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TargetMol | Compound Library

Anti-Cancer Approved Drug Library

Catalog No. L2110

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 1800 approved anti-cancer drugs based on published literatures and database to form this collection that can be used as positive controls in biological cancer investigation and cancer correlation study.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2110

Anti-Cancer Approved Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 1800 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • These FDA, EMA, or NMPA approved anti-cancer drugs have annotated bioactivity, safety, and bioavailability;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Autophagy
Apoptosis
Adrenergic Receptor
5-HT Receptor
Endogenous Metabolite
Antibacterial
COX
Antibiotic
Dopamine Receptor
Histamine Receptor
Sodium Channel
Potassium Channel
Calcium Channel
DNA/RNA Synthesis
AChR
Parasite
Glucocorticoid Receptor
Cytochromes P450
HIV Protease
EGFR
NF-κB
Estrogen/progestogen Receptor
Antifungal
VEGFR
Reactive Oxygen Species
GABA Receptor
Ferroptosis
Topoisomerase
PPAR
Mitophagy
Estrogen Receptor/ERR
PDGFR
c-Kit
Nucleoside Antimetabolite/Analog
SARS-CoV
Dehydrogenase
Prostaglandin Receptor
PDE
Microtubule Associated
Serotonin Transporter
Influenza Virus
Norepinephrine
ATPase
Proton pump
iGluR
JAK
FGFR
HDAC
HSV
Androgen Receptor
DNA Alkylator/Crosslinker
RAAS
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Src
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c-Met/HGFR
Adenosine Receptor
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ALK
GNRH Receptor
MAO
NMDAR
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Lipoxygenase
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P2Y Receptor
PI3K
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Imidazoline Receptor
p53
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