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Results for "

pkc

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    333
    TargetMol | Inhibitors_Agonists
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    TargetMol | Compound_Libraries
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    TargetMol | Natural_Products
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    TargetMol | Inhibitors_Agonists
PKC-theta inhibitor
T5423736048-65-0
PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.
  • $108
In Stock
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QTY
Staurosporine
CGP 41251, Antibiotic AM-2282, AM-2282
T668062996-74-1
Staurosporine (AM-2282) is a protein kinase inhibitor with ATP-competitive and non-selective inhibitory activity (IC50=6 15 2 3 3000 nM) against PKC, PKA, c-Fgr, phosphorylase kinase and TAOK2. Staurosporine also induces apoptosis.
  • $56
In Stock
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QTY
TargetMol | Inhibitor Hot
20-HETE
20-hydroxy Arachidonic Acid
T1402179551-86-3In house
20-HETE promotes cell proliferation and migration in cancer and can be used to study prostate tumors and cardiac hypertrophy by activating the protein kinase C pathway to increase FBXO10 expression.20-HETE promotes cell proliferation and migration in cancer and can be used to study prostate tumors and cardiac hypertrophy by activating the protein kinase C pathway.
  • $498
In Stock
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QTY
TargetMol | Inhibitor Hot
Phorbol 12,13-dibutyrate
Phorbol dibutyrate, PDBu
T1652637558-16-0In house
Phorbol 12,13-dibutyrate (Phorbol dibutyrate) is a PKC activator that inhibits α1-adrenoceptor-mediated positive inotropic effects in a concentration-dependent manner, induced by contraction of isolated rabbit vascular smooth muscle.
  • $56
In Stock
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QTY
TargetMol | Inhibitor Hot
Go 6983
Goe 6983
T6313133053-19-7
Go 6983, a pan-PKC inhibitor, targets PKCα, PKCβ, PKCγ, PKCδ, and PKCζ, with IC50 values of 7 nM, 7 nM, 6 nM, 10 nM, and 60 nM, respectively.
  • $36
In Stock
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TargetMol | Inhibitor Hot
Bisindolylmaleimide I
Go 6850, GF109203X
T6513133052-90-1
Bisindolylmaleimide I (GF109203X) is a potent and highly selective protein kinase C (PKC) inhibitor, exhibiting a Ki of 14 nM.
  • $61
In Stock
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TargetMol | Inhibitor Hot
Phorbol 12-myristate 13-acetate
PMA
TQ019816561-29-8
Phorbol 12-myristate 13-acetate (PMA), a member of the phorbol ester group of natural products, activates PKC, SphK, and NF-κB, and induces THP1 cell differentiation.
  • $44
In Stock
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QTY
TargetMol | Inhibitor Hot
Ionomycin calcium
SQ23377 calcium
T1166556092-82-1In house
Ionomycin calcium (SQ23377 calcium) is an effective and selective calcium ionophore, demonstrating high specificity for divalent cations (Ca>Mg>Sr=Ba).
  • $127
4-6 weeks
Size
QTY
Bisindolylmaleimide VIII
RO 318161, Ro 31-7549, Bis VIII
T71125125313-65-7In house
Bisindolylmaleimide VIII (Ro-31-7549) is a selective and potent protein kinase C (PKC) inhibitor with good inhibition of PKC-α, PKC-β I, PKC-β II, PKC-γ, and PKC-ε.Bisindolylmaleimide VIII Bisindolylmaleimide VIII inhibits T cell-mediated autoimmune diseases and enhances Fas-mediated apoptosis through a protein kinase C-independent mechanism.
  • $293 TargetMol
In Stock
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Safingol hydrochloride
SPC 100270 hydrochloride, L-threo-dihydrosphingosine hydrochloride
T83978139755-79-6In house
Safingol hydrochloride (L-threo-dihydrosphingosine hydrochloride) is a specific inhibitor of protein kinase C. It induces autophagy in solid tumor cells and cancer cell death by inhibiting the PKC and PI3-kinase pathways.BIIB 722 Mesylate is a selective sodium-hydrogen exchange inhibitor. Safingol hydrochloride inhibits PKC and PI3k.
