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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 2680 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 2680 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Autophagy
Apoptosis
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
DNA/RNA Synthesis
Antibacterial
Dopamine Receptor
Antibiotic
Histamine Receptor
VEGFR
COX
EGFR
Sodium Channel
PI3K
Calcium Channel
Potassium Channel
CDK
FLT
Cytochromes P450
Glucocorticoid Receptor
PDGFR
Topoisomerase
Parasite
Reactive Oxygen Species
JAK
HIV Protease
c-Kit
HDAC
FGFR
Microtubule Associated
c-Met/HGFR
mTOR
PPAR
Dehydrogenase
AChR
Ferroptosis
NF-κB
Prostaglandin Receptor
Src
GABA Receptor
Antifungal
Mitophagy
SARS-CoV
Tyrosine Kinases
Nucleoside Antimetabolite/Analog
Estrogen/progestogen Receptor
Androgen Receptor
Estrogen Receptor/ERR
Adenosine Receptor
Bcr-Abl
GPR
HER
Raf
Influenza Virus
PARP
Akt
iGluR
PDE
Aurora Kinase
HSP
ALK
Epigenetic Reader Domain
MEK
c-RET
HSV
p38 MAPK
P-gp
TRP/TRPV Channel
Norepinephrine
Opioid Receptor
RAAS
ROS
Serotonin Transporter
ATPase
ERK
NMDAR
Trk receptor
DNA Alkylator/Crosslinker
Endothelin Receptor
HBV
Phosphatase
PKC
Bcl-2 Family
c-Fms
GSK-3
HCV Protease
HIF/HIF Prolyl-Hydroxylase
Histone Methyltransferase
TAM Receptor
TNF
Virus Protease
Chk
CXCR
Proton pump
SGLT
AMPK
DNA-PK
E1/E2/E3 Enzyme
FAK
Guanylate cyclase
HIF
Progesterone Receptor
Retinoid Receptor
S1P Receptor
STAT
Carbonic Anhydrase
Caspase
DNA Alkylation
IL Receptor
LPL Receptor
MMP
p53
Reverse Transcriptase
TLR
Vasopressin Receptor
Antifolate
Antioxidant
CFTR
Interleukin
Mitochondrial Metabolism
Nrf2
P2X Receptor
Proteasome
ROS Kinase
ATM/ATR
GNRH Receptor
Hedgehog/Smoothened
HMG-CoA Reductase
IGF-1R
PLK
Syk
TGF-beta/Smad
ADC Cytotoxin
Beta Amyloid
CSF-1R
DHFR
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GluR
IAP
P2Y Receptor
PKA
ROCK
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Transferase
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Cannabinoid Receptor
DNA Methyltransferase
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Indoleamine 2,3-Dioxygenase (IDO)
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Casein Kinase
DNA
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Monoamine Oxidase
OX Receptor
RIP kinase
Sigma receptor
Sirtuin
Smo
Bradykinin Receptor
Glucagon Receptor
Hydroxylase
IRAK
Isocitrate Dehydrogenase (IDH)
IκB/IKK
Molecular Glues
PAK
Phospholipase
Pim
CCR
Cholinesterase (ChE)
DPP-4
Ephrin Receptor
GHSR
Glutathione Peroxidase
NADPH
NO Synthase
Serine Protease
Thrombin
Xanthine Oxidase
ABC Transporter
AhR
Aminopeptidase
Aromatase
Aryl Hydrocarbon Receptor
CaMK
CaSR
CGRP Receptor
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Cholecystokinin Receptor
CRFR
CRM1
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STING
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ribosome
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transporter
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BCRP
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CD73
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c-Myc
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DNA gyrase
Gap Junction Protein
Glucosidase
GST
HCN Channel
Hexokinase
IRE1
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LDL
Ligands for Target Protein for PROTAC
LPA Receptor
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NOD-like Receptor (NLR)
NOS
p97
PERK
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Reductase
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VDA
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ASK
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Complement System
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MALT
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MTH1
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NADPH-oxidase
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Neurotensin Receptor
NPC1L1
PAFR
PAI-1
PI4K
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RAR/RXR
RXFP receptor
SGK
Stemness kinase
Survivin
Thioredoxin
TOPK
UGT

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