T3593 |
Src Inhibitor 1
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Src Kinase Inhibitor 1,Src-l1 |
Src
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Src Inhibitor 1 是一种选择性的、高效的、ATP-竞争性的双位点 Src 酪氨酸激酶抑制剂,能够抑制 Src (IC50:44 nM) 和 Lck (IC50:88 nM)。 |
TP2289L |
RR-src acetate
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RR-src acetate(81156-93-6 Free base) |
Others
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RR-src acetate 是一种合成肽,来源于 pp60src 中磷酸化位点周围的氨基酸序列。 |
T13000 |
Src Inhibitor 3
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Others
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Src
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Src Inhibitor 3 是一种有效的 c-terminal Src 激酶抑制剂(CSK HTRF 中 IC50 <3 nM,Caliper 中 IC50 <4 nM)。 Src Inhibitor 3 增加由 T 细胞受体信号传导诱... |
TP2137L |
Pp60 c-src (521-533) (phosphorylated) acetate
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Others
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pp60 c-src (521-533) (phosphorylated) acetate 是粘着斑形成和细胞扩散的调节剂。它还调节细胞运动,是由促运动透明质酸受体 RHAMM 触发的信号通路中的关键成分。 |
T39185 |
Pp60 (v-SRC) Autophosphorylation Site, Phosphorylated
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pp60 (v-SRC) Autophosphorylation Site, Phosphorylated |
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pp60 (v-SRC) Autophosphorylation Site, Phosphorylated is a phosphorylated peptide derived from an EGFR substrate. It ser... |
T39149 |
Src Optimal Peptide Substrate
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Src Optimal Peptide Substrate, a highly specific substrate of Src, serves as a reliable indicator of Src activity. It en... |
TP2289 |
RR-src
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Others
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Tyrosine kinase substrate peptide |
T76391 |
P60c-src substrate II
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p60c-src substrate II 是酪氨酸激酶pp60c-src 的高效五肽底物。 |
T11745 |
KB SRC 4
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Others
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KB SRC 4 has antitumor activity. KB SRC 4 is a potent, and highly selective c-Src inhibitor, with a Ki of 44 nM and a Kd... |
T13062 |
T338C Src-IN-2
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Others
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T338C Src-IN-2 is a potent mutant inhibitor of c-Src T338C kinase(IC50 of 317 nM). T338C Src-IN-2 also inhibits T338C/V3... |
T1811 |
WH-4-023
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KIN001-112,Dual LCK/SRC inhibitor,KIN112 |
Src
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WH-4-023 是选择性Lck 和Src 抑制剂,它们的 IC50 分别为 2 nM、6 nM,对p38α 和 KDR 作用效果稍弱。 |
T13061 |
T338C Src-IN-1
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Others
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T338C Src-IN-1 is a potent mutant-Src T338C inhibitor(T338C,IC50=111 nM relative to WT c-Src (10-fold increase)). |
TP2137 |
Pp60 c-src (521-533) (phosphorylated)
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Peptide corresponding to the pp60c-src carboxy terminal regulatory domain; phosphorylated at Tyr527. Binds to pp60c-src ... |
T38439 |
DC-Srci-6649
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DC-Srci-6649 is a potent and selective inhibitor of c-Src kinase, effectively blocking its phosphorylation and stabilizi... |
T8499 |
ECF506
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Src
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eCF506 是一种高效的、口服具有活力的非受体酪氨酸激酶Src 抑制剂,其IC50<0.5 nM。 |
TQ0132 |
A 419259 trihydrochloride
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RK 20449 trihydrochloride |
Src
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A 419259 trihydrochloride 是一种 Src 家族激酶抑制剂,能够抑制 Src (IC50:9 nM)、Lck (IC50:3 nM)、Lyn (IC50:3 nM)。 |
T3063 |
PD173955
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PD-173955,PD 173955 |
Bcr-Abl
,
Apoptosis
,
Src
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PD173955是一种Src 激酶家族选择性抑制剂,对Src、Yes 和Abl 激酶IC50值约为22nM, 对 FGFRα 的效力较低,对InsR 和PKC 无活性。 |
T0152 |
Bosutinib
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SKI-606,伯舒替尼 |
Bcr-Abl
,
Src
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Autophagy
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Bosutinib 是一种合成的喹诺酮衍生物和双激酶抑制剂,靶向 Abl 和 Src 激酶的 IC50分别为 1 nM 和 1.2 nM。 |
T15675 |
Tirbanibulin Mesylate
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KX2-391 Mesylate,KX01 Mesylate |
Src
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Microtubule Associated
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Tirbanibulin Mesylate 是一种 Src 抑制剂,靶向 Src 的肽底物位点。在肿瘤细胞中,GI50值为 9-60 nM。 |
T6345 |
Tirbanibulin
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KX2-391,KX-01 |
Src
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Microtubule Associated
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KX2-391 是一种高度选择性的 Src 激酶抑制,靶向 Src 的多肽底物结合位点,对多种癌症有疗效。 |