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Anti-Cancer Approved Drug Library

Catalog No. L2110
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 1825 approved anti-cancer drugs based on published literatures and database to form this collection that can be used as positive controls in biological cancer investigation and cancer correlation study.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Compound Libraries | TargetMol
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 1825 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • These FDA, EMA, or NMPA approved anti-cancer drugs have annotated bioactivity, safety, and bioavailability;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

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Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L2110)

Publications Cited TargetMol Libraries

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Library Composition

Autophagy (334)
Apoptosis (245)
5-HT Receptor (160)
Adrenergic Receptor (159)
Endogenous Metabolite (151)
Antibacterial (138)
COX (120)
Antibiotic (116)
Dopamine Receptor (109)
Histamine Receptor (106)
DNA/RNA Synthesis (81)
Sodium Channel (79)
Calcium Channel (75)
Potassium Channel (73)
AChR (67)
Parasite (53)
Glucocorticoid Receptor (52)
P450 (44)
HIV Protease (43)
Reactive Oxygen Species (38)
Ferroptosis (37)
NF-κB (36)
Antifungal (36)
EGFR (34)
GABA Receptor (34)
Estrogen/progestogen Receptor (32)
c-Kit (32)
VEGFR (31)
Mitophagy (31)
Topoisomerase (30)
PPAR (29)
Nucleoside Antimetabolite/Analog (29)
PDGFR (29)
SARS-CoV (28)
Influenza Virus (27)
Prostaglandin Receptor (26)
Dehydrogenase (26)
Estrogen Receptor/ERR (25)
PDE (25)
Serotonin Transporter (23)
Proton pump (22)
Microtubule Associated (22)
DNA Alkylator/Crosslinker (21)
Norepinephrine (21)
ATPase (20)
iGluR (20)
Androgen Receptor (19)
Opioid Receptor (19)
HDAC (18)
FLT (17)
RAAS (17)
HSV (17)
Virus Protease (16)
JAK (16)
FGFR (16)
c-Met/HGFR (15)
Bcr-Abl (15)
Adenosine Receptor (15)
TRP/TRPV Channel (14)
Src (14)
HBV (14)
Tyrosine Kinases (14)
TNF (13)
Progesterone Receptor (13)
NMDAR (13)
Antifolate (13)
GNRH Receptor (13)
Retinoid Receptor (12)
Raf (12)
PKC (12)
CDK (12)
MAO (11)
DHFR (11)
P-gp (11)
SGLT (11)
MRP (11)
ROS (11)
Reverse Transcriptase (10)
ALK (10)
HMG-CoA Reductase (10)
AChE (10)
Drug Metabolite (10)
DNA Alkylation (10)
Proteasome (10)
Carbonic Anhydrase (10)
Antifection (9)
MMP (9)
CaMK (9)
AMPK (9)
HCV Protease (9)
PARP (9)
Lipoxygenase (9)
c-RET (9)
Phosphatase (9)
PI3K (8)
Monoamine Oxidase (8)
P2Y Receptor (8)
Chloride channel (8)
GluR (8)
HIF/HIF Prolyl-Hydroxylase (8)
BTK (8)
Monoamine Transporter (7)
NADPH (7)
mTOR (7)
ABC (7)
Guanylate cyclase (7)
STAT (7)
HER (7)
GPR (7)
Phospholipase (7)
CFTR (7)
MEK (7)
Neurokinin receptor (7)
Thrombin (7)
DNA (6)
Vasopressin Receptor (6)
Interleukin (6)
BCL (6)
Hedgehog/Smoothened (6)
S1P Receptor (6)
Mitochondrial Metabolism (6)
Aromatase (6)
ERK (6)
TAM Receptor (6)
DNA Methyltransferase (6)
Transferase (6)
IL Receptor (6)
Trk receptor (6)
ribosome (6)
Glutathione Peroxidase (5)
Leukotriene Receptor (5)
LPL Receptor (5)
Nrf2 (5)
Ras (5)
Endothelin Receptor (5)
Sigma receptor (5)
TLR (5)
Histone Methyltransferase (5)
Caspase (5)
CaSR (5)
FXR (5)
ROCK (5)
Wnt/beta-catenin (5)
P2X Receptor (5)
Antiviral (4)
Amino Acids and Derivatives (4)
Oxytocin Receptor (4)
p38 MAPK (4)
PKA (4)
GSK-3 (4)
IκB/IKK (4)
Beta Amyloid (4)
HIF (4)
Akt (4)
PGE Synthase (4)
GPCR19 (4)
Melatonin Receptor (4)
LTR (4)
HSP (4)
Smo (4)
DPP-4 (4)
NO Synthase (4)
Fatty Acid Synthase (4)
Annexin A (4)
ROS Kinase (4)
NOD (4)
CXCR (4)
Tyrosinase (4)
Antioxidant (3)
Aminopeptidase (3)
Free radical scavengers (3)
AhR (3)
FAK (3)
MT Receptor (3)
Adenosine deaminase (3)
Cysteine Protease (3)
Serine/threonin kinase (3)
Integrin (3)
c-Fms (3)
Ligand for E3 Ligase (3)
cholecystokinin (3)
Melanocortin Receptor (3)
Serine Protease (3)
Syk (3)
UGT (3)
Hydroxylase (3)
PAK (3)
GST (3)
Na-K-Cl cotransporter (3)
TGF-beta/Smad (3)
IGF-1R (3)
Isocitrate Dehydrogenase (IDH) (3)
Xanthine Oxidase (3)
Molecular Glues (3)
MAPK (2)
Monocarboxylate transporter (2)
Gamma-secretase (2)
GHSR (2)
CRM1 (2)
OAT (2)
CGRP Receptor (2)
ROR (2)
Cannabinoid Receptor (2)
IRE1 (2)
Gap Junction Protein (2)
Rho (2)
Aurora Kinase (2)
CAT (2)
NOS (2)
Aryl Hydrocarbon Receptor (2)
Protease-activated Receptor (2)
Somatostatin (2)
NOD-like Receptor (NLR) (2)
CCR (2)
TOPK (2)
LDL (2)
PLK (2)
Hexokinase (2)
Cell wall (2)
Beta-Secretase (2)
Glutathione reductase (2)
Lipid (2)
Reductase (2)
YAP (2)
Ephrin Receptor (2)
RSV (2)
IFNAR (2)
Decarboxylase (2)
Ligands for Target Protein for PROTAC (2)
DNA gyrase (2)
Arginase (2)
Hck (1)
CSF-1R (1)
Histone Acetyltransferase (1)
IAP (1)
S6 Kinase (1)
PAD (1)
Chk (1)
Sirtuin (1)
Glucagon Receptor (1)
OX Receptor (1)
VDA (1)
Bradykinin Receptor (1)
BACE (1)
p53 (1)
Imidazoline Receptor (1)
PD-1/PD-L1 (1)
Liver X Receptor (1)
Mdm2 (1)
ACK (1)
NPC1L1 (1)
Immunology/Inflammation related (1)
FAAH (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Histone Demethylase (1)
PDK (1)
MTH1 (1)
DUB (1)
Lipase (1)
Factor Xa (1)
JNK (1)
GRK (1)
Epigenetic Reader Domain (1)
RAR/RXR  (1)
PAFR (1)
NADPH-oxidase (1)
Thrombopoietin Receptor (1)
Adiponectin receptor (1)
cAMP (1)
Neprilysin (1)
ATP Citrate Lyase (1)
Hydrogenase (1)
Complement System (1)
Pyroptosis (1)
Platelet aggregation (1)
PROTAC Linker (1)
GluCls (1)
Na+/Ca2+ Exchanger (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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