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  • Cytochromes P450
    (8)
  • Cytochromes P450
    (6)
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    (2)
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Results for "

p-450

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    44
    TargetMol | Inhibitors_Agonists
  • Peptide Products
    1
    TargetMol | Peptide_Products
  • Dye Reagents
    3
    TargetMol | Dye_Reagents
  • Natural Products
    10
    TargetMol | Natural_Products
  • Recombinant Protein
    13
    TargetMol | Recombinant_Protein
  • Isotope Products
    2
    TargetMol | Isotope_Products
  • Antibody Products
    4
    TargetMol | Antibody_Products
Fadrozole hydrochloride
CGS 16949A
T7556102676-31-3
Fadrozole hydrochloride (CGS 16949A) is a model aromatase inhibitor that effectively suppresses estrogen production in fish ovaries.
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VP-4509
T643152190144-51-3
VP-4509 is an anti-methicillin-resistant Staphylococcus aureus (MRSA) agent (MIC: 49.3 μM). VP-4509 exhibits high antibacterial activity against the gram-negative bacterium Pseudomonas aeruginosa (ATCC9027).
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6-8 weeks
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Ginsenoside Rd
Sanchinoside Rd, Panaxoside Rd, Gypenoside VIII
T287852705-93-8
Ginsenoside Rd (Gypenoside VIII) may have properties that inhibit or prevent the growth of tumors.
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gsk-25
GSK25
T4488874119-56-9
GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and p70S6K (RSK1 IC50 of 398 nM, p70S6K IC50 of 1000nM), and a dramatically improved P450 profile (>2.2 uM at all isozymes tested).
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BVT948
T1484139674-97-0
BVT948 is a protein tyrosine phosphatase (PTP) inhibitor that also inhibits lysine methyltransferase SETD8 (KMT5A) and various cytochrome P450 (P450) isoforms.
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norfluoxetine hydrochloride
Norfluoxetine HCl
T2102957226-68-3
Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.
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Rhapontigenin 3'-O-glucoside
T410994356-22-6
Rhapontigenin 3'-O-glucoside is a derivative of Rhapontigenin, a P450 1A1 inhibitor, which may be used to prevent cancer.
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β-Amyrin
beta-Amyrin
TN1027559-70-6
β-Amyrin (beta-Amyrin) has antiviral, hepatoprotective, antinociceptive, anti-inflammatory
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α-Viniferin
ALPHA-VINIFERIN
TN137862218-13-7
α-Viniferin known as 2-arylbenzofuran flavonoids, that are inhibitors of prostaglandin H2 synthetase. α-Viniferin has anti-Alzheimer's disease, anti-tuberculosis, anti-tumor, anti-inflammation, anti-diabetes and other pharmacological activitie
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7-10 days
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Glabrol
TN169159870-65-4
5-Methylcytosine is a methylated nucleotide base found in eukaryotic DNA. It is an epigenetic modification formed by the action of DNA methyltransferases.
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Lasiodin
Lasiokaurin
TN185428957-08-6
Lasiodin (Lasiokaurin) is a diterpene compound from the plant Camellia sinensis that inhibits the proliferation of NPC cells. Lasiodin has antioxidant, antitumor and antibacterial activities, induces cell cycle length and apoptosis, induces cell migration and invasion, and can be used in the study of nasopharyngeal carcinoma.
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Retrorsine
TN2147480-54-6
Retrorsine selectively inhibits hepatocyte proliferation and following liver injury evokes small hepatocyte-like progenitor cells. Retrorsine can be used for the research of hepatocellular injury.
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7-10 days
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Voriconazole
UK-109496
T0120137234-62-9
Voriconazole (UK-109496) is a triazole antifungal agent that specifically inhibits STEROL 14-ALPHA-DEMETHYLASE and CYTOCHROME P-450 [CYP3A].
