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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 2680 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 2680 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Autophagy
Apoptosis
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
DNA/RNA Synthesis
Antibacterial
Dopamine Receptor
Antibiotic
VEGFR
Histamine Receptor
COX
EGFR
Sodium Channel
Potassium Channel
Calcium Channel
PI3K
CDK
FLT
Cytochromes P450
Glucocorticoid Receptor
PDGFR
Topoisomerase
Parasite
HIV Protease
JAK
Reactive Oxygen Species
c-Kit
HDAC
FGFR
Microtubule Associated
c-Met/HGFR
PPAR
mTOR
Dehydrogenase
Src
Ferroptosis
AChR
Prostaglandin Receptor
NF-κB
GABA Receptor
Mitophagy
Tyrosine Kinases
Antifungal
SARS-CoV
Estrogen/progestogen Receptor
Nucleoside Antimetabolite/Analog
Bcr-Abl
Estrogen Receptor/ERR
GPCR
Adenosine Receptor
Raf
Androgen Receptor
PARP
Influenza Virus
Akt
iGluR
PDE
Aurora Kinase
HSP
Epigenetic Reader Domain
ALK
P-gp
MEK
HER
p38 MAPK
TRP/TRPV Channel
HSV
c-RET
Serotonin Transporter
ROS
Opioid Receptor
Norepinephrine
ATPase
RAAS
ERK
NMDAR
Trk receptor
Histone Methyltransferase
DNA Alkylator/Crosslinker
Phosphatase
HBV
PKC
Endothelin Receptor
GSK-3
Virus Protease
Bcl-2 Family
c-Fms
TNF
TAM Receptor
HIF/HIF Prolyl-Hydroxylase
Proton pump
HCV Protease
CXCR
Chk
SGLT
DNA-PK
Progesterone Receptor
E1/E2/E3 Enzyme
Guanylate cyclase
STAT
AMPK
HIF
FAK
S1P Receptor
Carbonic Anhydrase
LPL Receptor
Caspase
DNA Alkylation
IL Receptor
MMP
TLR
Reverse Transcriptase
Retinoid Receptor
p53
Proteasome
Antioxidant
Antifolate
Gamma-secretase
P2X Receptor
Mitochondrial Metabolism
Vasopressin Receptor
Interleukin
ROS Kinase
CFTR
GNRH Receptor
PKA
ROCK
Hedgehog/Smoothened
IGF-1R
TGF-beta/Smad
Nrf2
ATM/ATR
Beta Amyloid
PLK
Syk
HMG-CoA Reductase
ADC Cytotoxin
Transferase
DHFR
P2Y Receptor
IAP
CSF-1R
GluR
S6 Kinase
Mdm2
Integrin
JNK
MRP
Wnt/beta-catenin
MAO
Antifection
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Ligand for E3 Ligase
Cannabinoid Receptor
Neurokinin receptor
DNA Methyltransferase
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BTK
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OX Receptor
Lipoxygenase
DNA
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Sigma receptor
Monoamine Oxidase
Pim
Glucagon Receptor
Molecular Glues
Isocitrate Dehydrogenase (IDH)
PAK
Bradykinin Receptor
IκB/IKK
Phospholipase
Hydroxylase
IRAK
NADPH
Glutathione Peroxidase
Serine Protease
Leukotriene Receptor
DPP-4
CCR
Cholinesterase (ChE)
Xanthine Oxidase
Ephrin Receptor
GHSR
Thrombin
NO Synthase
Chloride channel
PROTACs
CRM1
YAP
IFNAR
Tie-2
Melatonin Receptor
CaSR
Cholecystokinin Receptor
FXR
Aryl Hydrocarbon Receptor
IDO
ABC Transporter
Monoamine Transporter
Neuropeptide Y Receptor
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CaMK
Wee1
PGE Synthase
STING
GPCR19
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CRFR
RSV
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CGRP Receptor
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AhR
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MT Receptor
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transporter
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ribosome
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Oxytocin Receptor
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Arginase
Reductase
Cell wall
TOPK
VDA
c-Myc
Cysteine Protease
IRE1
LDL
DNA gyrase
Glucosidase
Hexokinase
HCN Channel
Telomerase
ATP Citrate Lyase
BCRP
Beta-Secretase
Acyltransferase
Porcupine
CD73
GST
LPA Receptor
Discoidin Domain Receptor (DDR)
Gap Junction Protein
NOD
p97
NOD-like Receptor (NLR)
MLK
Advanced Glycation End Products
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NPC1L1
Hydrogenase
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Hck
Liver X Receptor
Neurotensin Receptor
LIM Kinase
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Myosin
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PAFR
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GRK
GlyT
Anion Exchanger
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ACK1
MNK
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ASK
GluCls
PAI-1
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Neprilysin
Hippo pathway
KLF
PI4K
Aquaporin
RXFP receptor
SGK
Complement System
NADPH-oxidase
BMI-1
Imidazoline Receptor

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