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TargetMol | Compound Library

Anti-Cancer Approved Drug Library

Catalog No. L2110

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 2020 approved anti-cancer drugs based on published literatures and database to form this collection that can be used as positive controls in biological cancer investigation and cancer correlation study.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2110

Anti-Cancer Approved Drug Library

size

  • 1 mg
  • 10 µL x 10 mM (in DMSO)
  • 30 µL x 10 mM (in DMSO)
  • 50 µL x 10 mM (in DMSO)
  • 100 µL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 2020 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • These FDA, EMA, or NMPA approved anti-cancer drugs have annotated bioactivity, safety, and bioavailability;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
Adrenergic Receptor
5-HT Receptor
Antibiotic
COX
Dopamine Receptor
Histamine Receptor
Potassium Channel
DNA/RNA Synthesis
Parasite
Sodium Channel
NF-κB
Calcium Channel
AChR
ROS
Glucocorticoid Receptor
Cytochromes P450
Antifungal
Reactive Oxygen Species
EGFR
HIV Protease
VEGFR
GABA Receptor
SARS-CoV
Estrogen/progestogen Receptor
Ferroptosis
Virus Protease
Estrogen Receptor/ERR
Topoisomerase
Mitophagy
Influenza Virus
Akt
PPAR
c-Kit
Interleukin
TNF
Microtubule Associated
Prostaglandin Receptor
Nucleoside Antimetabolite/Analog
ERK
PDGFR
Dehydrogenase
Serotonin Transporter
p38 MAPK
c-Met/HGFR
Caspase
iGluR
PDE
JAK
HSV
HDAC
ATPase
Norepinephrine
TRP/TRPV Channel
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STAT
RAAS
PI3K
Bcr-Abl
CDK
Opioid Receptor
Bcl-2 Family
FGFR
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GNRH Receptor
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HIF/HIF Prolyl-Hydroxylase
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ribosome
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Aminopeptidase
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FAK
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TOPK
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IRE1
Cysteine Protease
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glycosidase
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Decarboxylase
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CGRP Receptor
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YAP
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IFNAR
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cAMP
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transporter
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GluCls
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PAI-1
Casein Kinase
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S6 Kinase
Imidazoline Receptor
Ferroportin
Drug-Linker Conjugates for ADC

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