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voltage

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    269
    TargetMol | Inhibitors_Agonists
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    TargetMol | Inhibitors_Agonists
Licarbazepine
​10,11-hydroxy-10,11 Dihydrocarbamezer
T780629331-92-8
Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial seizures and bipolar disorders.
  • $44
In Stock
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QTY
Dizocilpine
MK-801
T625977086-21-6
Dizocilpine (MK-801) is a selective non-competitive NMDA receptor antagonist with a Kd of 37.2 nM that exhibits anticonvulsant effects. It acts by binding to a site within the NMDA-associated ion channel, blocking the flow of Ca²⁺, and is commonly used to establish schizophrenia models.
  • $35
In Stock
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QTY
Dizocilpine Maleate
MK 801, Dizocilpine hydrogen maleate, (+)-Mk-801 Hydrogen Maleate, (+)-MK 801 maleate, (+)-MK 801 (Maleate)
T332077086-22-7
Dizocilpine Maleate (MK-801 maleate) is a potent, selective, and non-competitive NMDA receptor antagonist with a Kd value of 37.2 nM. It is commonly used in the treatment of various neurodegenerative diseases in which NMDA receptors may be involved, and can also be used to induce schizophrenia models.
  • $32
In Stock
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Erastin
T1765571203-78-6
Erastin is an iron death activator that acts on the mitochondrial VDAC in a ROS- and iron-dependent manner. Erastin has anti-tumor activity and acts selectively on tumor cells with RAS-carcinogenic mutations.
  • $41
In Stock
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TargetMol | Inhibitor Hot
VBIT-4
T132872086257-77-2
VBIT-4 is a voltage-dependent anion channel 1 (VDAC1) oligomerization inhibitor (Kd: 17 μM). VBIT-4 can be used for therapeutic purposes in apoptosis-associated disorders (such as neurodegenerative and cardiovascular diseases).
  • $68
In Stock
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TargetMol | Inhibitor Hot
Kv3 modulator 1
T117871380696-64-9In house
Kv3 modulator 1 is a voltage-gated potassium channel Kv3 modulator that can be used to study neurologic-level diseases.
  • $373
In Stock
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McN5691
RWJ26240, MCN 5691
T1197999254-95-2In house
McN5691 (RWJ26240) is a voltage-dependent calcium channel blocker with antihypertensive activity that can be used in the study of diseases caused by vascular smooth muscle abnormalities.
  • $293 TargetMol
In Stock
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PF-06305591
PF-6305591
T124241449473-97-5In house
PF-06305591 is an effective and selective blocker of voltage-gated sodium channel NaV1.8 (IC50 = 15 nM).
  • $44
In Stock
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(5R)-BW-4030W92
T13428189013-61-4In house
(5R)-BW-4030W92, the active enantiomer of BW-4030W92, is an orally available, non-selective, voltage-dependent, and use-dependent sodium channel antagonist used in the study of neurological disorders.
  • $700
In Stock
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QTY
E 0747 FA
E 0747 FA(99599-78-7 Free base)
T24021L In house
E 0747 FA is an antiarrhythmic compound that inhibits the voltage of action potential Vmax in Purkinje fibers of porcine heart.E 0747 FA inhibits Na channels in cardiac cells.
  • $195
In Stock
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SAK3
SAK-3, SAK 3
T261741256269-87-0In house
SAK3 is a novel modulator of nAChR activity that enhances T-type voltage-gated Ca2+ channel (T-VGCC) activity, and has potentiating effects on both Cav3.1 and Cav3.3 T-type Ca2+ channel currents.SAK3 is neuroprotective against scopolamine-induced cholinergic dysfunction in human neuroblastoma SH-SY5Y cells.SAK3 is used for the study of memory deficits and Alzheimer's disease. SAK3 can be used to study memory deficits and Alzheimer's disease.
