Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
Applied FilterClear all
TargetMol | Tags By Target
  • 5-HT Receptor
    (18)
  • Apoptosis
    (13)
  • Endogenous Metabolite
    (11)
  • Antioxidant
    (9)
  • GABA Receptor
    (8)
  • AChR
    (6)
  • Antibacterial
    (6)
  • COX
    (6)
  • Cholinesterase (ChE)
    (6)
  • Others
    (346)
Filter
Search Result
Results for "

rats

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    823
    TargetMol | Inhibitors_Agonists
  • Compound Libraries
    1
    TargetMol | Compound_Libraries
  • Peptide Products
    105
    TargetMol | Peptide_Products
  • Inhibitory Antibodies
    35
    TargetMol | Inhibitory_Antibodies
  • Natural Products
    107
    TargetMol | Natural_Products
  • Recombinant Protein
    7
    TargetMol | Recombinant_Protein
  • Isotope Products
    24
    TargetMol | Isotope_Products
  • Disease Modeling
    4
    TargetMol | Disease_Modeling_Products
  • Cell Research
    11
    TargetMol | Inhibitors_Agonists
Ziprasidone hydrochloride
Ziprasidone HCl, CP-88059 hydrochloride
T0031L122883-93-6
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
  • Inquiry Price
Size
QTY
Etomoxir
(R)-(+)-Etomoxir
T4535L124083-20-1
Etomoxir is a carnitine palmitoyltransferase 1a (CPT-1a) inhibitor that inhibits fatty acid oxidation by inhibiting CPT-1a and inhibits palmitate oxidation in humans, rats, and guinea pigs. Etomoxir has an inhibitory effect on adenine nucleotide translocase and can inhibit macrophage polarization by disrupting CoA homeostasis.
  • Inquiry Price
6-8 weeks
Size
QTY
TargetMol | Inhibitor Hot
CYP17-IN-1
T109232093317-51-0In house
CYP17-IN-1 is an effective oral inhibitor of CYP17 that can inhibit CYP17 in rats and humans with IC50 of 15.8 and 20.1 nM.
  • Inquiry Price
8-10 weeks
Size
QTY
Droloxifene
3-Hydroxytamoxifen
T1109882413-20-5In house
Droloxifene (3-Hydroxytamoxifen), a tamoxifen derivative, is an oral active and selective estrogen receptor modulator.Droloxifene induced p53 expression and apoptosis in McF-7 cells.Fluroxifene has anti-estrogen and anti-implantation effects.Fluroxifene prevented bone loss in ovariectomized rats.
  • Inquiry Price
6-8 weeks
Size
QTY
GW274150
T11518L210354-22-6In house
GW274150 is an orally active, selective and potent dual inhibitor of NADPH-dependent human nitric oxide synthase (iNOS) (Kd=40 nM) and rat inducible nitric oxide synthase (iNOS).GW274150 has a low activity against endothelial nitric oxide synthase (eNOS) and neuronal nitric oxide synthase (nNOS) in humans and rats. GW274150 showed protective effects in an inflammatory model of acute lung injury.
  • Inquiry Price
8-10 weeks
Size
QTY
INT-777
S-EMCA
T11662L1199796-29-6In house
INT-777 (S-EMCA) is a potent TGR5 agonist with an EC50 of 0.82 μM. INT-777 (S-EMCA) inhibits NLRP5-ASC inflammasome-mediated neuroinflammation via the TGR3 cAMP PKA signaling pathway after subarachnoid hemorrhage in rats.
  • Inquiry Price
8-10 weeks
Size
QTY
IQB-782
T1166840454-21-5In house
IQB-782 is a mucolytic agent with mucolytic expectorant activity.IQB-782 inhibits thrombin-activating fibrinolytic inhibitor (TAFI), protects rats from tobacco smoke-induced respiratory obstruction, reduces the viscosity of gastric mucin suspensions in vitro, and may be useful in studies of obstructive lung disease.IQB-782 has been shown to reduce the viscosity of gastric mucin suspensions in vitro.
  • Inquiry Price
6-8 weeks
Size
QTY
WAY127093B racemate
T13331145743-63-1In house
WAY127093B racemate is the racemic mixture of WAY127093B, a phosphodiesterase IV inhibitor with demonstrated oral activity in rats and guinea pigs.
  • Inquiry Price
6-8 weeks
Size
QTY
TargetMol | Inhibitor Sale
YM-46303
T13370171722-81-9In house
YM-46303 is a selective and potent muscarinic receptor antagonist that exhibits high affinity for the M3 receptor.YM-46303 can be used to study bradycardia in medullary rats.
  • Inquiry Price
6-8 weeks
Size
QTY
ZD-0892
T13389171964-73-1In house
ZD-0892 is a selective and potent inhibitor of neutrophil elastase, targeting human neutrophil elastase and porcine pancreatic elastase with Kis of 6.7 nM and 200 nM, respectively.
