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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 2760 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library

sizeIn stock

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Product Description Product Description

  • A unique collection of 2760 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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Apoptosis
Autophagy
Endogenous Metabolite
5-HT Receptor
Antibacterial
Adrenergic Receptor
DNA/RNA Synthesis
Dopamine Receptor
Antibiotic
VEGFR
COX
Potassium Channel
Calcium Channel
Histamine Receptor
Sodium Channel
EGFR
Parasite
PI3K
ROS
CDK
Cytochromes P450
Reactive Oxygen Species
NF-κB
FLT
JAK
PDGFR
Glucocorticoid Receptor
HIV Protease
FGFR
Topoisomerase
mTOR
c-Kit
HDAC
Akt
c-Met/HGFR
Microtubule Associated
PPAR
Virus Protease
Ferroptosis
AChR
Prostaglandin Receptor
SARS-CoV
Src
p38 MAPK
Dehydrogenase
Nucleoside Antimetabolite/Analog
GABA Receptor
Estrogen Receptor/ERR
Antifungal
Mitophagy
ERK
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Adenosine Receptor
Tyrosine Kinases
Bcr-Abl
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Caspase
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TNF
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PARP
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ALK
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HER
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RAAS
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Opioid Receptor
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AMPK
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MMP
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Leukotriene Receptor
Antifection
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OX Receptor
Sirtuin
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IκB/IKK
Cannabinoid Receptor
DNA Methyltransferase
IRAK
RIP kinase
Smo
DNA
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Phospholipase
Hydroxylase
Neurokinin receptor
Sigma receptor
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glycosidase
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MT Receptor
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transporter
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ribosome
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Gap Junction Protein
Protease-activated Receptor
MLK
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Ligands for Target Protein for PROTAC
Arginase
DYRK
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TOPK
VDA
Galectin
Cysteine Protease
RANKL/RANK
UGT
LDL
GRK
DNA gyrase
Hexokinase
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HCN Channel
Thrombopoietin Receptor
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PAI-1
LPA Receptor
PI4K
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p97
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BMI-1
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Drug-Linker Conjugates for ADC
PGC-1α

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