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Farglitazar

Name: Farglitazar
Brand: TargetMol
SKU: T27303
Price: 247 USD
Availability: InStock
Rating: 5 (10 reviews)

(Synonyms: GW 262570X, GI-262570, GI262570, GI-2570, GI 262570) Copy Product Info

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Synonyms: GW 262570X, GI-262570, GI262570, GI-2570, GI 262570

Catalog No. T27303 Copy Product Info

Purity: 99.86%

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Farglitazar (GI-262570) is a PPAR-γ agonist and insulin sensitizer that inhibits stellate cell activation by activating receptor γ via oxidative enzymes proliferators and is used in the study of diabetes.

Cas No. 196808-45-4

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Pack Size	Price	USA Stock	Global Stock
1 mg	$247	In Stock	In Stock
5 mg	$619	In Stock	In Stock
10 mg	$818	In Stock	In Stock
25 mg	$1,260	In Stock	In Stock
1 mL x 10 mM (in DMSO)	$747	In Stock	In Stock

For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)

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Custom-made molecule. TargetMol’s expert synthesis team delivers cost-effective solutions. Contact us for inquiries. Committed to serving you.

For research use only—not for human use. No sales to individuals. Use as intended only.

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Purity:99.86%

ee:100%

Appearance:Solid

Color:Yellow

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COA LCMS CSFC HNMR ORP

Product Introduction

Bioactivity

Description	Farglitazar (GI-262570) is a PPAR-γ agonist and insulin sensitizer that inhibits stellate cell activation by activating receptor γ via oxidative enzymes proliferators and is used in the study of diabetes.
Synonyms	GW 262570X, GI-262570, GI262570, GI-2570, GI 262570

Chemical Properties

Molecular Weight	546.61
Formula	C₃₄H₃₀N₂O₅
Cas No.	196808-45-4
Smiles	C(=O)(C1=C(N[C@@H](CC2=CC=C(OCCC=3N=C(OC3C)C4=CC=CC=C4)C=C2)C(O)=O)C=CC=C1)C5=CC=CC=C5
Relative Density.	1.257 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 80 mg/mL (146.36 mM)

In Vivo Formulation

10% DMSO+90% Saline: < 8 mg/mL (14.64 mM), Lower concentrations may be soluble, but exact solubility limit is unknown.

10% DMSO+40% PEG300+5% Tween 80+45% Saline: 8 mg/mL (14.64 mM), Suspension.

Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.8295 mL	9.1473 mL	18.2946 mL	91.4729 mL
5 mM	0.3659 mL	1.8295 mL	3.6589 mL	18.2946 mL
10 mM	0.1829 mL	0.9147 mL	1.8295 mL	9.1473 mL
20 mM	0.0915 mL	0.4574 mL	0.9147 mL	4.5736 mL
50 mM	0.0366 mL	0.1829 mL	0.3659 mL	1.8295 mL
100 mM	0.0183 mL	0.0915 mL	0.1829 mL	0.9147 mL

Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 µL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 µL Tween 80 and mix well until fully clarified.

3) Add 450 µL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc