Home Tools
Log in
Cart

Search Result

Search Results for " antiinflammatory "

Targets

30

Compounds

32

Natural Products

5

Recombinant Proteins

3

Libraries

Cat No. Product Name Synonyms Targets
T11020 DHODH-IN-11 Dehydrogenase , DNA/RNA Synthesis
DHODH-IN-11 is a leflunomide derivative and weak dihydroorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.03.
T22358 Etalocib LY293111,VML295 Apoptosis , Leukotriene Receptor , LTR
Etalocib (LY293111) is a novel diaryl ether carboxylic acid derivative, is a selective and potent inhibitor of the lipoxygenase pathway either via antagonism of the leukotriene B4 (LTB4) receptor or directly through 5'-l...
T21606L Anti-Inflammatory Peptide 1 Acetate Anti-Inflammatory Peptide 1 Acetate(118850-70-8 Free base) Phospholipase
Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) possesses a potent anti-inflammatory activity in vivo and is a strong inhibitor of phospholipase A2 (PLA2), whose increased presence and activity results in inflammati...
T41302 Itaconate-alkyne ITalk Others
Itaconate-alkyne (ITalk) is a bioorthogonal probe for quantitative and site-specific chemoproteomic profiling of itaconate in inflammatory macrophages and enables biochemical evaluation and proteomic analysis of its dire...
T12856 SC-26196 Others
SC-26196 is an orally active inhibitor of Delta6 desaturase (D6D) with IC50 of 0.2 µM in a rat liver microsomal assay, with antiinflammatory properties.
T1163 Betamethasone valerate Betnovate,Betaderm,Betamethasone 17-valerate,Luxiq Glucocorticoid Receptor
Betamethasone valerate (Luxiq) is a synthetic glucocorticoid with metabolic, immunosuppressive and anti-inflammatory actions.
T0383 Fenspiride hydrochloride Fenspiride HCl,Pneumorel,Fluiden,Decaspiride Adrenergic Receptor , PDE , Histamine Receptor
Fenspiride hydrochloride (Decaspiride) , an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use in Russia for the therapy of chronic and acute inflammatory ...
T10091 Anti-inflammatory agent 1 Others
Anti-inflammatory agent 1 is an anti-inflammatory compound.
T40380 17α-Hydroxyprogesterone acetate Others
17α-Hydroxyprogesterone acetate possesses progestational activity. 17α-Hydroxyprogesterone acetate shows antiinflammatory effects at the murine maternal-fetal interface.
T64332 Glimepiride sulfonamide Immunology/Inflammation related
Glimepiride sulfonamide is an antiinflammatory agent.
T19694 Hydronidone F351,F-351,F 351 Others
Hydronidone (F-351) is Non-Steroidal Antiinflammatory Drugs. It potentially for the treatment of hepatic fibrosis.
T0270 Hydrocortisone 17-butyrate Cortisol 17-butyrate,Hydrocortisone butyrate Glucocorticoid Receptor , Annexin A , Adrenergic Receptor
Hydrocortisone 17-butyrate (Cortisol 17-butyrate) is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.
T1586 Tenoxicam Ro-12-0068,Tenoxicamum,Mobiflex,Tilcotil COX
Tenoxicam (Tilcotil), an antiinflammatory agent with analgesic and antipyretic properties, is used to treat osteoarthritis and control acute pain.
T15126 Diflumidone R807 Others
Diflumidone, a non-steroidal, is an antiinflammatory drug.
T11196 Enazadrem Lipoxygenase
Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.
T12535 Prednisolone Tebutate Others
Prednisolone Tebutate is a synthetic glucocorticoid, and is an antiinflammatory and immunosuppressant.
T26912 Broperamole
Broperamole, an antiinflammatory, has been found to help with gastrointestinal microbleeding.
T7710L Mofebutazone sodium BRN0213056,BRN 0213056,BRN-0213056
Mofebutazone sodium is, a nonsteroidal antiinflammatory drug (NSAID), is used to treat joint and muscular pain.
T27573 Ibuproxam Ibuproxamum,G-277
Ibuproxam, a nonsteroidal antiinflammatory drug (NSAID), is used for the treatment of musculoskeletal pain, arthritis, and soft-tissue disorders.
T12063 MK-447 Others
MK-447 is a nonsteroidal antiinflammatory agent.
T15774 Losmiprofen Others
Losmiprofen is a nonsteroidal compound of antiinflammatory.
T11271 Fenclozine Others
Fenclozine is a non-steroidal antiinflammatory drug.
T27658 JNJ-10191584 VUF-6002,JNJ10191584
JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammation.
T68926 Indomethacin salicylate
Indomethacin salicylate is an antiinflammatory drug. It has shown remarkable inhibitory effects on carrageenin edema, ultraviolet erythema and adjuvant arthritis.
T60816 Protizinic acid
Protizinic acid inhibits phospholipase A2 (PLA2) with an IC 50 of 210 μM. Protizinic acid has antiinflammatory and antipyretic activity which is an orally active non-steroidal antiinflammatory agent [1] [2].
T40461 Ibuprofen alcohol
Ibuprofen alcohol, a nonsteroidal antiinflammatory drug (NSAID), exhibits very little activity for acid-sensing ion channels (ASICs).
T15021 CV-159 Others
CV-159 is a unique dihydropyridine Ca2+ antagonist with antiinflammatory activities. It has an anti-calmodulin (CaM) action.
T27167 Diclofenac Acyl Glucuronide
Diclofenac Acyl Glucuronide is a major biliary metabolite of Diclofenac (GLXC-07892), a nonsteroidal antiinflammatory drug and COX inhibitor.
T11998 Meloxicam-d3 Meloxicam D4 Others
Meloxicam D4 is deuterium labeled Meloxicam. Meloxicam is a non-steroidal antiinflammatory agent, inhibits COX activity,(Target:COX-1; IC50: 36.6 μM ;(Target:COX-2; IC50: 0.49 μM).
T69491 (E/Z)-Ensifentrine
(E/Z)-Ensifentrine is a potent and selective PDE3/4 inhibitor. (E/Z)-Ensifentrine acts as a long-acting inhibitor of the phosphodiesterase enzymes PDE-3 and PDE-4, producing both bronchodilator and antiinflammatory effec...

