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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 2680 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 2680 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
DNA/RNA Synthesis
Antibacterial
Dopamine Receptor
Antibiotic
Histamine Receptor
VEGFR
COX
EGFR
Sodium Channel
PI3K
Calcium Channel
Potassium Channel
CDK
FLT
Glucocorticoid Receptor
Cytochromes P450
PDGFR
Parasite
Topoisomerase
Reactive Oxygen Species
JAK
HIV Protease
c-Kit
HDAC
FGFR
Microtubule Associated
c-Met/HGFR
PPAR
mTOR
Dehydrogenase
AChR
Src
Ferroptosis
Prostaglandin Receptor
NF-κB
GABA Receptor
Antifungal
Mitophagy
Tyrosine Kinases
Nucleoside Antimetabolite/Analog
SARS-CoV
Androgen Receptor
Estrogen/progestogen Receptor
Adenosine Receptor
Estrogen Receptor/ERR
Bcr-Abl
Raf
GPR
HER
PARP
Influenza Virus
Akt
iGluR
PDE
Aurora Kinase
HSP
Epigenetic Reader Domain
ALK
P-gp
MEK
p38 MAPK
Serotonin Transporter
TRP/TRPV Channel
Opioid Receptor
HSV
Norepinephrine
c-RET
RAAS
ROS
ATPase
ERK
Trk receptor
DNA Alkylator/Crosslinker
Phosphatase
HBV
PKC
NMDAR
Endothelin Receptor
Bcl-2 Family
Histone Methyltransferase
HCV Protease
Virus Protease
GSK-3
c-Fms
TNF
TAM Receptor
HIF/HIF Prolyl-Hydroxylase
Proton pump
CXCR
Chk
DNA-PK
Progesterone Receptor
E1/E2/E3 Enzyme
Guanylate cyclase
SGLT
Retinoid Receptor
STAT
AMPK
HIF
FAK
S1P Receptor
Carbonic Anhydrase
LPL Receptor
Caspase
DNA Alkylation
IL Receptor
Vasopressin Receptor
MMP
TLR
Reverse Transcriptase
p53
Antioxidant
Antifolate
Gamma-secretase
P2X Receptor
Mitochondrial Metabolism
Interleukin
Nrf2
ROS Kinase
CFTR
Proteasome
GNRH Receptor
Hedgehog/Smoothened
IGF-1R
TGF-beta/Smad
ATM/ATR
Beta Amyloid
PLK
Syk
ADC Cytotoxin
Mdm2
Transferase
DHFR
P2Y Receptor
PKA
ROCK
IAP
CSF-1R
GluR
S6 Kinase
Integrin
JNK
MRP
Wnt/beta-catenin
MAO
Drug Metabolite
Antifection
Lipoxygenase
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Ligand for E3 Ligase
Neurokinin receptor
DNA Methyltransferase
HMG-CoA Reductase
Kinesin
BTK
RIP kinase
Smo
OX Receptor
DNA
Antiviral
Sirtuin
Casein Kinase
Cannabinoid Receptor
Sigma receptor
Monoamine Oxidase
Histone Demethylase
Pim
Glucagon Receptor
Molecular Glues
Isocitrate Dehydrogenase (IDH)
PAK
Bradykinin Receptor
IκB/IKK
Phospholipase
Hydroxylase
IRAK
NADPH
Glutathione Peroxidase
Serine Protease
Leukotriene Receptor
DPP-4
CCR
Cholinesterase (ChE)
Xanthine Oxidase
Ephrin Receptor
GHSR
Thrombin
NO Synthase
Chloride channel
PROTACs
CRM1
YAP
IFNAR
Tie-2
Melatonin Receptor
CaSR
Cholecystokinin Receptor
FXR
Aryl Hydrocarbon Receptor
IDO
ABC Transporter
Monoamine Transporter
Neuropeptide Y Receptor
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CaMK
Wee1
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STING
Aminopeptidase
GPCR19
CRFR
RSV
Kras
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CGRP Receptor
Ras
AhR
NOS
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Serine/threonin kinase
NAMPT
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MT Receptor
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Somatostatin
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MAPK
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transporter
Decarboxylase
ribosome
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PDK
Adenosine Deaminase
Tyrosinase
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PD-1/PD-L1
NEDD8
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
Arginase
Reductase
Cell wall
PERK
VDA
c-Myc
Kisspeptin
Liver X Receptor
Cysteine Protease
IRE1
LDL
DNA gyrase
Glucosidase
Hexokinase
HCN Channel
Telomerase
ATP Citrate Lyase
BCRP
Beta-Secretase
Acyltransferase
Porcupine
CD73
GST
LPA Receptor
Oxytocin Receptor
Discoidin Domain Receptor (DDR)
Gap Junction Protein
p97
NOD-like Receptor (NLR)
MLK
Advanced Glycation End Products
MicroRNA
NPC1L1
Monocarboxylate transporter
Hydrogenase
RAR/RXR
MALT
DYRK
TOPK
GTPase
Galectin
N-Acetylglucosaminyltransferase
Hck
Neurotensin Receptor
Glucokinase
Stemness kinase
Myosin
UGT
PAFR
MTH1
GRK
GlyT
Anion Exchanger
Thioredoxin
ACK1
Survivin
MNK
Histone Acetyltransferase
ASK
GluCls
PAI-1
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Neprilysin
Hippo pathway
PI4K
KLF
Aquaporin
RXFP receptor
SGK
Complement System
NADPH-oxidase
BMI-1
NOD
Imidazoline Receptor

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