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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 2680 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Product Description Product Description

  • A unique collection of 2680 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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Apoptosis
Autophagy
Endogenous Metabolite
5-HT Receptor
Antibacterial
Adrenergic Receptor
DNA/RNA Synthesis
Dopamine Receptor
Antibiotic
VEGFR
COX
Histamine Receptor
Potassium Channel
Calcium Channel
EGFR
Sodium Channel
Parasite
PI3K
Cytochromes P450
CDK
Reactive Oxygen Species
FLT
Glucocorticoid Receptor
PDGFR
Topoisomerase
HIV Protease
JAK
FGFR
c-Kit
HDAC
NF-κB
c-Met/HGFR
mTOR
Microtubule Associated
PPAR
Virus Protease
Ferroptosis
Prostaglandin Receptor
SARS-CoV
AChR
Src
Nucleoside Antimetabolite/Analog
Dehydrogenase
Mitophagy
Akt
GABA Receptor
Tyrosine Kinases
Bcr-Abl
Antifungal
Estrogen Receptor/ERR
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iGluR
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GPCR
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p38 MAPK
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DNA-PK
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Hydroxylase
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Leukotriene Receptor
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Smo
Phospholipase
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PAK
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Pim
IRAK
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Serine/threonin kinase
Bradykinin Receptor
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ribosome
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MT Receptor
transporter
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Melanocortin Receptor
NOD
NEDD8
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CD73
UGT
Thrombopoietin Receptor
BCRP
p97
IRE1
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OXPHOS
MLK
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
Galectin
Hexokinase
Complement System
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