Compounds

DHODH-IN-11
T11020
Synonym:
Target: Dehydrogenase, DNA/RNA Synthesis
Etalocib
T22358
Synonym: LY293111,VML295
Target: Apoptosis, Leukotriene Receptor, LTR
Anti-Inflammatory Peptide 1 Acetate
T21606L
Synonym: Anti-Inflammatory Peptide 1 Acetate(118850-70-8 Free base)
Target: Phospholipase
Itaconate-alkyne
T41302
Synonym: ITalk
Target: Others
SC-26196
T12856
Synonym:
Target: Others
Betamethasone valerate
T1163
Synonym: Betnovate,Betaderm,Betamethasone 17-valerate,Luxiq
Target: Glucocorticoid Receptor
Fenspiride hydrochloride
T0383
Synonym: Fenspiride HCl,Pneumorel,Fluiden,Decaspiride
Target: Adrenergic Receptor, PDE, Histamine Receptor
Anti-inflammatory agent 1
T10091
Synonym:
Target: Others
17α-Hydroxyprogesterone acetate
T40380
Synonym:
Target: Others
Glimepiride sulfonamide
T64332
Synonym:
Target: Immunology/Inflammation related
Hydronidone
T19694
Synonym: F351,F-351,F 351
Target: Others
Hydrocortisone 17-butyrate
T0270
Synonym: Cortisol 17-butyrate,Hydrocortisone butyrate
Target: Glucocorticoid Receptor, Annexin A, Adrenergic Receptor
Tenoxicam
T1586
Synonym: Ro-12-0068,Tenoxicamum,Mobiflex,Tilcotil
Target: COX
Diflumidone
T15126
Synonym: R807
Target: Others
Enazadrem
T11196
Synonym:
Target: Lipoxygenase
Prednisolone Tebutate
T12535
Synonym:
Target: Others
Broperamole
T26912
Synonym:
Target:
Mofebutazone sodium
T7710L
Synonym: BRN0213056,BRN 0213056,BRN-0213056
Target:
Ibuproxam
T27573
Synonym: Ibuproxamum,G-277
Target:
MK-447
T12063
Synonym:
Target: Others
Losmiprofen
T15774
Synonym:
Target: Others
Fenclozine
T11271
Synonym:
Target: Others
JNJ-10191584
T27658
Synonym: VUF-6002,JNJ10191584
Target:
Indomethacin salicylate
T68926
Synonym:
Target:
Protizinic acid
T60816
Synonym:
Target:
Ibuprofen alcohol
T40461
Synonym:
Target:
CV-159
T15021
Synonym:
Target: Others
Diclofenac Acyl Glucuronide
T27167
Synonym:
Target:
Meloxicam-d3
T11998
Synonym: Meloxicam D4
Target: Others
(E/Z)-Ensifentrine
T69491
Synonym:
Target:
Cat No. Product Name Synonyms Targets
TN1006 Tirucallol NOS , NO Synthase , Prostaglandin Receptor
Tirucallol is an antiinflammatory agent isolated from Euphorbia lactea.Tirucallol exerts a topical anti-inflammatory effect in vivo, via a mechanism of action related to the neutrophil migration.
TN1712 Gossypin NF-κB , S6 Kinase
Gossypin has antidiabetic, antioxdiant, anticonvulsant, anti-allergic, antiinflammatory, antinociceptive, cytotoxic and antibacterial activities; it inhibits the NF-kappaB activation pathway, which may explain its role i...
T6S2384 Poliumoside Reductase
Poliumoside is a natural compound which exhibits significant inhibition of advanced glycation end product formation with IC50 value of 4.6-25.7 μM, it also exhibits great inhibitory effects on rat lens aldose reductase w...
TL0007 Bisdemethoxycurcumin Curcumin III,Didemethoxycurcumin Epigenetic Reader Domain , Wnt/beta-catenin
Bisdemethoxycurcumin (Curcumin III) is a natural demethoxy derivative of curcumin. It is a potent activator of macrophage phagocytosis, interacting with 1α, 25-dihydroxy vitamin D3 to stimulate amyloid-β clearance by mac...
T3S0153 Xanthatin Apoptosis , VEGFR , Lipoxygenase , Wnt/beta-catenin , Antibacterial
1. Xanthatin has cytotoxic activity. 2. Xanthatin has antibacterial and antifungal activies against MRSA. 3. Xanthatin may have therapeutic potential against NSCLC. 4. Xanthatin can inhibit murine melanoma B16-F1 cell pr...
