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Cat No. | Product Name | Synonyms | Targets |
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T23965 | DAT 582 | DAT582,DAT-582 | |
DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agent | |||
T70527 | DAT-230 | ||
DAT-230 is a promising microtubule inhibitor that has great potential for the treatment of fibrosarcoma in vitro and in vivo. DAT-230 exhibited potent anti-proliferative activity against various cancer cells. DAT-230 -tr... | |||
T25290 | DAT1 | DAT-1,DAT 1 | |
DAT1 is an antimitotic and antiangiogenic that acts by binding to the colchicine binding site of tubulin. | |||
T0322 | Fipexide | Dopamine Receptor , AChR | |
Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983. It was served as a nootropic drug in France and Italy, mainly for the therapy of senile dementia, but is... | |||
T22714 | Decynium 22 | Others | |
Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor | |||
T6414 | Bisacodyl | Fenilaxan,Dulcolax,Brocalax | Others |
Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation. | |||
T70525 | ARC39 | ||
ARC39 is acid sphingomyelinase inhibitor (IC50 =20 nM). | |||
T1871 | GBR 12935 dihydrochloride | GBR12935,GBR-12935,GBR 12935 | Dopamine Receptor |
GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels. | |||
T1993 | J-147 | J147 | Epigenetic Reader Domain , Dopamine Receptor , Monoamine Oxidase |
J-147 is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging. It is a curcumin derivative and a potent neurogenic and neuroprotective drug candidate... | |||
T39429 | AHN 1-055 hydrochloride | 3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride | Dopamine Receptor |
AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM). | |||
T11087 | DOV-216,303 Free Base | DOV-216303 | Dopamine Receptor , Serotonin Transporter , Norepinephrine |
DOV-216,303 Free Base (DOV-216303) is an inhibitor of serotonin, norepinephrine, and dopamine reuptake with with IC50s of 14, 20 and 78 nM. DOV-216,303 Free Base exhibits antidepressant effects. | |||
T3526 | Dasotraline hydrochloride | SEP-225289 hydrochloride | Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Norepinephrine |
Dasotraline hydrochloride (SEP-225289 hydrochloride) (SEP-225289 hydrochloride) is a triple reuptake inhibitor that inhibits dopamine, norepinephrine, and serotonin transporters with IC50 values of 4, 6, and 11 nM, respe... | |||
T10758L | Centanafadine hydrochloride | EB-1020 hydrochloride | Dopamine Receptor , Serotonin Transporter , Adrenergic Receptor , Norepinephrine |
Centanafadine hydrochloride (EB-1020 hydrochloride) is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83 nM for human NE, DA, and serotonin... | |||
T7745 | Diclofensine hydrochloride | Ro 8-4650 hydrochloride | Others , Dopamine Receptor |
Diclofensine hydrochloride (Ro 8-4650 hydrochloride) is a Novel Antidepressant, on Peripheral Adrenergic Function | |||
T2092 | Amitifadine hydrochloride | DOV-21947 hydrochloride,EB-1010 hydrochloride | Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Norepinephrine |
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI). | |||
T69807 | EGFR-IN-451 | ||
EGFR-IN-451 is an EGFR inhibitor, attenuating Ang II-induced Kidney Fibrosis. | |||
T7153 | Vanoxerine dihydrochloride | GBR-12909 dihydrochloride,I893 dihydrochloride | Dopamine Receptor |
Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM) | |||
T0991 | Desipramine hydrochloride | NSC-114901,Desmethylimipramine,JB-8181,EX-4355,Norimipramine,G-35020 | Dopamine Receptor , 5-HT Receptor , Serotonin Transporter , Adrenergic Receptor |
Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervous system (CNS), Desipramine hydrochloride blocks the re-upt... | |||
T7341 | Diclofensine | Ro 8-4650 | Dopamine Receptor , Monoamine Transporter |
Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine. | |||
T29534 | ABT-925 fumarate dihydrate | ABT 925,LU201640,ABT925,ABT-925,BSF201640,DAT201 | |
ABT-925 is a selective dopamine D3 receptor (DRD3) antagonist with an in vitro affinity approximately 100 times higher for dopamine D3 receptors than for D2 receptors. | |||
T1970 | Gedatolisib | PF-05212384,PKI-587 | PI3K , mTOR |
