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Search Results for "yap"

Targets

Compounds

Cat No. Product Name
TP2160L1 YAP-TEAD-IN-1 acetate YAP-TEAD-IN-1 acetate (1659305-78-8 Free base) YAP
YAP-TEAD-IN-1 acetate 是一种有效的、竞争性的 YAP-TEAD 相互作用抑制剂,IC50 为 25 nM。
T60218 YAP/TAZ inhibitor-2  YAP
YAP/TAZ inhibitor-2 是一种有效的具有口服活性的TEAD-YAP/TAZ 抑制剂,EC50值为 3 nM。YAP/TAZ inhibitor-2 具有抗增殖和抗肿瘤活性。
TP2160 YAP-TEAD-IN-1 Others
YAP-TEAD-IN-1 is a competitive inhibitor of YAP–TEAD interaction (IC50: 25 nM). It shows a higher binding affinity to TE...
T13364 YAP/TAZ inhibitor-1 ROCK
YAP/TAZ inhibitor-1 is an inhibitor of YAP/TAZ (IC50 of <0.100 μΜ in firefly luciferase assay).
TP2160L YAP-TEAD-IN-1 TFA Others
YAP-TEAD-IN-1 TFA is a competitive inhibitor of YAP–TEAD interaction (IC50: 25 nM). It shows a higher binding affinity t...
T7038 4-Methylayapin 4-METHYL-6,7-METHYLENEDIOXYCOUMARIN,4-甲基-6,7-亚甲基二氧代香豆素 Others
4-Methylayapin 用作中间体。
TN1489 3'-Methoxyapiin 3'-甲氧基芹菜苷,3'-Methoxy apiin,Graveobioside B Others
3'-Methoxyapiin 是一种来自 Eminium spiculatum 植物的类黄酮。
T9053 Lats-IN-1 Others , YAP
Lats-IN-1 是一种 ATP 竞争性的、高效的Lats1和Lats2激酶抑制剂,能促进有丝分裂后哺乳动物组织的 Yap 依赖性增殖。
T22372 MYF-01-37 1-[3-Methyl-3-[3-(trifluoromethyl)anilino]pyrrolidin-1-yl]prop-2-en-1-one Others , YAP
MYF-01-37 是共价TEAD 抑制剂,靶向 Cys380,能够可逆地抑制 YAP/TEAD 相互作用。
T3112 Verteporfin CL 318952,BPD-MA,维替泊芬 Autophagy , VDA , YAP , Apoptosis
Verteporfin 是一种用于光动力疗法的光敏剂,用于消除与年龄相关的黄斑变性等疾病相关的眼内异常血管。 它是一种苯并卟啉衍生物单酸环A,可抑制YAP 的活性。
T8421 TED-347 YAP
TED-347 是不可逆的、共价的 YAP-TEAD 蛋白质-蛋白质相互作用变构抑制剂,对 TEAD4•Yap1 蛋白质-蛋白质相互作用的 EC50为 5.9 μM。它与 TEAD4 中央口袋内的 Cys-367 特异性共价结合(Ki:10...
TMPY-06815 SYAP1 Protein, Human, Recombinant (His Tag)
Synapse-associated protein 1 (SYAP1), also known as PRO3113 and BSTA, belongs to the synapse-associated BSD domain famil...
TN2422 6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide Others
6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide is a natural product from Carthamus tinctorius Linn.
TMPY-02648 PACAP receptor/ADCYAP1R1 Protein, Human, Recombinant (hFc Tag)
Pituitary adenylate cyclase activating polypeptide (PACAP, Adcyap1) activation of PAC1 receptors ( Adcyap1r1) significan...
TN1210 2-Hydroxy-1-Methoxyaporphine P450
2-Hydroxy-1-Methoxyaporphine can inhibit CYP2D6 activity, it also increase the glucose consumption significantly as rosi...
TN2353 8-Hydroxyapigenin Others
8-Hydroxyapigenin is Yellow crystalline powder, soluble in organic solvents such as methanol, ethanol, DMSO, etc., deriv...
TN2907 3,6-Dimethoxyapigenin Others
Standard reference
T9566 PY-60 YAP , Annexin A
PY-60 有效激活针对膜联蛋白 A2 (Kd = 1.4 µM) 的 YAP 转录活性。 PY-60 在能够通过增殖重塑表皮的成年动物中激活促增殖、依赖于 YAP 的转录程序。
T67872 VT104 YAP
VT104是一种有效的YAP/TAZ 抑制剂,具有口服活性,可用于癌症研究。VT104阻止内源性TEAD1和TEAD3蛋白棕榈酰化。
T62077 VT103
VT103 是一种 VT101 的类似物,是一种选择性的、口服具有活力的 TEAD1 蛋白棕榈酰化抑制剂。 VT103 能够抑制 YAP/TAZ-TEAD 促进的基因转录,阻断 TEADauto-palmitoylation,并阻断 YAP...
YAP-TEAD-IN-1 acetate
TP2160L1
synonym: YAP-TEAD-IN-1 acetate (1659305-78-8 Free base)
Target:
YAP/TAZ inhibitor-2 
T60218
synonym:
Target:
YAP-TEAD-IN-1
TP2160
synonym:
Target:
YAP/TAZ inhibitor-1
T13364
synonym:
Target:
YAP-TEAD-IN-1 TFA
TP2160L
synonym:
Target:
4-Methylayapin
T7038
synonym: 4-METHYL-6,7-METHYLENEDIOXYCOUMARIN,4-甲基-6,7-亚甲基二氧代香豆素
Target:
3'-Methoxyapiin
TN1489
synonym: 3'-甲氧基芹菜苷,3'-Methoxy apiin,Graveobioside B
Target:
Lats-IN-1
T9053
synonym:
Target:
MYF-01-37
T22372
synonym: 1-[3-Methyl-3-[3-(trifluoromethyl)anilino]pyrrolidin-1-yl]prop-2-en-1-one
Target:
Verteporfin
T3112
synonym: CL 318952,BPD-MA,维替泊芬
Target:
TED-347
T8421
synonym:
Target:
SYAP1 Protein, Human, Recombinant (His Tag)
TMPY-06815
synonym:
Target:
6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide
TN2422
synonym:
Target:
PACAP receptor/ADCYAP1R1 Protein, Human, Recombinant (hFc Tag)
TMPY-02648
synonym:
Target:
2-Hydroxy-1-Methoxyaporphine
TN1210
synonym:
Target:
8-Hydroxyapigenin
TN2353
synonym:
Target:
3,6-Dimethoxyapigenin
TN2907
synonym:
Target:
PY-60
T9566
synonym:
Target:
VT104
T67872
synonym:
Target:
VT103
T62077
synonym:
Target:
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