T8293 γ-Tocopherol (+)-γ-Tocopherol COX
(+)-γ-Tocopherol ((+)-γ-Tocopherol) is one of the naturally occurring forms of Vitamin E. It is the most abundant Tocopherol in soybean and corn oils.
T6S1369 Vitexin Apigenin-8-C-glucoside Antioxidant
1. Vitexin has antinociceptive and antispasmodic activities. 2. Vitexin exhibits a prominent first-pass effect. 3. Vitexin has antioxidant, antimyeloperoxidase, and α-glucosidase inhibitory activities. 4. Vitexin can eit...
TN1563 Dehydropachymic acid Autophagy , Immunology/Inflammation related
Dehydropachymic acid shows antiinflammatory activity.
T5783 Rosamultin Antioxidant , HIV Protease
Rosamultin has antioxidant, antiinflammatory/antinociceptive properties,and has anti-human immunodeficiency virus (HIV) activity.
TN1490 Chrysoeriol ERK , p38 MAPK , Akt
Chrysoeriol has antioxidant, antiinflammatory, antitumor, antimicrobial, antiviral, and free radical scavenging activities, it also shows selective bronchodilator effect.
T3021 Bulleyaconitine A Bulleyaconi cine A Sodium Channel
Bulleyaconitine A (Bulleyaconi cine A), an analgesic and antiinflammatory drug isolated from Aconitum plants, has several potential targets, such as voltage-gated Na+ channels.
TN1047 Ingenol mebutate Ingenol 3-Angelate,PEP005 gp120/CD4 , HIV Protease , PKC
Ingenol mebutate (Ingenol 3-Angelate) is a potent activator of PKC subtypes including PKC-α, PKC-β, PKC-γ, PKC-δ, and PKC-ε with Kis of 0.3, 0.105, 0.162, 0.376, and 0.171 nM. Ingenol mebutate exhibits antiinflammatory a...
T6S0627 Mesaconitine TNF
1. Mesaconitine has antiinflammatory activity. 2. Mesaconitine has antinociceptive activity through cyclic AMP and stimulation of the central β-adrenergic system.
T0492 Dimethyl fumarate DMF Reactive Oxygen Species , HIV Protease , Nrf2 , Endogenous Metabolite , Autophagy
Dimethyl fumarate (DMF), a fumarate derivative, is used as antiinflammatory and immunomodulatory agent.
TCS0862 P-Anisic acid 4-Methoxybenzoic acid,Draconic Acid,4-Anisic Acid Endogenous Metabolite , Antibacterial
1. 4-Methoxybenzoic acid could be used as raw material in cosmetic and dermatologic products and/or aroma components in foodstuffs, it has antiinflammatory and antimicrobial activities.
TN4660 Niranthin Anti-infection , HBV , PAFR , Topoisomerase
Niranthin is a potent anti-leishmanial agent, inhibits the relaxation activity of heterodimeric type IB topoisomerase of L. donovani and acts as a non-competitive inhibitor interacting with both subunits of the enzyme. N...
TN1249 3-Epiursolic acid Cysteine Protease , Immunology/Inflammation related
3-Epiursolic acid may have antiinflammatory activity, it shows inhibition on Cathepsins L (catL), the IC50 value of 6.5 μM, cathepsins L (catL) and B play an important role in tumor progression and have been considered p...
T2838 Naringenin Naringetol,S-Dihydrogenistein,Pelargidanon,Salipurol,NSC 11855,NSC 34875 P450 , Influenza Virus , Reactive Oxygen Species , Endogenous Metabolite , PPAR
Naringenin (NSC-11855) is a flavanone that is considered to have a bioactive effect on human health as antioxidant, free radical scavenger, antiinflammatory, carbohydrate metabolism promoter, immunity system modulater. T...
T2897 (Rac)-Shikonin (±)-Shikonin,Alkanet extract,Anchusin,Anchusa acid Others