Gedatolisib (PF-05212384) is a highly effective dual inhibitor targeting the PI3Kα/γ (IC50: 0.4/5.4 nM)and mTOR (IC50: 1.6 nM) in the PI3K/mTOR signaling pathway. | |||
T23445 | Anxiolytic/nonsedative agent-1 | TCS 1205 | GABA Receptor |
Anxiolytic/nonsedative agent-1 (TCS 1205) is a potent and selective GABAA agonist. Anxiolytic/nonsedative agent-1 shows appreciable affinity for the BzR in bovine brain membranes with Kis of 14, 121, 239 nM for α1β2γ2, α... | |||
T19668 | Tiomolibdate diammonium | Ammonium molybdenum sulfide,Ammonium tetrathiomolybdate,NSC 286644,ATTM,Coprexa | Others |
Tiomolibdate diammonium (NSC-286644) is an inhibitor of superoxide dismutase 1 (SOD1) exerting antiangiogenic and antitumor activities. Tiomolibdate diammonium inhibits the activities of cuproenzymes, including SOD1 and ... | |||
T13110 | Tedatioxetine hydrobromide | Lu AA 24530 hydrobromide | Dopamine Receptor , 5-HT Receptor , Norepinephrine |
Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and an antagonist of 5-HT2A, 5-HT2C, 5-HT3, and α1A-adrenergic receptors, which can be used to treat depress... | |||
T29645 | Adatanserin hydrochloride | WY50324 hydrochloride | 5-HT Receptor |
Adatanserin hydrochloride (WY50324 hydrochloride) is a novel 5-HT(1A)/5-HT(2) receptor ligand with potential neuroprotective effects and inhibition of ischemic efflux of endogenous amino acids, which can be used in the s... | |||
T15378L | Gemcitabine elaidate hydrochloride | CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride | Others |
Gemcitabine elaidate (CP-4126) hydrochloride is lipophilic pro-drug of Gemcitabine. Gemcitabine elaidate hydrochloride is converted to Gemcitabine by esterases in order to be phosphorylated. In contrast to gemcitabine, G... | |||
T9901A-007 | Datopotamab | Others | |
Datopotamab (CDP7657) is a TROP2-targeting antibody that is a naked antibody to Datopotamab deruxtecan and can be used to synthesize active antibody conjugators (Datopotamab deruxtecan). | |||
T34795 | Tedatioxetine | Lu AA-24530,Lu AA24530,Lu AA 24530 | |
Tetaxetine( LU AA24530) has been reported as a triple reuptake inhibitor (5-HT > NE > DA) and 5-HT2A, 5-HT2C, 5-HT3 and α1A-adrenergic receptor antagonist.Meanwhile, it is an antidepressant agent. | |||
T7747 | Datelliptium chloride hydrochloride | DNA/RNA Synthesis | |
Datelliptium chloride hydrochloride is a DNA-intercalating agent derived from ellipticine. with anti-tumor activities. | |||
T23631 | Adatanserin | WY-50324,WY 50324,WAY SEB 324,WY50324 | 5-HT Receptor |
Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist with potential neuroprotective activity for the study of coke oven and depression. | |||
T5159 | Olodaterol hydrochloride | BI-1744 HCl,BI 1744 hydrochloride | Adrenergic Receptor |
Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and activating β2-adrenergic receptors... | |||
T74398 | DATPT | Reactive Oxygen Species , Antibacterial | |
DATPT is a small molecule 12WLVSKF17 peptide mimetic molecule.DATPT inhibits SNX9-p47phox interactions and inhibits the production of reactive oxygen species and inflammatory cytokines.DATPT has anti-inflammatory and ant... | |||
T39630 | Zandatrigine | NBI-921352,XEN901 | Sodium Channel |
Zandatrigine (NBI-921352) is a blocker of sodium channel protein type 8 subunit alpha and can be used in studies about nervous system pathologies of epilepsy treatment. | |||
T22867 | Indatraline hydrochloride | Others | |
Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET) | |||
T75384 | Cy5-dATP | ||
Cy5-dATP is a Cy5 -labeled dATP . Cy5-dATP can be incorporated into a DNA primer [1] [2] . | |||
T126401 | Cordatin | ||
Cordatin is a useful organic compound for research related to life sciences. The catalog number is T126401 and the CAS number is 110382-43-9. | |||
T70323 | Diethanolamine Fusidate | ||
Diethanolamine Fusidate is a bacteriostatic antibiotic with similar activity and better absorption after oral administration (in animals) than the sodium salt of Fusidic Acid. This product inhibits protein synthesis in p... | |||
T15378 | Gemcitabine elaidate | Gemcitabine 5'-elaidate,Gemcitabine (elaidate),CO-101,CP-4126 | Apoptosis , Nucleoside Antimetabolite/Analog , Autophagy |
Gemcitabine elaidate (CP-4126), is a lipophilic, unsaturated fatty acid ester derivative of gemcitabine (dFdC), an antimetabolite deoxynucleoside analogue, with potential antineoplastic activity. Upon hydrolysis intracel... | |||
