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Compounds

Cat No. Product Name
T23965 DAT 582 DAT-582,DAT582
DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agent
T70527 DAT-230
DAT-230 is a promising microtubule inhibitor that has great potential for the treatment of fibrosarcoma in vitro and in ...
T25290 DAT1 DAT-1,DAT 1
DAT1 is an antimitotic and antiangiogenic that acts by binding to the colchicine binding site of tubulin.
T5165 10-Deacetyltaxol 去乙酰紫衫醇,10-去乙酰紫杉醇,Deacetyltaxol,10-DAT,10-Desacetyl Paclitaxel,Deacetyl Paclitaxel,10-deacetyl-paclitaxel Others , Microtubule Associated
10-Deacetyltaxol 是从红豆杉中分离得到的一种紫杉醇衍生物,对人脑胶质细胞瘤和神经母细胞瘤细胞具有细胞毒性。它能促进微管蛋白的聚合,在体外抑制由钙离子诱导的微管解聚。
T15378L Gemcitabine elaidate hydrochloride CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride Others
Gemcitabine elaidate (CP-4126) hydrochloride 是 Gemcitabine 的亲脂性前药。Gemcitabine elaidate hydrochloride 通过酯酶转化为 Gemcitabine...
T5735 Methyl deacetylasperulosidate 去乙酰车叶草苷酸甲酯,6α-Hydroxygeniposide,Deacetyl asperulosidic acid methyl ester Others
Methyl deacetylasperulosidate 是环烯醚萜类化合物,能够降低正常小鼠的血糖水平,对小鼠具有通便作用。
T7747 Datelliptium chloride hydrochloride DNA/RNA Synthesis
Datelliptium chloride hydrochloride 是一种衍生自玫瑰树碱的 DNA 嵌入剂,具有抗肿瘤活性。
T2938 (E/Z)-Polydatin 云杉新甙,(E/Z)-Piceid,Polydatin,(E/Z)-虎杖苷 Phospholipase
(E/Z)-Polydatin 是从虎杖的根和根茎中分离得到的一种单晶化合物。它具有抗血小板聚集、心脏保护作用、抗低密度脂蛋白 (LDL) 氧化作用、抗炎和免疫调节功能。
T3427 Polydatin 虎杖苷,Polydotin Peceid,Piceid Apoptosis , Mitophagy , NF-κB , Autophagy
Polydatin 是从传统中药虎杖根中提取的一种天然产物,在多个实验模型中具有抗炎作用。它可抑制 G6PD,并诱导氧化和内质网应激。
T1970 Gedatolisib PF-05212384,PKI-587 mTOR , PI3K
Gedatolisib 是一种高效的双重 PI3Kα (IC50:0.4 nM),PI3Kγ (IC50:5.4 nM) 和 mTOR (IC50:1.6 nM)抑制剂。它在 mTOR 复合物mTORC1和mTORC2中同样有效。
TN3831 (-)-Denudatin B Denudatin B Potassium Channel , ATPase , PAFR , Calcium Channel
(-)-Denudatin B 源自 Magnolia fargesii。 (-)-Denudatin B 通过抑制胶原蛋白和凝血酶诱导的磷酸肌醇分解,在高浓度下具有非特异性抗血小板作用。
T19668 Tiomolibdate diammonium ATTM,Ammonium tetrathiomolybdate,Ammonium molybdenum sulfide,NSC 286644,Coprexa,四硫钼酸铵 Others
Tiomolibdate diammonium 是超氧化物歧化酶 1 (SOD1) 的抑制剂,具有抗血管生成和抗肿瘤活性。 Tiomolibdate diammonium 抑制铜酶的活性,包括 SOD1 和 COX。
T23445 Anxiolytic/nonsedative agent-1 TCS 1205 GABA Receptor
Anxiolytic/nonsedative agent-1 是一种有效的选择性 GABAA 激动剂。Anxiolytic/nonsedative agent-1 对牛脑膜中的 BzR 显示出明显的亲和力,对 α1β2γ2、α2β2γ2、α...