  • $195 TargetMol
In Stock
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Ellagic acid
Gallogen, Elagostasine
T0465476-66-4
Ellagic acid (Gallogen), a thickened tetracyclic natural product, is a potent CK2 inhibitor (IC50=40 nM; Ki=20 nM) with ATP-competitive properties. Ellagic acid is an antioxidant and also possesses antiproliferative activity.
  • $44
In Stock
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Piceatannol
trans-Piceatannol, Astringenin
T061010083-24-6
Piceatannol (Astringenin) is an anti-inflammatory, immunomodulatory and antiproliferative agent. It inhibits p56lck and syk protein tyrosine kinases and inhibits NF-κB activation and gene expression of TNF-induced. It is synthetic from the conversion of resveratrol by cytochrome P450 1B1.
  • $39
In Stock
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Fasudil
HA-1077, AT877
T1606103745-39-7
Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.
  • $33
In Stock
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α-Vitamin E
Vitamin E, D-α-Tocopherol, Alpha-Tocopherol, 5,7,8-Trimethyltocol, (+)-alpha-Tocopherol
T164859-02-9
α-Vitamin E (Dexrabeprazole Sodium) is a naturally-occurring form of vitamin E, a fat-soluble vitamin with potent antioxidant properties.
  • $38
In Stock
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Fasudil hydrochloride
HA-1077 hydrochloride, Fasudil HCl, Fasudil (HA-1077) HCl, AT-877 hydrochloride
T3060105628-07-7
Fasudil hydrochloride (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively.
  • $35
In Stock
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Mitoxantrone
mitozantrone
T658865271-80-9
Mitoxantrone (mitozantrone) is an anthracenedione antibiotic with antineoplastic activity. Mitoxantrone intercalates into and crosslinks DNA, thereby disrupting DNA and RNA replication. This agent also binds to topoisomerase II, resulting in DNA strand breaks and inhibition of DNA repair. Mitoxantrone is less cardiotoxic compared to doxorubicin.
  • $33
In Stock
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N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
T92561071135-06-2
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein kinase C D (PKC PKD) inhibitor[1].
  • $148
In Stock
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Afuresertib
GSK2110183C, GSK2110183
T19111047644-62-1
Afuresertib (GSK2110183) is an orally bioavailable inhibitor of the serine threonine protein kinase Akt (protein kinase B) with potential antineoplastic activity.
  • $33
In Stock
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TargetMol | Inhibitor Sale
Chelerythrine chloride
T34193895-92-9
Chelerythrine Chloride is a cell-permeable inhibitor of protein kinase C, competitive with respect to the phosphate acceptor and non-competitive with respect to ATP.
  • $63
In Stock
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D-ERYTHRO-SPHINGOSINE
trans-4-Sphingenine, Sphingosine-1-phosphate, Sphingosine (d18:1), Sphinganine, Erythrosphingosine, erythro-C18-Sphingosine
T5891123-78-4
D-erythro-Sphingosine (trans-4-Sphingenine) is a protein kinase C (PKC) inhibitor. D-erythro-Sphingosine (Erythrosphingosine) is also a PP2A activator
  • $39
In Stock
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Enzastaurin
LY317615
T6280170364-57-5
Enzastaurin (LY317615) (LY317615) is an effective PKCβ selective inhibitor (IC50: 6 nM), 6- to 20-fold selectivity against PKCα γ ε.
  • $43
In Stock
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Ro 31-8220 Mesylate
Ro 31-8220 methanesulfonate, Bisindolylmaleimide IX mesylate
T6643138489-18-6
Ro 31-8220 Mesylate (Bisindolylmaleimide IX mesylate) is a pan-PKC inhibitor for PKC-α βI βII γ ε (IC50: 5 24 14 27 24 nM), and also shows potent inhibition against MSK1, MAPKAP-K1b, S6K1, and GSK3β.
  • $44
In Stock
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Chelerythrine
Toddalin, Cheleritrine, Broussonpapyrine
T6S005234316-15-9
1. Chelerythrine (Broussonpapyrine) may have antimanic effect . 2. Chelerythrine can inhibit telomerase activity. 3. Chelerythrine is a well-known protein kinase C inhibitor . 4. Chelerythrine has potential antiproliferative and antitumor effects.
  • $50
In Stock
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HA-100
T764884468-24-6
HA-100 is an inhibitor of protein kinase
  • $57
In Stock
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