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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 2680 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Product Description Product Description

  • A unique collection of 2680 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
DNA/RNA Synthesis
Antibacterial
Dopamine Receptor
Antibiotic
VEGFR
COX
Histamine Receptor
EGFR
Sodium Channel
Potassium Channel
Calcium Channel
PI3K
CDK
FLT
Cytochromes P450
Glucocorticoid Receptor
PDGFR
Parasite
Topoisomerase
HIV Protease
JAK
c-Kit
Reactive Oxygen Species
FGFR
HDAC
Microtubule Associated
mTOR
PPAR
c-Met/HGFR
Dehydrogenase
AChR
Ferroptosis
Src
NF-κB
GABA Receptor
Prostaglandin Receptor
Antifungal
Mitophagy
Nucleoside Antimetabolite/Analog
Tyrosine Kinases
SARS-CoV
Bcr-Abl
Estrogen/progestogen Receptor
Adenosine Receptor
Androgen Receptor
Estrogen Receptor/ERR
Raf
GPCR
Influenza Virus
PARP
Akt
iGluR
HSP
PDE
ALK
Aurora Kinase
Epigenetic Reader Domain
P-gp
HER
MEK
c-RET
HSV
p38 MAPK
TRP/TRPV Channel
Opioid Receptor
ROS
Serotonin Transporter
ATPase
ERK
NMDAR
Norepinephrine
RAAS
Trk receptor
DNA Alkylator/Crosslinker
Endothelin Receptor
Histone Methyltransferase
Phosphatase
PKC
Bcl-2 Family
c-Fms
GSK-3
HCV Protease
HIF/HIF Prolyl-Hydroxylase
TAM Receptor
TNF
Virus Protease
Chk
CXCR
HBV
SGLT
AMPK
E1/E2/E3 Enzyme
FAK
Guanylate cyclase
HIF
p53
Progesterone Receptor
S1P Receptor
STAT
Carbonic Anhydrase
Caspase
DNA Alkylation
DNA-PK
IL Receptor
LPL Receptor
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Retinoid Receptor
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TLR
Antifolate
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CFTR
Gamma-secretase
Interleukin
Mitochondrial Metabolism
MMP
Nrf2
P2X Receptor
Proteasome
ROS Kinase
Vasopressin Receptor
ATM/ATR
Beta Amyloid
GNRH Receptor
Hedgehog/Smoothened
HMG-CoA Reductase
IGF-1R
PLK
ROCK
Syk
TGF-beta/Smad
ADC Cytotoxin
CSF-1R
DHFR
GluR
IAP
P2Y Receptor
PKA
S6 Kinase
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Cannabinoid Receptor
DNA Methyltransferase
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BTK
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Casein Kinase
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Histone Demethylase
Lipoxygenase
Monoamine Oxidase
OX Receptor
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Smo
Bradykinin Receptor
Glucagon Receptor
Hydroxylase
IRAK
Isocitrate Dehydrogenase (IDH)
IκB/IKK
Molecular Glues
PAK
Phospholipase
Pim
CCR
DPP-4
Ephrin Receptor
GHSR
Glutathione Peroxidase
Leukotriene Receptor
NADPH
NO Synthase
Serine Protease
Thrombin
Xanthine Oxidase
ABC Transporter
AhR
Aminopeptidase
Aromatase
Aryl Hydrocarbon Receptor
CaMK
CaSR
CGRP Receptor
Chloride channel
Cholecystokinin Receptor
Cholinesterase (ChE)
CRFR
CRM1
Fatty Acid Synthase
FXR
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IDO
IFNAR
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Melatonin Receptor
Monoamine Transporter
Neuropeptide Y Receptor
PGE Synthase
PROTACs
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STING
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Wee1
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Annexin A
Decarboxylase
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MT Receptor
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NAMPT
NOD
NOS
OAT
Oxytocin Receptor
PD-1/PD-L1
PDK
PERK
Protease-activated Receptor
PYK2
Rho
ribosome
ROR
Serine/threonin kinase
Somatostatin
transporter
Tyrosinase
Acyltransferase
Amino Acids and Derivatives
Arginase
ATP Citrate Lyase
BCRP
Beta-Secretase
CD73
Cell wall
c-Myc
Discoidin Domain Receptor (DDR)
DNA gyrase
Gap Junction Protein
Glucosidase
GST
HCN Channel
Hexokinase
IRE1
LDL
Ligands for Target Protein for PROTAC
LPA Receptor
MLK
NEDD8
NOD-like Receptor (NLR)
p97
Porcupine
Reductase
Telomerase
TOPK
VDA
ACK1
Advanced Glycation End Products
Anion Exchanger
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ASK
BMI-1
Complement System
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DYRK
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Imidazoline Receptor
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Neprilysin
Neurotensin Receptor
NPC1L1
PAFR
PAI-1
PI4K
Pyroptosis
RXFP receptor
SGK
Stemness kinase
Survivin
Thioredoxin
Thyroid hormone receptor(THR)
UGT

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