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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Cat. No. Product name CAS No. Purity Chemical Structure
T15565 Imetit dihydrobromide 32385-58-3 98%
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
T10911 H3 receptor antagonist 1 935840-13-4 98%
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
TN2895 3,5-Dicaffeoyl-epi-quinic acid 879305-14-3 98%
3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
T11324 FRG8701 108498-50-6 98%
FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
T3037 Cyclizine dihydrochloride 5897-18-7 98%
Cyclizine Dihydrochloride is a histamine H1 antagonist. It is given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in mo...
T12054 MK-0249 862309-06-6 98%
MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
T19604 WZ4141 1222776-76-2 98%
WZ4141 is an intermediate in compound synthesis.
T10794 Chlorcyclizine hydrochloride 14362-31-3 98%
Chlorcyclizine hydrochloride is an antagonist of histamine H1.
TN3062 4'-O-Methylnyasol 79004-25-4 98%
4'-O-Methylnyasol may have potential to be developed as medicines for the treatment of allergies by inhibiting the activation of mast cells.
T10769 Cetirizine D4 1219803-84-5 98%
Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
TN1913 Marmin 14957-38-1 98%
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
T11531 H3R-IN-1 Hydrochloride 2319790-07-1 98%
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
T13040 SUN 1334H 607736-84-5 98%
SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
T12756 ROS 234 dioxalate 1781941-93-2 98%
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
TN5279 Zeorin 22570-53-2 98%
Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
T19234 Cetirizine D8 dihydrochloride 2070015-04-0 98%
Cetirizine D8 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagoni...
T6562 Latrepirdine dihydrochloride 97657-92-6 98%
Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
T11532 H4R antagonist 1 1429375-54-1 98%
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
TN4918 Roseoside 54835-70-0 98%
Roseoside possesses strong antioxidant properties, inhibiting lipid oxidation by 86.4, at 50 microg/mL. Roseoside has insulinotropic activity, enhances insulin r...
T10575 BMY-25271 78441-82-4 98%
BMY-25271 is an antagonist of histamine H2 receptor.
Imetit dihydrobromide
T15565
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
H3 receptor antagonist 1
T10911
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
3,5-Dicaffeoyl-epi-quinic acid
TN2895
3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
FRG8701
T11324
FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
Cyclizine dihydrochloride
T3037
Cyclizine Dihydrochloride is a histamine H1 antagonist. It is given by mouth or parenterally for the control of postoperative and drug-induced vomiting and in mo...
MK-0249
T12054
MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
WZ4141
T19604
WZ4141 is an intermediate in compound synthesis.
Chlorcyclizine hydrochloride
T10794
Chlorcyclizine hydrochloride is an antagonist of histamine H1.
4'-O-Methylnyasol
TN3062
4'-O-Methylnyasol may have potential to be developed as medicines for the treatment of allergies by inhibiting the activation of mast cells.
Cetirizine D4
T10769
Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
Marmin
TN1913
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
H3R-IN-1 Hydrochloride
T11531
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
SUN 1334H
T13040
SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
ROS 234 dioxalate
T12756
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
Zeorin
TN5279
Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
Cetirizine D8 dihydrochloride
T19234
Cetirizine D8 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagoni...
Latrepirdine dihydrochloride
T6562
Latrepirdine is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihi...
H4R antagonist 1
T11532
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
Roseoside
TN4918
Roseoside possesses strong antioxidant properties, inhibiting lipid oxidation by 86.4, at 50 microg/mL. Roseoside has insulinotropic activity, enhances insulin r...
BMY-25271
T10575
BMY-25271 is an antagonist of histamine H2 receptor.
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