(Rac)-Shikonin (Anchusin) is a natural red naphthoquinone pigment, has antimicrobial, anti-tumor, and anti-inflammatory effects; a purified shikonin preparation is widely used for the production of medicinals, cosmetics,...
TN1413 Atranorin Endogenous Metabolite , NO Synthase , Ras
Atranorin shows significant antinociceptive and antiinflammatory activities, it has a relevant redox-active action, acting as a pro-oxidant or antioxidant agent depending on the radical, also, it will exert cytoprotectiv...
T3836 Eudesmin MAPK , S6 Kinase
Eudesmin shows antiinflammatory, neuritogenic, anticonvulsant and sedative effects, the mechanism of eudesmin may be related to up-regulation of GABAA and GAD65 expressions, and anti-apoptosis of neuron the in brain.50 m...
TN2080 Pinoresinol (+)-Pinoresinol Apoptosis , NF-κB , CDK , p53
Pinoresinol ((+)-Pinoresinol) has antiinflammatory, hepatoprotective, and fungicidal activities, it can protect pial microcirculation from I-reperfusion injury, to increase nitric oxide release and to reduce oxidative st...
T4958 (-)-Alkannin Alkannin,Shikonin Apoptosis , PI3K
(-)-Alkannin (Shikonin) is a natural red naphthoquinone pigment, has antimicrobial, anti-tumor, and anti-inflammatory effects; a purified shikonin preparation is widely used for the production of medicinals, cosmetics, a...
T4S0145 Corylifol A Corylinin hCE , STAT , UGT
1. Corylifol A (Corylinin) displays cytotoxic activity against HepG2 and Hep3B hepatocellular carcinoma cell lines, with IC50 values of 4.6 and 13.5 ug/ml, respectively. 2. Corylifol A and Biochanin A can be the potentia...
TN3436 Ar-Curcumene Others
ar-Curcumene has antiinflammatory activity, it could be used as antiinflammatory drugs in respiratory infections. ar-Curcumene is effective as oviposition deterrents against Anopheles stephensi, Aedes aegypti, and Culex ...
TN2002 Obovatol BCL , Caspase , JAK
Obovatol has antioxidant, neuroprotective, antiinflammatory, antithrombotic and antitumour effects, it is a potent NF-κB inhibitors for Alzheimer's disease treatment.
T4S1472 Cucurbitacin S
Cucurbitacins from Wilbrandia ebracteata have analgesic effects. Cucurbitacin S has anticancer and antiinflammatory activities.
TN3620 Celaphanol A NF-κB
Celaphanol A shows moderate inhibition in both NF-κB activation and nitric oxide production, suggests that it is a possible inhibitor of the NF-kappaB pathway and has antiinflammatory activity.
TN7116 6'-Hydroxy-3,4,2',3',4'-pentamethoxychalcone Others
6'-Hydroxy-3,4,2',3',4'-pentamethoxychalcone is an alkenylphenol from Piper obliquum with antiinflammatory and antibacterial activities.
TN3444 Aristolactam BII HIV Protease
Aristolactam BII exhibits antimicrobial and antiinflammatory activity, it shows significant activity towards DPPH radical scavenging and potent inhibitory effects against tyrosinase mushroom. Aristolactam BII also exerts...
TN1080 Kaji-ichigoside F1
Kaji-ichigoside F1 shows antiinflammatory/antinociceptive action in acetic acid-induced writhing and hot plate testing and in a carrageenan-induced paw edema model in mice and rats. Kaji-ichigoside F1 exhibits in vivo he...
TN4648 Nepetoidin B IL Receptor , p38 MAPK , TNF , NOS , NF-κB , COX , Antibacterial , JNK , Antifection , Antifungal
Nepetoidin B has anti-fungal, anti-bacterial, and antiinflammatory effects, it can inhibit LPS-stimulated NO production possibly via modulation of iNOS mediated by MKP-5/NF-κB pathways in RAW 264.7 cells.

