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Cyproheptadine hydrochloride sesquihydrate (Synonyms: Periactin hydrochloride)

Name: Cyproheptadine hydrochloride sesquihydrate
Brand: TargetMol
SKU: T0174
Price: 29 USD
Availability: InStock
Rating: 5 (10 reviews)

Catalog No. T0174 Copy Product Info

Purity: 99.99%

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Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.

Cyproheptadine hydrochloride sesquihydrate

Copy Product Info

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Catalog No. T0174

Synonyms Periactin hydrochloride

Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.

Cas No. 41354-29-4

Pack Size	Price	USA Stock	Global Stock	Quantity
500 mg	$29	In Stock	-

For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)

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For research use only—not for human use. No sales to individuals. Use as intended only.

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Purity:99.99%

Appearance:Solid

Color:White

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COA LCMS

Product Introduction

Bioactivity

Description	Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
Targets&IC50	5-HT2:0.6 nM, SETD7/9:1 μM
Synonyms	Periactin hydrochloride

Chemical Properties

Molecular Weight	341.88
Formula	C₂₁H₂₄ClNO
Cas No.	41354-29-4
Smiles	O.O.O.Cl.Cl.CN1CC\C(CC1)=C1/c2ccccc2C=Cc2ccccc12.CN1CC\C(CC1)=C1/c2ccccc2C=Cc2ccccc12
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: < 1 mg/mL (insoluble or slightly soluble)

DMSO: 70 mg/mL (204.75 mM), Sonication is recommended.

Ethanol: 20 mg/mL (58.5 mM), Sonication is recommended.

In Vivo Formulation

10% DMSO+40% PEG300+5% Tween 80+45% Saline: 2.5 mg/mL (7.31 mM), Sonication is recommended.

Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.

Solution Preparation Table

Ethanol/DMSO

	1mg	5mg	10mg	50mg
1 mM	2.9250 mL	14.6250 mL	29.2500 mL	146.2501 mL
5 mM	0.5850 mL	2.9250 mL	5.8500 mL	29.2500 mL
10 mM	0.2925 mL	1.4625 mL	2.9250 mL	14.6250 mL
20 mM	0.1463 mL	0.7313 mL	1.4625 mL	7.3125 mL
50 mM	0.0585 mL	0.2925 mL	0.5850 mL	2.9250 mL

DMSO

	1mg	5mg	10mg	50mg
100 mM	0.0293 mL	0.1463 mL	0.2925 mL	1.4625 mL

Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density.

Calculator

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

SETD9SETD7HistoneMethyltransferaseHistone MethyltransferaseHistamineReceptorHistamine ReceptorCyproheptadine hydrochloride sesquihydrate5HTReceptor5-HT25-HT Receptor5HT Receptor

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