20
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T0517 | Pancreatin | Pancreatic enzymes,pancrelipase | Others |
Pancreatin (pancrelipase) is a mixture of several digestive enzymes secreted by the exocrine cells of the pancreas. It is composed of amylase, lipase and protease. | |||
T21508 | Anhydrotetracycline hydrochloride | Antibacterial , Antibiotic | |
Anhydrotetracycline (hydrochloride) is a potent competitive inhibitor of broad-spectrum tetracycline destructase enzymes. | |||
T60050 | ANT3310 | Antibacterial | |
ANT3310 is an inhibitor of broad-spectrum covalent Serine β-Lactamase with IC50s ranging from 1 nM to 175 nM for AmpC, CTX-M-15, TEM-1, OXA-48, OXA-23, and KPC-2. ANT3310 can be used in studies about bacterial infection. | |||
T7086 | Tris(benzyltriazolylmethyl)amine | TBTA | Others |
Tris(benzyltriazolylmethyl)amine (TBTA) is a tertiary amine with three 1, 2, 3-triazole groups. It complexes with, and stabilizes, copper(I) to accelerate azide-alkyne cycloadditions, as used in click chemistry. | |||
T23801 | WCK-4234 sodium | WCK-4234,WCK4234,WCK 4234 | Antibacterial |
WCK-4234 sodium (WCK 4234) is an inhibitor of β-lactamase can be used in studies targeting MDR infections. WCK-4234 sodium inhibits class A, C, and D β-lactamases and OXA carbapenemases. | |||
T2761 | Naringin dihydrochalcone | Naringin DC | P450 , NF-κB |
Naringin dihydrochalcone (Naringin DC) is an inhibitor of CYP enzymes, used as an artificial sweetener. | |||
T4174 | NSC 191412 | Others | |
NSC 191412 interacts with a variety of enzymes and receptors, including acetylcholinesterase and receptors for the neurotransmitter dopamine, and is an agonist or activator of these enzymes and receptors. | |||
T60040 | α-Cyclopentyl-4-(2-quinolinylmethoxy)benzeneacetic acid | Others , Aminopeptidase | |
α-Cyclopentyl-4-(2-quinolinylmethoxy)benzeneacetic acid was identified as possible dual inhibitors for hLTA4H and hLTC4S enzymes by the computer-aided methodology. | |||
T9679 | N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)pyrazine-2-carboxamide | Antibacterial | |
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)pyrazine-2-carboxamide exhibit an inhibitory effect on bacterial DNA helicases, nucleases, or helicase-nuclease enzyme complexes, such as, for example, one or more enzym... | |||
T21634 | N-Oxalylglycine | Oxalylglycine | Others |
N-Oxalylglycine (Oxalylglycine) is a cell permeable inhibitor of α-ketoglutarate-dependent enzymes. | |||
T0325 | Diperodon hydrochloride | Diothane hydrochloride,Proctodon,Diperocaine | Others |
Diperodon hydrochloride (Diperocaine) is a local anesthetic that can be broken down by serolytic enzymes to produce local anesthetic effects. | |||
T3215 | JNJ-42165279 | JNJ42165279 | FAAH , Autophagy |
JNJ-42165279 covalently inactivates the FAAH enzyme but is highly selective with regard to other enzymes, ion channels, transporters, and receptors. JNJ-42165279 (10 μM) exhibits high selectivity against a panel of 50 re... | |||
T6S0078 | Oxypeucedanin hydrate | Prangolarin Hydrate | Antioxidant |
1. Oxypeucedanin hydrate (Prangolarin Hydrate) has antioxidant activity. 2. Oxypeucedanin hydrate is an antimutagenic agent. 3. Oxypeucedanin hydrate exhibits carbohydrate metabolizing enzymes inhibitory effect. | |||
T6S1652 | Benzoylpaeoniflorin | COX | |
1. Benzoylpaeoniflorin is active against cyclooxygenase-1 and cyclooxygenase-2 enzymes. | |||
T11994 | Melagatran | Thrombin | |
Melagatran, a direct and orally active thrombin inhibitor, specifically inhibits thrombin without affecting other enzymes in the coagulation cascade or fibrinolytic enzymes. It does not rely on endogenous co-factors to e... | |||
T34076 | Piprozolin | W3699,W-3699,W 3699 | |
Piprozolin (W 3699) is a new type of choleretic acid that shows slight analgesic properties at high doses during chronic experiments.Piprozolin has a slight induction of certain enzymes of the oxidative system. | |||
T12580 | PTUPB | COX , Epoxide Hydrolase | |
PTUPB is a potent and dual inhibitor of sEH and COX-2 enzymes(IC50 of 0.9 nM and 1.26 μM, respectively). | |||
T2876 | Flavone | 2-Phenyl-4-benzopyron,2-Phenyl-4-chromone,2-Phenylchromone | NOS , Endogenous Metabolite |
Flavone (2-Phenyl-4-chromone) have effects on CYP (P450) activity which are enzymes that metabolize most drugs in the body. | |||
T1482 | Ciclopirox | HOE296b | ATPase , Ferroptosis , Antibacterial , Autophagy , Antifungal |
Ciclopirox (HOE296b) exerts its action by binding to and chelating trivalent cations, such as Fe3+ and Al3+, thereby inhibiting the availability of essential co-factors for enzymes. Ciclopirox is a synthetic, broad-spect... | |||
T7782 | 3'-Deoxyguanosine | Others | |
3'-Deoxyguanosine is a ligand that can be complexed with enzymes, such as purine nucleoside phosphorylase, and receptors. |