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Search Results for "vegfr"

Targets

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Compounds

Cat No. Product Name
T37078 VEGFR-2-IN-6 VEGFR
VEGFR-2-IN-6 (WO 02/059110, example 64) is a potent inhibitor of VEGFR2, a crucial receptor involved in the regulation o...
T2056 VEGFR-2-IN-5 UNC0064-12,2,4-Pyrimidinediamine with linker,2, 4-Pyrimidinediamine with linker VEGFR
UNC0064-12 是 VEGFR2 抑制剂,摘自专利文献 WO2013055780A1 中第 69 页。
T23504 VEGFR-IN-1 VEGFR Tyrosine Kinase Inhibitor II Others
VEGFR inhibitor
T63112 VEGFR-IN-3
VEGFR-IN-3 (compound 3f) 是 VEGFR 抑制剂。VEGFR-IN-3 抑制 OVCAR-4 和 MDA-MB-468 癌细胞的生长,其 IC50值分别为 0.29 和 0.35 μM。VEGFR-IN-3 可用于癌...
T68526 VEGFR-IN-V
VEGFR-IN-V is a potent, vascular endothelial growth factor receptor-​2 (VEGFR-2) tyrosine kinase inhibitor.
T62763 VEGFR-2-IN-12
VEGFR-2-IN-12 (compound 6g) 是一种 2-oxoquinoxalinyl-1,2,4-triazole,是一种 VEGFR-2 的有效抑制剂 (IC50: 0.037 μM)。VEGFR-2-IN-12 能够高度抑...
T61861 VEGFR-2-IN-20
VEGFR-2-IN-20 (Compound 7) is a highly effective VEGFR inhibitor with significant potential for cancer research [1].
T62796 VEGFR-2-IN-13
VEGFR-2-IN-13 (Compound 19a) 是一种有效的 VEGFR-2 抑制剂 (IC50: 3.4 nM)。VEGFR-2-IN-13 能够将 HepG2 的细胞周期停滞在 G2/M 期,诱导细胞凋亡 (apoptosis...
T63168 VEGFR-2-IN-26
VEGFR-2-IN-26 (compound 5h) 是一种 VEGFR-2 的高效抑制剂 (IC50: 15.5 nM)。VEGFR-2-IN-26 对白血病、中枢神经系统、非小肺、卵巢、肾、前列腺和乳腺癌细胞表现出良好的抗增殖作用。
T61631 VEGFR-2-IN-23
VEGFR-2-IN-23 (compound 11b) is a highly potent and selective inhibitor of VEGFR-2, with an impressive IC 50 value of 0....
T61137 VEGFR-2-IN-19
VEGFR-2-IN-19 (Compound 15b) is a highly efficacious inhibitor of VEGFR2, a receptor involved in angiogenesis. Its mecha...
T64060 VEGFR-2-IN-21
VEGFR-2-IN-21 是 VEGFR-2 的有效抑制剂 (IC50: 0.10 μM),表现出抗癌作用。
T62071 VEGFR-2-IN-16
VEGFR-2-IN-16 (Compound 15b) 是一种 VEGFR-2 的有效抑制剂 (IC50: 86.36 nM),表现出抗肿瘤效果。
T62901 VEGFR-2-IN-27
VEGFR-2-IN-27 (compound 7a) 是一种 VEGFR-2 的高效抑制剂 (IC50: 14.8 nM),能够用于抗癌研究。
T61561 VEGFR-2-IN-18
VEGFR-2-IN-18 (Compound 15d) is a high-potency inhibitor of VEGFR-2, with an IC 50 value of 60 nM. This compound effecti...
T63822 VEGFR-2-IN-22
VEGFR-2-IN-22 (Compound 25) 是 VEGFR-2 和 β-tubulin 聚合抑制剂,对 VEGFR-2 的 IC50=19.82 nM。VEGFR-2-IN-22 能够诱导细胞凋亡 (apoptosis)。
T63804 VEGFR-2-IN-28
VEGFR-2-IN-28 是 VEGFR-2 的有效抑制剂 (IC50: 0.83 μM)。VEGFR-2-IN-28 能够诱导细胞凋亡 (apoptosis),表现出抗肿瘤效果。
T62314 VEGFR-2-IN-25
VEGFR-2-IN-25 (compound 5d) 是一种 VEGFR-2 的高效抑制剂 (IC50: 12.1 nM)。VEGFR-2-IN-25 能够用于研究抗癌。
T63002 VEGFR-2-IN-15
VEGFR-2-IN-15 (Compound 14b) 是一种 VEGFR-2 的有效抑制剂。VEGFR-2-IN-15 能够抑制 HepG2 细胞在 Pre-G1 期的生长,诱导细胞凋亡。
T72890 VEGFR-2-IN-30
VEGFR-2-IN-30 是一种 VEGFR-2 抑制剂 (IC50: 66 nM)。VEGFR-2-IN-30 还抑制 PDGFR、EGFR 和 FGFR1,IC50s 分别为 180、98、82 nM。VEGFR-2-IN-30 将癌...
VEGFR-2-IN-6
T37078
synonym:
Target:
VEGFR-2-IN-5
T2056
synonym: UNC0064-12,2,4-Pyrimidinediamine with linker,2, 4-Pyrimidinediamine with linker
Target:
VEGFR-IN-1
T23504
synonym: VEGFR Tyrosine Kinase Inhibitor II
Target:
VEGFR-IN-3
T63112
synonym:
Target:
VEGFR-IN-V
T68526
synonym:
Target:
VEGFR-2-IN-12
T62763
synonym:
Target:
VEGFR-2-IN-20
T61861
synonym:
Target:
VEGFR-2-IN-13
T62796
synonym:
Target:
VEGFR-2-IN-26
T63168
synonym:
Target:
VEGFR-2-IN-23
T61631
synonym:
Target:
VEGFR-2-IN-19
T61137
synonym:
Target:
VEGFR-2-IN-21
T64060
synonym:
Target:
VEGFR-2-IN-16
T62071
synonym:
Target:
VEGFR-2-IN-27
T62901
synonym:
Target:
VEGFR-2-IN-18
T61561
synonym:
Target:
VEGFR-2-IN-22
T63822
synonym:
Target:
VEGFR-2-IN-28
T63804
synonym:
Target:
VEGFR-2-IN-25
T62314
synonym:
Target:
VEGFR-2-IN-15
T63002
synonym:
Target:
VEGFR-2-IN-30
T72890
synonym:
Target:
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