  • $129 TargetMol
In Stock
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Besipirdine
HP 749 free base, P-867493, P867493, HP 749, HP749, P 867493
T26778119257-34-0In house
Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine inhibits voltage-dependent sodium-potassium channels and inhibits biogenic amine uptake.Besipirdine reduces schedule-induced irritability and thirst and enhances cholinergic and adrenergic activity in the CNS in the rat. Besipirdine reduces schedule-induced thirst and enhances cholinergic and adrenergic neurotransmission in the central nervous system.
  • $293
In Stock
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Besipirdine hydrochloride
HP 749 hydrochloride, Besipirdine hydrochloride(119257-34-0 Free base)
T26778L130953-69-4In house
Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine hydrochloride inhibits voltage-dependent sodium-potassium channels and inhibits biogenic amine uptake.Besipirdine hydrochloride reduces schedule-induced thirst and enhances cholinergic and adrenergic neurotransmission in the central nervous system in rats.
  • $195 TargetMol
In Stock
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Hymenidin
T27564107019-95-4In house
Hymenidin, an alkaloid isolated from the Okinawan sponge Hymeniacidon sp. is a 5-hydroxytryptaminergic receptor antagonist and voltage-gated potassium channel inhibitor with potential antiprotozoal effects.It selectively binds to FOXO1 DNA and reduces depolarization-induced elevation of cellular calcium.
  • $2,420
1-2 weeks
Size
QTY
JNJ-26489112
JNJ26489112, JNJ 26489112
T27672871824-55-4In house
JNJ-26489112 is a CNS-active agent and inhibitor of voltage-gated Na+ channels and N-type Ca2+ channels with broad-spectrum anticonvulsant activity in rodents and can be used to study neurological disorders.
  • $195
In Stock
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Atagabalin HCl
PD-0200390 HCl, Atagabalin HCl(223445-75-8 Free base)
T30188L223445-67-8In house
Atagabalin HCl is a novel voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) ligand that affects slow-wave sleep and can be used to treat insomnia.
  • $572
In Stock
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TargetMol | Inhibitor Sale
HSK16149
T602522209104-84-5In house
HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.
  • Inquiry Price
7-10 days
Size
QTY
IEM 1754 2HBr
IEM 1754 dihydrobromide
T6134162831-31-4In house
IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.
  • $30
In Stock
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Elgodipine
T68060119413-55-7In house
Elgodipine significantly reduced the incidence and severity of exercise-induced angina pectoris systemically and was able to inhibit vascular smooth muscle proliferation through a mechanism independent of the expression of the transcription factors c-fos and c-jun. The Elgodipine-induced inhibition was voltage-dependent. Elgodipine is a potential compound for the treatment of angina pectoris.
  • $54
In Stock
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TargetMol | Inhibitor Sale
Flosatidil
T68073113593-34-3In house
Flosatidil is a small molecule voltage-gated calcium channel complex (VDCCs) blocker for the treatment of neurological disorders and cardiovascular diseases, and can be used in the study of angina pectoris.
  • $55
In Stock
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Crobenetine
Crobenetine Free Base, BIII 890
T69795221019-25-6In house
Crobenetine (BIII 890 CL) Free Base is a selective NaV channel blocker that eliminates VTD-induced [Ca2+] elevation.
  • $310
In Stock
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Phenytoin sodium
5,5-Diphenylhydantoin sodium salt, Diphantoine, Dilantin sodium, Diphenylhydantoin Sodium
T0008630-93-3
Phenytoin sodium (Diphantoine) is an inactive stabilizer for voltage-gated sodium channel .
  • $45
In Stock
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Procainamide hydrochloride
Procapan, Procainamide HCl, Pronestyl, Procanbid
T0018614-39-1
Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog of procaine. Procainamide hydrochloride reversibly binds to and blocks activated (open) voltage-gated sodium channels, thereby blocks the influx of sodium ions into the cell, which leads to an increase in threshold for excitation and inhibit depolarization during phase 0 of the action potential.
  • $31
In Stock
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Primidone
Primaclone, Mysoline, NCI-C56360
T0024125-33-7
Primidone (NCI-C56360) is a potent anticonvulsant agent. It is a neuronal voltage-gated sodium channel blocker and has value in the study of epilepsy, essential tremor, and psychiatric disorders.
  • $33
In Stock
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