T3273 Bifendate Bifendatatum,联苯双酯 Reverse Transcriptase , HBV
Bifendatatum 是 Schisandrin C 的合成中间体,在慢性 B 型肝炎的研究中具有抗HBV 功效,用于治疗病毒性肝炎和药物性肝损伤引起的转氨酶升高。
T2736 Sodium Demethylcantharidate 去甲斑蝥酸钠,Sodium norcantharidin Others , Endogenous Metabolite
Sodium Demethylcantharidate 是内源性代谢产物的一种。
T5159 Olodaterol hydrochloride BI 1744 hydrochloride,BI-1744 HCl,盐酸奥达特罗 Adrenergic Receptor
BI1744 hydrochloride 是一种长效的、选择性 β2-adrenoceptor(β2-AR) 激动剂 (EC50=0.1 nM;pKi= 9.14 for human β2-adrenoceptor),可用于慢性阻塞性肺疾病...
T7958 Methyl arachidate Methyl Icosanoate,花生酸甲酯 Others , Aminopeptidase
Methyl Icosanoate 是一种天然化合物,具有白三烯 A4 水解酶 (LTA4H) 抑制活性。
T39630 Zandatrigine XEN901,NBI-921352 Sodium Channel
NBI-921352 是钠通道蛋白 8 型亚基 α 的阻断剂,可用于癫痫治疗的神经系统病理学研究。
T3150 Caudatin 告达亭苷元,告达庭 Apoptosis , Others
Caudatin 是白首乌中的一种甾体类天然产物,具有抗肿瘤和抗血管生成作用。它是一种 C-21 甾体糖苷,可使细胞周期停滞,诱导细胞凋亡。
T22867 Indatraline hydrochloride Others
Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET)
DAT 582
T23965
synonym: DAT-582,DAT582
Target:
DAT-230
T70527
synonym:
Target:
DAT1
T25290
synonym: DAT-1,DAT 1
Target:
10-Deacetyltaxol
T5165
synonym: 去乙酰紫衫醇,10-去乙酰紫杉醇,Deacetyltaxol,10-DAT,10-Desacetyl Paclitaxel,Deacetyl Paclitaxel,10-deacetyl-paclitaxel
Target:
Gemcitabine elaidate hydrochloride
T15378L
synonym: CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride
Target:
Methyl deacetylasperulosidate
T5735
synonym: 去乙酰车叶草苷酸甲酯,6α-Hydroxygeniposide,Deacetyl asperulosidic acid methyl ester
Target:
Datelliptium chloride hydrochloride
T7747
synonym:
Target:
(E/Z)-Polydatin
T2938
synonym: 云杉新甙,(E/Z)-Piceid,Polydatin,(E/Z)-虎杖苷
Target:
Polydatin
T3427
synonym: 虎杖苷,Polydotin Peceid,Piceid
Target:
Gedatolisib
T1970
synonym: PF-05212384,PKI-587
Target:
(-)-Denudatin B
TN3831
synonym: Denudatin B
Target:
Tiomolibdate diammonium
T19668
synonym: ATTM,Ammonium tetrathiomolybdate,Ammonium molybdenum sulfide,NSC 286644,Coprexa,四硫钼酸铵
Target:
Anxiolytic/nonsedative agent-1
T23445
synonym: TCS 1205
Target:
Bifendate
T3273
synonym: Bifendatatum,联苯双酯
Target:
Sodium Demethylcantharidate
T2736
synonym: 去甲斑蝥酸钠,Sodium norcantharidin
Target:
Olodaterol hydrochloride
T5159
synonym: BI 1744 hydrochloride,BI-1744 HCl,盐酸奥达特罗
Target:
Methyl arachidate
T7958
synonym: Methyl Icosanoate,花生酸甲酯
Target:
Zandatrigine
T39630
synonym: XEN901,NBI-921352
Target:
Caudatin
T3150
synonym: 告达亭苷元,告达庭
Target:
Indatraline hydrochloride
T22867
synonym:
Target:
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