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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP1216 | CaM kinase II inhibitor TFA salt | Autocamtide-2-related inhibitory peptide (TFA) | CaMK |
CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM. | |||
T76690 | Mavrilimumab | CAM 3001 | Virus Protease , CSF-1R |
Mavrilimumab (CAM 3001) is a monoclonal antibody with antiviral activity that has an affinity for the α subunit of the granulocytic-macrophage colony-stimulating factor (GM-CSF) receptor and blocks downstream intracellul... | |||
T70136 | CAM 4750 | ||
CAM 4750 is a nonpeptide tachykinin NK1 receptor antagonist. | |||
T41211 | CAM 833 | ||
CAM 833 is an effective positivity inhibitor, which can inhibit the interaction between BRCA2 and RAD51. The Kd of ChimRAD51 protein is 366 nM. CAM 833 inhibited the oligocoagulation of RAD51 and promoted the process of ... | |||
T70410 | Cam 2445 | ||
Cam 2445 is a nonpeptide, alpha-methyltryptophan derivative; an NK1 neurokinin receptor antagonist that is a potentially useful treatment for arthritis, asthma, migraine, anxiety, psychosis, and emesis. | |||
T70137 | CAM 4515 | ||
CAM 4515 is a nonpeptide tachykinin NK1 receptor antagonist. | |||
T28331 | PD 136450 | Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189 | |
Cholecystokinin type B receptor antagonist PD-136,450 is a partial secretory agonist in the stomach and a full agonist in the pancreas of the rat. Gastrin (cholecystokinin type B (CCK-B)) receptor antagonists may help to... | |||
T30442 | Bialamicol Hydrochloride | Camoform hydrochloride,CAM 807,CAM-807,CI 301 | |
Bialomicol Hydrochloride is a bio-active chemical. | |||
T41184 | Clocinnamox mesylate | C-CAM,NIH 10443 | |
Clocinnamox mesylate is a systemically active, irreversibleμ-opioid receptor antagonist (apparent Kivalues are 0.7, 1.9 and 5.7 nM for mouseμ,δandκreceptors respectively). | |||
T16366 | NVR 3-778 | HBV | |
NVR 3-778 is a first-in-Class and oral bioavailable HBV CAM belonging to the SBA class It has anti-HBV activity. | |||
T70211 | CAM741 | ||
CAM741 is a novel selective inhibitor of vascular cell adhesion molecule 1 (VCAM1) synthesis in endothelial cells, blocking the process of cotranslational translocation, which is dependent on the signal peptide of VCAM1. | |||
T69908 | Pidnarulex HCl | ||
Pidnarulex HCl is the salt form of CX-5461, a first-in-class non-genotoxic small molecule targeted inhibitor of RNA polymerase I (Pol I) that activates the p53 pathway without causing DNA damage. CX-5461 selectively inhi... | |||
T69909 | CAM4066 | ||
CAM4066 is a novel potent and selective CK2alpha inhibitor. | |||
TN1008 | Psoralenoside | CaMK , Calcium Channel , Histamine Receptor | |
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activity, antitumor effects and antibacterial activity. | |||
T70210 | FT-1101 free base | ||
FT-1101 is an orally bioavailable, potent and selective BET inhibitor. FT-1101 binds to the acetylated lysine recognition motifs in the bromodomain sites of BET proteins, thereby preventing the interaction between the B... | |||
T8846 | Beta-Escin | B-escin,AESCINE | Immunology/Inflammation related |
beta-Escin is a natural mixture of triterpenoid saponins isolated from horse chestnut (Aesculus hippocastanum) seeds, can be used as a vasoprotective anti-inflammatory, anti-edematous and anti-nociceptive agent. | |||
T70135 | Nepaprazole sodium dihydrate | ||
Nepaprazole sodium dihydrate is a proton pump inhibitor potentially for treatment of gastric ulcers. | |||
T70409 | 6alpha-Fluorotestosterone | ||
6alpha-Fluorotestosterone is a synthetic nonaromatizable androgen analog of testosterone. It binds to and activates specific nuclear receptors inhibits and is equipotent to testosterone. | |||
T23525 | W-9 hydrochloride | N-(6-aminohexyl)-5-chloronaphthalene-2-sulfonamide hydrochloride | CaMK |
W-9 hydrochloride is a calmodulin antagonist. | |||
T20792 | W-7 hydrochloride | W 7 HCl,W7 HCl,W-7 HCl | CaMK , Apoptosis , Myosin , PDE |
W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochloride induces apoptosis and has antitumor activity. |