, respectively. Additionally, it demonstr...

Natural Products

Oxypeucedanin
T3S0081
Synonym: (+-)-Oxypeucedanin,Oxypeucadanin
Target: Potassium Channel
Tannic acid
T0801
Synonym: Gallotannic acid
Target: Potassium Channel, HER, CXCR
Daurisoline
T3054
Synonym: (R,R)-Daurisoline
Target: Others, Potassium Channel, Autophagy
Ononetin
T23107
Synonym: 2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone
Target: TRP/TRPV Channel
(-)-Sparteine sulfate pentahydrate
T0792
Synonym: (-)-Sparteine Sulfate,Lupinidine sulfate pentahydrate,(-)-Sparteine sulfate salt,sulfate pentahydrate
Target: Sodium Channel
Quinine hydrochloride dihydrate
T6631
Synonym: Quinine HCl Dihydrate
Target: Potassium Channel, Parasite
Tuberostemonine
T6S0084
Synonym: Tuberstemonine
Target: Parasite
Picrotoxinin
T16535
Synonym:
Target: Chloride channel, GABA Receptor
Berbamine
T3S0807
Synonym:
Target: CaMK, NF-κB, Autophagy
(+)-Sparteine
T7853
Synonym: Pachycarpine
Target: AChR
physalin F
T8716
Synonym:
Target: Apoptosis
(-)-Sparteine
TMA2106
Synonym:
Target: P450
D-Mannuronic Acid
T27191
Synonym:
Target:
Sparteine sulfate
T3029
Synonym: Depasan,Tocosimplex,Actospar
Target: Others, Sodium Channel
(+)-Sparteine sulfate pentahydrate
T62265
Synonym:
Target:
Chlorotoxin TFA
T75722
Synonym:
Target:
Chlorahololide C
TN3636
Synonym:
Target: Potassium Channel
Quinine sulfate
T21266
Synonym:
Target:
Capillarisin
TN3587
Synonym:
Target: MMP, ERK, IL Receptor, BCL, VEGFR, TNF, NOS, NF-κB, TLR, MAPK, COX, DNA/RNA Synthesis, Prostaglandin Receptor, JNK, STAT
Stephanine
TN5061
Synonym:
Target: Adrenergic Receptor, Antifection
1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone
T75697
Synonym:
Target:
Cat No. Product Name
L7300 Potassium Channel Blocker Library

160 compounds
A unique collection of 160 potassium channel blockers and agonists for high throughput and high content screening;
L7400 Sodium Channel Blocker Library

128 compounds
A unique collection of 128 sodium channel blockers and agonists for high throughput and high content screening;
L5800 Drug Metabolite/Impurity Library

200 compounds
A unique collection of 200 drug isomers/metabolites for high throughput screening (HTS) and high content screening (HCS);
L7110 Anti-Hypertension Compound Library

719 compounds
719 hypertension-related small molecules for high-throughput and high-content screening.

Libraries

Potassium Channel Blocker Library
L7300
Compounds: 160
Sodium Channel Blocker Library
L7400
Compounds: 128
Drug Metabolite/Impurity Library
L5800
Compounds: 200
Anti-Hypertension Compound Library
L7110
Compounds: 719
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