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Search Result

Search Results for "sodium channel"

Targets

Sodium Channel

Libraries

Sodium Channel Blocker Library
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Compounds

Cat No. Product Name
T12951 Sodium Channel inhibitor 2 Sodium Channel
Sodium Channel inhibitor 2 is a blocker of sodium channel.
T12948 Sodium Channel inhibitor 1 Others
Sodium Channel inhibitor1 is a novel and selective voltage-gated sodium channel for pain treatment. (IC50 Value of 0.16 ...
T13177L Tocainide Sodium Channel
Tocainide 是口服有活性的 sodium channel 阻滞剂，阻断产生疼痛的病灶中(神经膜上)的钠通道。它是利多卡因 (lignocaine) 的伯胺类似物，可用于研究心律不齐。
T12608 QX-314 chloride Sodium Channel
QX-314 chloride 是钠离子通道永久性电荷阻滞剂，具有膜不渗透性。
T15260 Evenamide NW-3509 Sodium Channel
Evenamide 是一种口服有效的电压门控钠通道 (sodium channel, VGSC) 阻滞剂，Ki 为 0.4 µM，在精神分裂症中有研究价值。Evenamide 在精神病，躁狂症，抑郁和攻击性的各种啮齿动物模型中具有显著功效。
TQ0014 GNE-131 Sodium Channel
GNE-131 是有效的人类钠离子通道 NaV1.7(hNaV1.7)选择性抑制剂，IC50为 3 nM。
T0008 Phenytoin sodium Diphenylhydantoin Sodium,Dilantin sodium,Diphantoine,5,5-Diphenylhydantoin sodium salt,苯妥英钠 Sodium Channel , Virus Protease
Phenytoin sodium 是一种有效的电压门控钠离子通道阻滞剂，可减少小鼠乳腺肿瘤的生长和转移，具有抗癫痫活性。
T5850 Benzamil Benzamil (hydrochloride) Na+/Ca2+ Exchanger , Sodium Channel
Benzamil 是 Amiloride 类似物，是 Na+/Ca2+交换体抑制剂，抑制 TRPP3 介导的 Ca2+激活电流，IC50为 1.1 μM。它也是一种非选择性上皮钠通道 (ENaC) 阻滞剂，能增强肌源性血管收缩。
T7182 Metaflumizone BAS-320I,氰氟虫腙 Sodium Channel , Parasite
Metaflumizone 是一种缩氨基脲杀虫剂，是钠离子通道阻滞剂。
T9683 VX-150 Sodium Channel
VX-150 是一种口服有效的，高选择性的 NaV1.8抑制剂。VX-150 在各种疼痛适应症中有研究的价值。
T4539 Nicainoprol RU-42924,尼卡普醇 Sodium Channel
Nicainoprol 是一种快速钠通道阻断剂，是有效的抗心律失常剂。
T6633 Ranolazine RS 43285-003,CVT 303,Ranexa,雷诺嗪 Sodium Channel , Calcium Channel
Ranolazine 具有抗心绞痛和抗缺血的功效，通过抑制内向钠电流的后期作用 (对INa 和IKr 的IC50值分别为 6 μM 和 12 μM) 发挥作用，而不会影响心率或血压。Ranolazine 还是脂肪酸氧化 (FAO) 的部分抑...
T19644 Benzonatate Sodium Channel
Benzonatate 是外周口服镇咳药，对咳嗽延伸受体 (cough stretch receptors) 的活性具有抑制作用。它是丁卡因样代谢物，能够阻断呼吸延伸受体的钠通道并产生局部麻醉作用。
T12181 NaV1.7 inhibitor-1 Sodium Channel
NaV1.7 inhibitor-1 是有效的、选择性的电压门控钠通道 (Nav) 1.7 抑制剂，对于hNaV1.7的IC50为 0.6 nM，其选择性是 hNaV1.5 的 80 倍。
T22675 Co 102862 V 102862 Sodium Channel , Others
Co 102862 是一种电压门控钠通道阻滞剂。 Co 102862 可用于抗惊厥的研究。
T37688 Cyfluthrin Reactive Oxygen Species , Sodium Channel
Cyfluthrin 属于 II 型拟除虫菊酯，对多种昆虫都有杀灭效果。Cyfluthrin 是Nav1.8钠通道调节剂。它可应用于农业、兽医、杀虫剂、拟除虫菊酯和贮存产品等领域。
T7811 Pilsicainide HCl 盐酸吡西卡呢,SUN 1165 Sodium Channel
Pilsicainide HCl 是一种纯钠通道阻滞剂。
T23213 QX-222 chloride QX 222,Lidocaine N-Methyl Hydrochloride Sodium Channel
QX 222 chloride 是 Lignocaine 的一种三甲基类似物，是有效的 Na+通道阻滞剂。
T0440 Oxcarbazepine GP 47680,奥卡西平 Sodium Channel , Apoptosis
Oxcarbazepine 是一种钠通道阻滞剂，有效抑制胶质母细胞瘤细胞生长并诱导胶质母细胞瘤细胞凋亡或 G2/M 停滞，具有抗癌和抗惊厥作用。
T7502 PF 05089771 tosylate Sodium Channel
PF 05089771 tosylate 是口服有效的、选择性的Nav1.7丙烯酰胺抑制剂。PF 05089771 tosylate 具有用于疼痛和糖尿病神经性疾病的研究。
Sodium Channel inhibitor 2
T12951
synonym:
Target:
Sodium Channel inhibitor 1
T12948
synonym:
Target:
Tocainide
T13177L
synonym:
Target:
QX-314 chloride
T12608
synonym:
Target:
Evenamide
T15260
synonym: NW-3509
Target:
GNE-131
TQ0014
synonym:
Target:
Phenytoin sodium
T0008
synonym: Diphenylhydantoin Sodium,Dilantin sodium,Diphantoine,5,5-Diphenylhydantoin sodium salt,苯妥英钠
Target:
Benzamil
T5850
synonym: Benzamil (hydrochloride)
Target:
Metaflumizone
T7182
synonym: BAS-320I,氰氟虫腙
Target:
VX-150
T9683
synonym:
Target:
Nicainoprol
T4539
synonym: RU-42924,尼卡普醇
Target:
Ranolazine
T6633
synonym: RS 43285-003,CVT 303,Ranexa,雷诺嗪
Target:
Benzonatate
T19644
synonym:
Target:
NaV1.7 inhibitor-1
T12181
synonym:
Target:
Co 102862
T22675
synonym: V 102862
Target:
Cyfluthrin
T37688
synonym:
Target:
Pilsicainide HCl
T7811
synonym: 盐酸吡西卡呢,SUN 1165
Target:
QX-222 chloride
T23213
synonym: QX 222,Lidocaine N-Methyl Hydrochloride
Target:
Oxcarbazepine
T0440
synonym: GP 47680,奥卡西平
Target:
PF 05089771 tosylate
T7502
synonym:
Target:
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