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Perlolyrine

Name: Perlolyrine
Brand: TargetMol
SKU: TN6548
Price: 48 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. TN6548Cas No. 29700-20-7

Alias Tribulusterine

Perlolyrine (Tribulusterine) is a naturally occurring alkaloid with molecular docking capacity (-5.73 to -6.59 kJ/mol) with MAPK1, MAPK14, and SRC, with potential anticancer and anti-inflammatory effects.

Perlolyrine

🥰Excellent

Purity: 99.62%

Catalog No. TN6548Alias TribulusterineCas No. 29700-20-7

Pack Size	Price	Availability
1 mg	$48	In Stock
5 mg	$117	In Stock
10 mg	$187	In Stock
25 mg	$376	In Stock
50 mg	$591	In Stock
100 mg	$969	In Stock
200 mg	$1,280	In Stock

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Purity:99.62%

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COA LCMS HNMR

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity

Description	Perlolyrine (Tribulusterine) is a naturally occurring alkaloid with molecular docking capacity (-5.73 to -6.59 kJ/mol) with MAPK1, MAPK14, and SRC, with potential anticancer and anti-inflammatory effects.
In vitro	Perlolyrine inhibits α-MSH-induced melanogenesis in B16F10 mouse melanoma cells in a dose-dependent manner (5-25 μM, 48 h). At 25 μM, Perlolyrine reduces melanin content by over 50% without affecting cell viability. Perlolyrine also suppresses the expression of melanogenesis-related genes such as MITF, tyrosinase, and TRP-1[1].
Alias	Tribulusterine

Chemical Properties

Molecular Weight	264.28
Formula	C₁₆H₁₂N₂O₂
Cas No.	29700-20-7
Smiles	OCC=1OC(=CC1)C2=NC=CC=3C4=CC=CC=C4NC23
Relative Density.	1.382 g/cm3 (Predicted)

Storage & Solubility Information

Storage

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 80 mg/mL (302.71 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.7839 mL	18.9193 mL	37.8387 mL	189.1933 mL
5 mM	0.7568 mL	3.7839 mL	7.5677 mL	37.8387 mL
10 mM	0.3784 mL	1.8919 mL	3.7839 mL	18.9193 mL
20 mM	0.1892 mL	0.9460 mL	1.8919 mL	9.4597 mL
50 mM	0.0757 mL	0.3784 mL	0.7568 mL	3.7839 mL
100 mM	0.0378 mL	0.1892 mL	0.3784 mL	1.8919 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc