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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T76653 | Polybia-MP1 | ||
Polybia-MP1 is an antimicrobial mastoparan peptide [1] . | |||
T80585 | Anti-Mouse GM-CSF Antibody (MP1-22E9) | c-Fms | |
Anti-Mouse GM-CSF Antibody is a rat-derived IgG2a isotype inhibitor that targets mouse granulocyte-macrophage colony-stimulating factor (GM-CSF). | |||
T69977 | BC-1485 | ||
BC-1485 is a first-in-class inhibitor of Fibrosis-inducing E3 ligase 1 (FIEL1 ), which disrupts FIEL1-directed PIAS4 ubiquitination. | |||
T71901 | MP-1 | ||
MP-1 is a covalent inhibitor of fumarate hydratase (FH) that exhibits cytotoxicity dependent on FH. MP-1 engages a functional cysteine in the Zn-finger domain of the tRNA methyltransferase enzyme TRMT1. | |||
T3983 | TMP195 | TFMO 2,TMP 195 | HDAC |
TMP195 (TFMO 2) is a selective class IIa histone deacetylase (HDAC) inhibitor. | |||
T78269 | Anti-Mouse PD-1 Antibody (RMP1-14) | PD-1/PD-L1 | |
RMP1-14 is an IgG1-like immunoglobulin and anti-Mouse PD-1 antibody that blocks PD-1/PD-L1 signaling. | |||
T16124 | MMP13-IN-3 | MMP | |
MMP13-IN-3 is >1000 selective over other MMPs. MMP13-IN-3 is an effective, selective, and orally active MMP-13 inhibitor (IC50=1 nM) for the potential treatment of osteoarthritis. | |||
T76244 | Amp1EP9 | ||
Amp1EP9, an antimicrobial peptide, serves as a potent and non-toxic candidate for the development of effective antimicrobial agents. It holds promise for research into multidrug-resistant bacterial infections [1]. | |||
T82063 | Integrin signaling inhibitor, mP13 | ||
Integrin Signaling Inhibitor mP13 is a compound that impedes both inside-out and outside-in integrin-mediated signaling processes, such as fibrinogen binding, platelet adhesion, and clot retraction [1]. | |||
T83487 | [Pmp1,Tyr(OEt)2] AVP | ||
[Pmp1,Tyr(OEt)2] AVP, a linear analog of the cyclic arginine vasopressin (AVP) antagonist, retains the antagonistic properties of its parent compound while featuring modified phenylalanine (Pmp) and diethyltyrosine (Tyr(... | |||
T41079 | MMP13-IN-2 | MMP13-IN-2 | |
MMP13-IN-2 is a highly potent, selective, and orally active inhibitor of MMP-13. It demonstrates exceptional potency against MMP-13, with an IC50 value of 0.036 nM, and exhibits selectivities greater than 1,500-fold over... | |||
T78774 | MMP13-IN-4 | MMP | |
MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1]. | |||
T72306 | Mycobacterial Zmp1-IN-1 | ||
Mycobacterial Zmp1-IN-1, a zinc metalloprotease-1 (Zmp1) inhibitor, demonstrates dose-dependent anti-mycobacterial activity against Mtb H37Ra, making it suitable for tuberculosis (TB) research. | |||
T80336 | DFTamP1 | ||
DFTamP1 is an antimicrobial peptide that exhibits activity against Staphylococcus aureus USA300, with a minimum inhibitory concentration (MIC) of 3.1 μM [1]. | |||
T80282 | CPcAMP1/26 | ||
cPcAMP1/26, an antimicrobial peptide, exhibits potent bactericidal activity against A. hydrophila and S. aureus by inducing depolarization of the bacterial plasma membrane and elevating intracellular ROS (Reactive Oxygen... | |||
T78775 | MMP13-IN-5 | MMP | |
MMP13-IN-5 (compound 13m) is a potent, selective MMP-2/MMP-13 inhibitor with IC50 values of 3.6 μM for MMP-2 and 14.6 μM for MMP-13, implicated in the pathology of osteoarthritis (OA) [1]. |