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Targets

Libraries

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Compounds

Cat No. Product Name
T3593 Src Inhibitor 1 Src Kinase Inhibitor 1,Src-l1 Src
Src Inhibitor 1 是一种选择性的、高效的、ATP-竞争性的双位点 Src 酪氨酸激酶抑制剂,能够抑制 Src (IC50:44 nM) 和 Lck (IC50:88 nM)。
TP2289L RR-src acetate RR-src acetate(81156-93-6 Free base) Others
RR-src acetate 是一种合成肽,来源于 pp60src 中磷酸化位点周围的氨基酸序列。
T13000 Src Inhibitor 3 Others , Src
Src Inhibitor 3 是一种有效的 c-terminal Src 激酶抑制剂(CSK HTRF 中 IC50 <3 nM,Caliper 中 IC50 <4 nM)。 Src Inhibitor 3 增加由 T 细胞受体信号传导诱...
TP2137L Pp60 c-src (521-533) (phosphorylated) acetate Others
pp60 c-src (521-533) (phosphorylated) acetate 是粘着斑形成和细胞扩散的调节剂。它还调节细胞运动,是由促运动透明质酸受体 RHAMM 触发的信号通路中的关键成分。
T39185 Pp60 (v-SRC) Autophosphorylation Site, Phosphorylated pp60 (v-SRC) Autophosphorylation Site, Phosphorylated
pp60 (v-SRC) Autophosphorylation Site, Phosphorylated is a phosphorylated peptide derived from an EGFR substrate. It ser...
T39149 Src Optimal Peptide Substrate
Src Optimal Peptide Substrate, a highly specific substrate of Src, serves as a reliable indicator of Src activity. It en...
TP2289 RR-src Others
Tyrosine kinase substrate peptide
T76391 P60c-src substrate II
p60c-src substrate II 是酪氨酸激酶pp60c-src 的高效五肽底物。
T11745 KB SRC 4 Others
KB SRC 4 has antitumor activity. KB SRC 4 is a potent, and highly selective c-Src inhibitor, with a Ki of 44 nM and a Kd...
T13062 T338C Src-IN-2 Others
T338C Src-IN-2 is a potent mutant inhibitor of c-Src T338C kinase(IC50 of 317 nM). T338C Src-IN-2 also inhibits T338C/V3...
T1811 WH-4-023 KIN001-112,Dual LCK/SRC inhibitor,KIN112 Src
WH-4-023 是选择性Lck 和Src 抑制剂,它们的 IC50 分别为 2 nM、6 nM,对p38α 和 KDR 作用效果稍弱。
T13061 T338C Src-IN-1 Others
T338C Src-IN-1 is a potent mutant-Src T338C inhibitor(T338C,IC50=111 nM relative to WT c-Src (10-fold increase)).
TP2137 Pp60 c-src (521-533) (phosphorylated)
Peptide corresponding to the pp60c-src carboxy terminal regulatory domain; phosphorylated at Tyr527. Binds to pp60c-src ...
T38439 DC-Srci-6649
DC-Srci-6649 is a potent and selective inhibitor of c-Src kinase, effectively blocking its phosphorylation and stabilizi...
T8499 ECF506 Src
eCF506 是一种高效的、口服具有活力的非受体酪氨酸激酶Src 抑制剂,其IC50<0.5 nM。
TQ0132 A 419259 trihydrochloride RK 20449 trihydrochloride Src
A 419259 trihydrochloride 是一种 Src 家族激酶抑制剂,能够抑制 Src (IC50:9 nM)、Lck (IC50:3 nM)、Lyn (IC50:3 nM)。
T3063 PD173955 PD-173955,PD 173955 Bcr-Abl , Apoptosis , Src
PD173955是一种Src 激酶家族选择性抑制剂,对Src、Yes 和Abl 激酶IC50值约为22nM, 对 FGFRα 的效力较低,对InsR 和PKC 无活性。
T0152 Bosutinib SKI-606,伯舒替尼 Bcr-Abl , Src , Autophagy
Bosutinib 是一种合成的喹诺酮衍生物和双激酶抑制剂,靶向 Abl 和 Src 激酶的 IC50分别为 1 nM 和 1.2 nM。
T15675 Tirbanibulin Mesylate KX2-391 Mesylate,KX01 Mesylate Src , Microtubule Associated
Tirbanibulin Mesylate 是一种 Src 抑制剂,靶向 Src 的肽底物位点。在肿瘤细胞中,GI50值为 9-60 nM。
T6345 Tirbanibulin KX2-391,KX-01 Src , Microtubule Associated
KX2-391 是一种高度选择性的 Src 激酶抑制,靶向 Src 的多肽底物结合位点,对多种癌症有疗效。
Src Inhibitor 1
T3593
synonym: Src Kinase Inhibitor 1,Src-l1
Target:
RR-src acetate
TP2289L
synonym: RR-src acetate(81156-93-6 Free base)
Target:
Src Inhibitor 3
T13000
synonym:
Target:
pp60 c-src (521-533) (phosphorylated) acetate
TP2137L
synonym:
Target:
pp60 (v-SRC) Autophosphorylation Site, Phosphorylated
T39185
synonym: pp60 (v-SRC) Autophosphorylation Site, Phosphorylated
Target:
Src Optimal Peptide Substrate
T39149
synonym:
Target:
RR-src
TP2289
synonym:
Target:
p60c-src substrate II
T76391
synonym:
Target:
KB SRC 4
T11745
synonym:
Target:
T338C Src-IN-2
T13062
synonym:
Target:
WH-4-023
T1811
synonym: KIN001-112,Dual LCK/SRC inhibitor,KIN112
Target:
T338C Src-IN-1
T13061
synonym:
Target:
pp60 c-src (521-533) (phosphorylated)
TP2137
synonym:
Target:
DC-Srci-6649
T38439
synonym:
Target:
eCF506
T8499
synonym:
Target:
A 419259 trihydrochloride
TQ0132
synonym: RK 20449 trihydrochloride
Target:
PD173955
T3063
synonym: PD-173955,PD 173955
Target:
Bosutinib
T0152
synonym: SKI-606,伯舒替尼
Target:
Tirbanibulin Mesylate
T15675
synonym: KX2-391 Mesylate,KX01 Mesylate
Target:
Tirbanibulin
T6345
synonym: KX2-391,KX-01
Target:
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