Natural Products

Tirucallol
TN1006
Synonym:
Target: NOS, NO Synthase, Prostaglandin Receptor
Gossypin
TN1712
Synonym:
Target: NF-κB, S6 Kinase
Poliumoside
T6S2384
Synonym:
Target: Reductase
Bisdemethoxycurcumin
TL0007
Synonym: Curcumin III,Didemethoxycurcumin
Target: Epigenetic Reader Domain, Wnt/beta-catenin
Xanthatin
T3S0153
Synonym:
Target: Apoptosis, VEGFR, Lipoxygenase, Wnt/beta-catenin, Antibacterial
γ-Tocopherol
T8293
Synonym: (+)-γ-Tocopherol
Target: COX
Vitexin
T6S1369
Synonym: Apigenin-8-C-glucoside
Target: Antioxidant
Dehydropachymic acid
TN1563
Synonym:
Target: Autophagy, Immunology/Inflammation related
Rosamultin
T5783
Synonym:
Target: Antioxidant, HIV Protease
Chrysoeriol
TN1490
Synonym:
Target: ERK, p38 MAPK, Akt
Bulleyaconitine A
T3021
Synonym: Bulleyaconi cine A
Target: Sodium Channel
Ingenol mebutate
TN1047
Synonym: Ingenol 3-Angelate,PEP005
Target: gp120/CD4, HIV Protease, PKC
Mesaconitine
T6S0627
Synonym:
Target: TNF
Dimethyl fumarate
T0492
Synonym: DMF
Target: Reactive Oxygen Species, HIV Protease, Nrf2, Endogenous Metabolite, Autophagy
p-Anisic acid
TCS0862
Synonym: 4-Methoxybenzoic acid,Draconic Acid,4-Anisic Acid
Target: Endogenous Metabolite, Antibacterial
Niranthin
TN4660
Synonym:
Target: Anti-infection, HBV, PAFR, Topoisomerase
3-Epiursolic acid
TN1249
Synonym:
Target: Cysteine Protease, Immunology/Inflammation related
Naringenin
T2838
Synonym: Naringetol,S-Dihydrogenistein,Pelargidanon,Salipurol,NSC 11855,NSC 34875
Target: P450, Influenza Virus, Reactive Oxygen Species, Endogenous Metabolite, PPAR
(Rac)-Shikonin
T2897
Synonym: (±)-Shikonin,Alkanet extract,Anchusin,Anchusa acid
Target: Others
Atranorin
TN1413
Synonym:
Target: Endogenous Metabolite, NO Synthase, Ras
Eudesmin
T3836
Synonym:
Target: MAPK, S6 Kinase
Pinoresinol
TN2080
Synonym: (+)-Pinoresinol
Target: Apoptosis, NF-κB, CDK, p53
(-)-Alkannin
T4958
Synonym: Alkannin,Shikonin
Target: Apoptosis, PI3K
Corylifol A
T4S0145
Synonym: Corylinin
Target: hCE, STAT, UGT
ar-Curcumene
TN3436
Synonym:
Target: Others
Obovatol
TN2002
Synonym:
Target: BCL, Caspase, JAK
Cucurbitacin S
T4S1472
Synonym:
Target:
Celaphanol A
TN3620
Synonym:
Target: NF-κB
6'-Hydroxy-3,4,2',3',4'-pentamethoxychalcone
TN7116
Synonym:
Target: Others
Aristolactam BII
TN3444
Synonym:
Target: HIV Protease
Kaji-ichigoside F1
TN1080
Synonym:
Target:
Nepetoidin B
TN4648
Synonym:
Target: IL Receptor, p38 MAPK, TNF, NOS, NF-κB, COX, Antibacterial, JNK, Antifection, Antifungal