T16780 | Rodatristat | KAR5417 | Others |
Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively). | |||
T39121 | Odatroltide | DHDMIQK(KAP),Odatroltide | |
Odatroltide is a nanoscale P-selectin inhibitor that serves as a nano-delivery system for 6,7-dihydroxyl-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid and KPAK to specifically target the thrombus. | |||
T76875 | Zanidatamab | ||
Zanidatamab (ZW25) is a bispecific, humanized monoclonal antibody that targets two distinct epitopes (ECD2 and ECD4) of the HER2 receptor, exhibiting anti-tumor activity [1]. | |||
T77104 | Obrindatamab | ||
Obrindatamab, a humanized anti-B7-H3/CD3 bispecific antibody, targets B7-H3 and CD3, facilitating redirected cytotoxic T-lymphocyte (CTL) activity towards B7-H3-expressing cancer cells. It is utilized in cancer research ... | |||
T81033 | TAT-P4-(DATC5)2 | ||
TAT-P4-(DATC5)2 is a potent peptide inhibitor targeting the PDZ domain of protein interacting with C kinase-1 (PICK1), exhibiting a high affinity with a dissociation constant (K_i) of 1.7 nM. This compound has demonstrat... | |||
T73265 | Tolindate | ||
Tolindate, a potent PXR agonist, demonstrates antifungal activity and possesses an EC50 value of 8.3 µM. | |||
T124428 | Datumetine | ||
Datumetine is a useful organic compound for research related to life sciences and the catalog number is T124428. | |||
T31385 | Desethyl-etomidate | R28141,Etomidate acid,R-28141,R 28141 | |
Desethyl-etomidate is a biochemical. | |||
T82717 | Cis-Indatraline hydrochloride | cis-Lu 19-005 | |
Cis-indatraline hydrochloride (cis-Lu 19-005) is an active compound utilized in the research of neurodegenerative diseases [1]. | |||
T24458 | Methyl acetimidate | ||
Methyl acetimidate is an effective in vitro antisickling agent. It has few detrimental effects on the red cell. | |||
T7429 | Datelliptium chloride | DNA/RNA Synthesis | |
Datelliptium chloride is a DNA-intercalating agent derived from ellipticine. Datelliptium chloride shows anti-tumor activities. | |||
T38630 | Ludaterone | ||
Ludaterone is an antiandrogen agent, with potent antiandrogenic activity. |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5165 | 10-Deacetyltaxol | 10-DAT,10-Desacetyl Paclitaxel,Deacetyltaxol,10-deacetyl-paclitaxel,Deacetyl Paclitaxel | Others , Microtubule Associated |
10-Deacetyltaxol (10-DAT) is extracted from Taxus brevifolia barks. | |||
TN6552 | 5,7-Dimethoxyluteolin | Dopamine Receptor | |
5,7-Dimethoxyluteolin is a natural product from Hovenia acerba. 5,7-Dimethoxyluteolin is a dopamine transporter (DAT) activator with an EC50 of 3.417 μM. | |||
T7958 | Methyl arachidate | Methyl Icosanoate | Others , Aminopeptidase |
Methyl arachidate (Methyl Icosanoate) is an esterified form of arachidic acid | |||
T2736 | Sodium Demethylcantharidate | Sodium norcantharidin | Others , Endogenous Metabolite |
Sodium Demethylcantharidate (Sodium norcantharidin) is extracted from Mylabris phqlarata pallas and has potent antitumor activity. | |||
T3150 | Caudatin | Apoptosis , Others | |
Caudatin is one of the species of C-21 steroidal glycosides mainly isolated from the root of Cynanchum bungei Decne and exhibits potent anticancer activities. | |||
T3273 | Bifendate | Bifendatatum | HBV , Reverse Transcriptase |
Bifendate (Bifendatatum) is commonly used to treat the transaminase elevation that caused by viral hepatitis and drug-induced liver injury. | |||
TN3831 | (-)-Denudatin B | Denudatin B | ATPase , Potassium Channel , Calcium Channel , PAFR |
(-)-Denudatin B (Denudatin B) is derived from Magnolia fargesii. (-)-Denudatin B has nonspecific antiplatelet action at high concentration by inhibiting phosphoinositides breakdown induced by collagen and thrombin. | |||
T3427 | Polydatin | Piceid,Polydotin Peceid | Apoptosis , Mitophagy , NF-κB , Autophagy |
Polydatin (Piceid), the glycoside of Resveratrol, is originally isolated from the Chinese herb Polygonum cuspidatum. The compound can inhibit platelet aggregation and elevate the ratios of LDL-C/HDL-C and TC/HDL-C. In th... | |||
T2938 | (E/Z)-Polydatin | Polydatin,(E/Z)-Piceid | Phospholipase |
