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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 2680 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Product Description Product Description

  • A unique collection of 2680 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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Apoptosis
Autophagy
Endogenous Metabolite
5-HT Receptor
Antibacterial
Adrenergic Receptor
DNA/RNA Synthesis
Dopamine Receptor
Antibiotic
VEGFR
COX
Histamine Receptor
Potassium Channel
Calcium Channel
EGFR
Sodium Channel
Parasite
PI3K
Cytochromes P450
CDK
Reactive Oxygen Species
FLT
HIV Protease
Glucocorticoid Receptor
Topoisomerase
PDGFR
JAK
FGFR
c-Kit
NF-κB
HDAC
c-Met/HGFR
mTOR
Microtubule Associated
PPAR
Virus Protease
Ferroptosis
AChR
Prostaglandin Receptor
SARS-CoV
Src
Dehydrogenase
Nucleoside Antimetabolite/Analog
Mitophagy
Akt
GABA Receptor
Tyrosine Kinases
Antifungal
Bcr-Abl
Estrogen Receptor/ERR
Estrogen/progestogen Receptor
iGluR
Influenza Virus
GPCR
Adenosine Receptor
Raf
Androgen Receptor
p38 MAPK
PARP
HSP
Caspase
Epigenetic Reader Domain
Bcl-2 Family
Ras
PDE
Interleukin
ERK
HSV
Aurora Kinase
TNF
Serotonin Transporter
P-gp
ALK
TRP/TRPV Channel
MEK
HIF/HIF Prolyl-Hydroxylase
HER
ATPase
c-RET
HBV
PKC
ROS
Opioid Receptor
c-Fms
MDM-2/p53
RAAS
Phosphatase
NMDAR
Norepinephrine
Trk receptor
Histone Methyltransferase
HCV Protease
DNA Alkylator/Crosslinker
Endothelin Receptor
STAT
Proton pump
E1/E2/E3 Enzyme
Mitochondrial Metabolism
MMP
AMPK
TAM Receptor
ROS Kinase
LPL Receptor
GSK-3
Chk
Retinoid Receptor
FAK
Progesterone Receptor
Gamma-secretase
Guanylate cyclase
CXCR
IGF-1R
SGLT
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HIF
p53
S1P Receptor
Carbonic Anhydrase
DNA-PK
JNK
Molecular Glues
DNA Alkylation
IL Receptor
TLR
Beta Amyloid
CFTR
Proteasome
Antioxidant
PKA
Antifolate
ROCK
Drug Metabolite
P2X Receptor
Vasopressin Receptor
GluR
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Nrf2
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S6 Kinase
ADC Cytotoxin
Transferase
GNRH Receptor
Wnt/beta-catenin
Hedgehog/Smoothened
PLK
Syk
HMG-CoA Reductase
DHFR
P2Y Receptor
CSF-1R
IAP
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Lipoxygenase
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NO Synthase
Kinesin
Monoamine Oxidase
Mdm2
Integrin
MRP
MAO
IDO
BTK
Antifection
OX Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Sirtuin
Casein Kinase
IκB/IKK
Ligand for E3 Ligase
Cannabinoid Receptor
Neurokinin receptor
DNA Methyltransferase
Histone Demethylase
Serine Protease
Leukotriene Receptor
RIP kinase
Smo
PAK
DNA
Antiviral
Phospholipase
Hydroxylase
Sigma receptor
Tie-2
Pim
Glucagon Receptor
Angiotensin-converting Enzyme (ACE)
MAPK
Ephrin Receptor
IRAK
IKZF
Reductase
NADPH
Glutathione Peroxidase
Serine/threonin kinase
FXR
DPP-4
CCR
Bradykinin Receptor
Cholinesterase (ChE)
Xanthine Oxidase
Telomerase
GHSR
Thrombin
NOD-like Receptor (NLR)
PD-1/PD-L1
Chloride channel
PROTACs
CRM1
YAP
IFNAR
PERK
Melatonin Receptor
c-Myc
CaSR
Cholecystokinin Receptor
Photosensitizer
PYK2
Glutaminase
Aryl Hydrocarbon Receptor
ABC Transporter
Na-K-Cl cotransporter
Glucosidase
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Neuropeptide Y Receptor
CaMK
Wee1
PGE Synthase
STING
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GPCR19
CRFR
RSV
GST
Aromatase
CGRP Receptor
AhR
NOS
ROR
LTR
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NAMPT
Annexin A
MT Receptor
Somatostatin
KSP
DUB
ATP Citrate Lyase
Beta-Secretase
OAT
Free radical scavengers
transporter
Decarboxylase
FKBP
ribosome
Melanocortin Receptor
PDK
Oxytocin Receptor
Adenosine Deaminase
Cuproptosis
Discoidin Domain Receptor (DDR)
NOD
Tyrosinase
Protease-activated Receptor
NEDD8
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
Arginase
Cell wall
TOPK
VDA
Galectin
Cysteine Protease
IRE1
UGT
LDL
DNA gyrase
Hexokinase
HCN Channel
Thrombopoietin Receptor
OXPHOS
BCRP
Acyltransferase
Porcupine
CD73
Histone Acetyltransferase
LPA Receptor
SGK
Complement System
Gap Junction Protein
p97
MLK
Thyroid hormone receptor(THR)
Advanced Glycation End Products
MicroRNA
NPC1L1
Monocarboxylate transporter
Hydrogenase
RAR/RXR
MALT
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DYRK
Necroptosis
MIF
GTPase
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OCT
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Hck
Liver X Receptor
LIM Kinase
Neurotensin Receptor
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ASK
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PI4K
KLF
Aquaporin
RXFP receptor
NADPH-oxidase
BMI-1
Imidazoline Receptor
Vitamin
PGC-1α

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