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPK-00765 Pentraxin 2/SAP Protein, Human, Recombinant (hFc) Human HEK293
Pentraxin-2 (PTX-2), also known as serum amyloid P component (SAP/APCS), is a constitutive, antiinflammatory, innate immune plasma protein whose circulating level is decreased in chronic human fibrotic recombinant human ...
TMPK-00113 Pentraxin 2/SAP Protein, Mouse, Recombinant (hFc) Mouse HEK293
Pentraxin-2 (PTX-2), also known as serum amyloid P component (SAP/APCS), is a constitutive, antiinflammatory, innate immune plasma protein whose circulating level is decreased in chronic human fibrotic recombinant human ...
TMPY-02138 Uteroglobin Protein, Human, Recombinant (His) Human HEK293
Uteroglobin (UG), also known as Secretoglobin 1A member 1 (SCGB1A1), Blastokinin, Clara cell secretor protein (CCSP) or Clara cell-specific 10-kDa protein (CC10), is the founding member of the secretoglobin family of sma...
TMPJ-00021 LGALS1 Protein, Human, Recombinant (His) Human E. coli
Galectin-1 is a member of growing family of evolutionary conserved animal lectins. Galectin-1 is widely expressed in many cells and tissues. Galectins consists of a Galectin domain and two Beta-galactoside binding domain...
TMPY-02328 Uteroglobin Protein, Mouse, Recombinant (His) Mouse HEK293
Uteroglobin (UG), also known as Secretoglobin 1A member 1 (SCGB1A1), Blastokinin, Clara cell secretor protein (CCSP) or Clara cell-specific 10-kDa protein (CC10), is the founding member of the secretoglobin family of sma...
Cat No. Product Name
L4710 Nonsteroidal Anti-Inflammatory Compound Library

530 compounds
530 non-steroidal anti-inflammatory compounds for high-throughput and high-content screening.
L6710 Anti-Inflammatory Traditional Chinese Medicine Compound Library

1260 compounds
A collection of 1260 TCM monomers with anti-inflammatory activity or targeting molecular therapeutic targets in inflammation, a powerful tool for drug discovery and mechanism study;
L6120 Flavonoid Natural Product Library

477 compounds
A unique collection of 477 flavonoids can be used for high throughput and high content screening;
TargetMol