(E/Z)-Polydatin (Polydatin), is a natural precursor and glycoside form of resveratrol with a monocrystalline structure. While it is isolated from the bark of Picea sitchensis or Polygonum cuspidatum, Polydatin may be det... | |||
T5735 | Methyl deacetylasperulosidate | Deacetyl asperulosidic acid methyl ester,6α-Hydroxygeniposide | Others |
Methyl deacetylasperulosidate (6α-Hydroxygeniposide) is a natual product isolated from the herbs of Hedyotis diffusa Willd,it can lower the blood glucose level in normal mice. | |||
T38415 | Adenosine 5′-monophosphoramidate sodium | ||
Adenosine 5′-monophosphoramidate sodium is a derivative of adenosine used as an intermediate for nucleotide synthesis. It significantly influences the accumulation of cyclic AMP. | |||
TN3772 | Datiscin | Others | |
Datiscin is a natural product for research related to life sciences. The catalog number is TN3772 and the CAS number is 16310-92-2. | |||
TN6027 | Pedatisectine F | 2-Methyl-6-(1,2,3,4-tetrahydroxybutyl)pyrazine | |
Pedatisectine F is a natural product of Pinellia, Araceae. The catalog number is TN6027 and the CAS number is 206757-32-6. Pedatisectine F can be used as a reference standard. | |||
TN3262 | 8(17),12E,14-Labdatrien-20-oic acid | Others | |
8(17),12E,14-Labdatrien-20-oic acid is a natural product from Isodon yuennanensis. | |||
T3S0626 | Denudatine | Others | |
1. Denudatine has effects on action potential of ventricular fibers and has inhibition on arrhythmogenic action of aconitine. | |||
TN3773 | Daturabietatriene | Others | |
Daturabietatriene is a natural product from Pinus yunnanensis. | |||
TN3774 | Daturametelin I | Others | |
Daturametelin I is a natural product for research related to life sciences. The catalog number is TN3774 and the CAS number is 904667-65-8. | |||
TN3776 | Daturataturin A | Others | |
Daturataturin A is a natural product of Datura, Solanaceae. The catalog number is TN3776 and the CAS number is 133360-51-7. Daturataturin A can be used as a reference standard. | |||
TN6570 | Daturaolone | ||
Daturaolone has potency in reducing the harmful effects or in maintaining the normal hepatic physiological mechanisms in both acute and chronic hepato-toxic induced liver damage in rats. Daturaolone also possesses in viv... | |||
TN3788 | Decursidate | Others | |
Decursidate is a natural product of Peucedanum, Apiaceae. The catalog number is TN3788 and the CAS number is 272122-56-2. Decursidate can be used as a reference standard. | |||
TN5218 | Valerosidate | Others | |
Valerosidate is a natural product from Valeriana jatamansi. | |||
T75637 | Demethylcantharidate disodium | ||
Demethylcantharidate disodium, an endogenous metabolite, demonstrates significant anticancer efficacy against various cancers by inducing apoptosis in hepatocellular carcinoma cells through endoplasmic reticulum (ER) str... | |||
TN7002 | Methyl linolelaidate | ||
Methyl linolelaidate is a natural product. | |||
TN3775 | Daturataturin A aglycone | Others | |
Daturataturin A aglycone is a natural product for research related to life sciences. The catalog number is TN3775 and the CAS number is 904665-71-0. | |||
TN2161 | Rotundatin | Others | |
Rotundatin is a natural product from Dendrobium rotundatum. |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-01596 | AADAT Protein, Human, Recombinant (His & SUMO) | Human | E. coli |
Transaminase with broad substrate specificity. Has transaminase activity towards aminoadipate, kynurenine, methionine and glutamate. Shows activity also towards tryptophan, aspartate and hydroxykynurenine. Accepts a vari... | |||
TMPH-00445 | GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His) | Chinese hamster | Yeast |
GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His) is expressed in Yeast. | |||
TMPY-05690 | Human mastadenovirus B (HAdV-B) encapsidation protein IVa2 Protein (His) | HAdV-B | Baculovirus-Insect Cells |
TMPH-00444 | GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His & Myc) | Chinese hamster | E. coli |
GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His & Myc) is expressed in E. coli. |
Cat No. | Product Name | ||
---|---|---|---|
L2900 | Oxidation-Reduction Compound Library | 1279 compounds | |
1279 small molecule compounds with pro-oxidant or anti-oxidant activity for high-throughput and high-content screening. |