  • Inquiry Price
6-8 weeks
Size
QTY
Epsilon-momfluorothrin
Momfluorothrin, (Z,1R,3R)-
T136831065124-65-3In house
Epsilon-momfluorothrin (Momfluorothrin, (Z,1R,3R)-), a type I synthetic pyrethroid insecticide, exerts its insecticidal properties and triggers activation of the constitutive androstane receptor (CAR). Notably, its administration in rats has been observed to induce the development of hepatocellular tumors.
  • Inquiry Price
Size
QTY
TargetMol | Inhibitor Sale
Terbufibrol
T1391956488-59-6In house
Terbufibrol reduces the levels of serum total cholesterol in normal and hypercholesterolemic male rats.
  • Inquiry Price
8-10weeks
Size
QTY
Abaperidone
T14083183849-43-6In house
Abaperidone is a potent 5-HT2A receptor and dopamine D2 receptor antagonist with an IC50 of 6.2 for 5-HT2A receptors and 17 nM for dopamine D2 receptors.Abaperidone is a potentially atypical anti-psychotropic compound that reduces basal hsp70 mRNA expression in rat striatum and prefrontal cortex. expression in the striatum and prefrontal cortex of rats.
  • Inquiry Price
8-10weeks
Size
QTY
TargetMol | Inhibitor Sale
CGP48369
T14942135689-23-5In house
CGP48369 is a potent angiotensin II receptor antagonist with antihypertensive effects that enhances endothelium-dependent relaxation of coronary arteries in spontaneously hypertensive rats.
  • Inquiry Price
6-8 weeks
Size
QTY
Epristeride
SKF105657, ONO-9302
T15239119169-78-7In house
Epristeride (ONO-9302) is an orally active, selective and non-competitive steroidal 5-α-reductase isoform 2 inhibitor that inhibits SR isoform 2.Episteride reduces prostate size and improves symptoms in men with BPH.Episteride induces atrophy and apoptosis of the ventral prostate in rats.
  • Inquiry Price
6-8 weeks
Size
QTY
MRS 1754
T16140264622-58-4In house
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor, exhibiting very low affinity for A1 and A3 receptors in both humans and rats.
  • Inquiry Price
6-8weeks
Size
QTY
Furaprofen
R 803, R803, R-803
T1671567700-30-5In house
Furaprofen is an orally available, selective and potent HCV inhibitor with anti-inflammatory activity, inhibits carrageenan-induced paw edema in rats and inhibits cotton pellet-induced granulomas in rats at higher doses.
  • Inquiry Price
6-8 weeks
Size
QTY
Ranirestat
SX-3030, SX3030, AS-3201, AS3201, AS 3201
T16723147254-64-6In house
Ranirestat (AS-3201) is an orally active and potent aldose reductase (AR) inhibitor with neuroprotective properties that ameliorates peripheral nerve dysfunction in rats with advanced diabetic polyneuropathy.Ranirestat inhibits the inflammatory response of high glucose-exposed endothelial cells and may be useful for the study of diabetic sensory-motor polyneuropathy.
  • Inquiry Price
8-10 weeks
Size
QTY
Tiopinac
RS40974, RS-40974, RS 40974
T1710161220-69-7In house
Tiopinac (RS 40974) has anti-inflammatory and analgesic activity, and exhibits anti-flammatory activity in adrenalectomized rats.
  • Inquiry Price
6-8 weeks
Size
QTY
AMN082
AMN 082 dihydrochloride
T2193597075-46-2In house
AMN082 is an mGluR7 agonist with antidepressant effects. AMN082 has a neuroprotective effect on neuronal apoptosis in rats with traumatic brain injury and attenuates cocaine- and morphine-induced locomotor sensitization and cross-sensitization in mice.
  • Inquiry Price
7-10 days
Size
QTY
Spizofurone
Espizofurona, AG-629
T2482172492-12-7In house
Spizofurone (Espizofurona) has antiulcer activity, protective effect on the gastric mucosa of rats, and can increase alkaline secretion in isolated bullfrog duodenal mucosa.
  • Inquiry Price
6-8 weeks
Size
QTY
Crilvastatin
PMD-387, PMD387, PMD 387
T25276120551-59-9In house
Crilvastatin (PMD 387) is a novel, non-competitive hydroxymethylglutaryl coenzyme A reductase inhibitor with cholesterol-lowering activity, inhibiting cholesterol uptake in rats with hereditary hypercholesterolemia.
  • Inquiry Price
6-8 weeks
Size
QTY
Golexanolone
Golexanolonum, Golexanolona, GR-3027
T254582089238-18-4In house
Golexanolone (Golexanolona) is a novel GABA-A receptor-modulating steroid antagonist that reduces peripheral inflammation and neuroinflammation and improves cognitive and motor function in rats with chronic hyperammonemia, and may be used to study hepatic encephalopathy.
  • Inquiry Price
6-8 weeks
Size
QTY
Quinacainol
RP-54272, RP 54272, PK-10139, PK10139, PK 10139
T2601086073-85-0In house
Quinacainol (RP 54272) is a new antiarrhythmic compound with class I antiarrhythmic effects in rats.
  • Inquiry Price
6-8weeks
Size
QTY
TargetMol | Inhibitor Sale