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Itraconazole
R51211
T101184625-61-6
Itraconazole (R51211) is a triazole antifungal agent that inhibits cytochrome P-450-dependent enzymes necessary for ERGOSTEROL synthesis.
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Tegafur
Fluorafur, FT-207, NSC 148958, FT 207
T137817902-23-7
Tegafur (FT 207) is a congener of the antimetabolite fluorouracil with antineoplastic activity. Tegafur is a prodrug that is gradually converted to fluorouracil in the liver by the cytochrome P-450 enzyme.
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Diniconazole
Rac-diniconazole
T595283657-24-3
Diniconazole (Rac-diniconazole) is a fungicide. It is known as a plant hormone abscisic acid (ABA) catabolic inhibitor, and acts as a potent competitive inhibitor of recombinant Arabidopsis ABA 8'-hydroxylase, CYP707A3.
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Sulconazole mononitrate
Exelderm, Sulconazole Nitrate, RS 44872
T668661318-91-0
Sulconazole mononitrate (Exelderm) is the nitrate salt form of sulconazole, a synthetic imidazole derivative with the antifungal property. Sulconazole mononitrate inhibits fungal cytochrome P-450 sterol C-14 alpha-demethylation, resulting in the accumulation of fungal 14 alpha-methyl sterols and inhibition of the synthesis of ergosterol, an important component of the fungal cell membrane. Inhibition of ergosterol synthesis leads to a disruption of cell membrane permeability, and ultimately inhibition of cell wall synthesis. In addition, Sulconazole mononitrate seems to interfere with the autolytic degradation of fungal DNA and RNA.
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Zoxazolamine
NSC 24995, Contrazole
T092261-80-3
Zoxazolamine (NSC-24995) is a uricosuric and muscle relaxant. Zoxazolamine acts centrally as a muscle relaxant, but the mechanism of its action is not understood.
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Proadifen hydrochloride
U-5446, RP-5171, SKF-525A
T159762-68-0
Proadifen hydrochloride (RP-5171) is an inhibitor of drug metabolism and cytochrome P-450 enzyme system activity.
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LY 43578
LY-43578, LY43578
T2791826766-35-8
LY 43578 is an orally active aromatase inhibitor. LY43578 could inhibit O-demethylation of P-450-dependent p-nitroanisole and N-demethylation of ethylmorphine (IC50 of 0.3 and 5 μm, respectively) in rat liver microsomes. LY 43578 can be used to study neurological and cardiovascular diseases.
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6-8 weeks
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RPR132595A
NPC
T19553185304-42-1
RPR132595A is an active CPT-11 metabolite, it is generated by cytochrome P-450 3A4 (CYP3A4).
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4-6 weeks
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Octachlorodibenzo-p-dioxin
OCDD
T2033133268-87-9
Octachlorodibenzo-p-dioxin (OCDD) is an environmental contaminant with no acute toxicity when administered. In rats, the systemic elimination half-life of Octachlorodibenzo-p-dioxin (50 μg kg intravenously or 50-5000 μg kg orally) is 3-5 months. It can accumulate and concentrate in the liver and adipose tissue after low-dose, repeated exposure. Repeated dosing of Octachlorodibenzo-p-dioxin leads to increased activity of 7-ethoxyresorufin-O-deethylase (7-EROD) and elevated total cytochrome P-450 levels.
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Cytochrome P450 2C9
S-Mephenytoin 4-hydroxylase, Human cytochrome P450 2C9, Cytochrome P 450 2C9, Cyp2C9
T25283329978-01-0
Cytochrome P450 2C9 is a cytochrome P-450 subtype that possesses specificity for acidic xenobiotics. It oxidizes a wide range of important clinical drugs under the categories of nonsteroidal anti-inflammatory agents, anticoagulants, hypoglycemic agents, a
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    Lab 170250F
    Lab-170250F,Lab170250F
    T2559188630-25-5
    Lab 170250F is a potent cytochrome P-450-obtusifoliol-14-demethylase inhibitor.
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    6-8 weeks
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