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Search Results for " muscarinic "

296

Compounds

25

Natural Products

9

Recombinant Proteins

1

Libraries

Cat No. Product Name Synonyms Targets
T80183 Muscarinic toxin 7
Muscarinic toxin 7 (MT7) is a peptide exhibiting selective, noncompetitive antagonistic activity at the muscarinic M1 receptor [1].
T80477 Muscarinic toxin 3 MT3 Adrenergic Receptor
Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57 for α1B, 8.13 for α1D, 8.49 for α2A, <6.5 for α2B, and 7.29 ...
T81893 M1/M4 muscarinic agonist 2
Compound 40 is a selective M1/M4 muscarinic antagonist with an IC50 of 19 nM for M1 receptors and 42 nM for M4 receptors [1].
T11078 Deschloroclozapine Serotonin Transporter
Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist. Deschloroclozapine binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively.
T4981 Anisotropine Methylbromide Prostaglandin Receptor , AChR
Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.
T1760 TBPB AChR
TBPB is an allosteric M1 mAChR agonist.
T11095L DREADD agonist 21 5-HT Receptor , Adrenergic Receptor , AChR , Histamine Receptor
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
T1281 Tropicamide Ro 1-7683 AChR
Tropicamide (Ro 1-7683) is a synthetic muscarinic antagonist with actions similar to atropine and with an anticholinergic property. Upon ocular administration, tropicamide binds to and blocks the muscarinic receptors in ...
T7555 Piperidolate hydrochloride AChR
Piperidolate hydrochloride is an antimuscarinic, could restrain the abnormal activity caused by acetylcholine. inhibits intestinal cramp induced by acetylcholine (rats and dogs).
T9419 Fesoterodine (R) Fesoterodine AChR
Fesoterodine ((R) Fesoterodine) is an orally active, competitive mAChR antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. It is used for the overactive bladder (OAB).
T9694 Emraclidine CVL-231 AChR
Emraclidine (CVL-231) is a muscarinic M4 receptor positive allosteric modulator and can be used in neurological diseases studies.
T23116 Oxotremorine sesquifumarate AChR
Oxotremorine sesquifumarate is a muscarinic agonist.
T2390 Cevimeline hydrochloride hemihydrate AChR
Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.
T28827 Sofpironium bromide BBI4000,BBI 4000,BBI-4000 Others , AChR
Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.
T6575 LY2119620 AChR
LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.
T4979 Procyclidine hydrochloride (±)-Procyclidine hydrochlorid NMDAR , iGluR
Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.
T1475 Fesoterodine fumarate Toviaz,SPM 907 AChR
Fesoterodine fumarate (Toviaz) is the fumarate salt form of fesoterodine, a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties. Fesoterodine is rapidly hydrolyzed in vivo...
T5655 MAChR-IN-1 hydrochloride AChR
mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.
T8219 VU0238441 AChR
VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.
T13066 TAK-071 AChR
TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).
T17244 VU0467154 AChR
VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor. The response to ACh with pEC50s of 7.75, 6.2, and 6 for a rat, human, and cynomolgus monkey M4 receptor, respectively.
T6548 Irsogladine Dicloguamine PDE , AChR
Irsogladine (Dicloguamine) is an anti-gastric ulcer agent that facilitates gap-junctional intercellular communication through M1 muscarininc acetylcholine receptor binding.
T7405 Piperidolate AChR
Piperidolate inhibits intestinal cramp induced by acetylcholine
T13325 VU 0365114 AChR
VU 0365114 is a positive allosteric modulator of mAChR M5 (EC50: 2.7 μM).
T9420 Prifinium bromide Others
Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.
T23524 W-84 dibromide HDMPPA AChR
W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.
T0794 Mepenzolate Bromide Colibantil,Cantil,Cantilaque AChR
Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.
T4997 Umeclidinium bromide GSK573719A AChR
Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.
T3993 BQCA benzylquinolone carboxylic acid AChR
BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.
T13385 Zamifenacin fumarate UK-76654 fumarate AChR
Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.
T8224 VU0119498 AChR
VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.
T4494 CLOZAPINE N-OXIDE Dopamine Receptor , 5-HT Receptor , AChR , Drug Metabolite
Clozapine N-oxide is the major metabolite of Clozapine and is blood-brain barrier permeable. Clozapine N-oxide is an agonist of DREADDs and activates the DREADD receptors hM3Dq and hM4Di. Clozapine N-oxide is also a dopa...
T0099 Tolterodine tartrate Detrol LA,PNU-200583E,Kabi-2234 AChR
Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.
T8383 Cyclopentolate Hydrochloride AChR
Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.
T1460 Dicyclomine hydrochloride AChR
Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.
T9353 OXOMEMAZINE AChR , Histamine Receptor
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low ...
T7002 Trihexyphenidyl hydrochloride Triesifenidile,Benzhexol hydrochloride,Tremin,Artane hydrochloride AChR
Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.
T9019 JHU37152 JHU 37152 AChR
JHU37152 (JHU 37152) is a Designer Receptors Exclusively Activated by Designer Drug (DREADD) agonist with Ki of 1.8 nM and 8.7 nM for human muscarinic acetylcholine M3 receptors (hM3Dq) and hM4Di in vitro, respectively. ...
T23508 VU 0255035 AChR
muscarinic M1 antagonist
T8007 VU 0238429 SCR-1481B1,VU0238429 AChR
VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).
T0427 Homatropine Methylbromide Homatropine methobromide AChR
Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.
T16411 Otenzepad AF-DX 116 AChR
Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.
T29123 VU0152099 VU 0152099,VU-0152099 AChR
VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).
T9018 JHU37160 JHU 37160 AChR
JHU37160 (JHU 37160) is a Designer Receptors Exclusively Activated by Designer Drug (DREADD) agonist with Ki of 1.9 nM and 3.6 nM for human muscarinic acetylcholine M3 receptors (hM3Dq) and hM4Di in vitro, respectively. ...
T1179 Tiotropium bromide Tiopropium,BA679 BR AChR
Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD). Tiotropium is a muscarinic receptor antagonist, on topical a...
T15942 MK-7622 M1 receptor modulator AChR
MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.
T3619 VU0357017 hydrochloride ML071 hydrochloride,CID-25010775,VU 0357017 hydrochloride AChR
VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.37 ± 0.15).
T22380 Nor-benzetimide Others , AChR
Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.
T28069 ML380 ML 380,ML-380 AChR
ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).
T0720 Gallamine triethiodide Benzkurin,Flaxedil AChR
Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.

Compounds

Muscarinic toxin 7
T80183
Synonym:
Target:
Muscarinic toxin 3
T80477
Synonym: MT3
Target: Adrenergic Receptor
M1/M4 muscarinic agonist 2
T81893
Synonym:
Target:
Deschloroclozapine
T11078
Synonym:
Target: Serotonin Transporter
Anisotropine Methylbromide
T4981
Synonym:
Target: Prostaglandin Receptor, AChR
TBPB
T1760
Synonym:
Target: AChR
DREADD agonist 21
T11095L
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor, AChR, Histamine Receptor
Tropicamide
T1281
Synonym: Ro 1-7683
Target: AChR
Piperidolate hydrochloride
T7555
Synonym:
Target: AChR
Fesoterodine
T9419
Synonym: (R) Fesoterodine
Target: AChR
Emraclidine
T9694
Synonym: CVL-231
Target: AChR
Oxotremorine sesquifumarate
T23116
Synonym:
Target: AChR
Cevimeline hydrochloride hemihydrate
T2390
Synonym:
Target: AChR
Sofpironium bromide
T28827
Synonym: BBI4000,BBI 4000,BBI-4000
Target: Others, AChR
LY2119620
T6575
Synonym:
Target: AChR
Procyclidine hydrochloride
T4979
Synonym: (±)-Procyclidine hydrochlorid
Target: NMDAR, iGluR
Fesoterodine fumarate
T1475
Synonym: Toviaz,SPM 907
Target: AChR
mAChR-IN-1 hydrochloride
T5655
Synonym:
Target: AChR
VU0238441
T8219
Synonym:
Target: AChR
TAK-071
T13066
Synonym:
Target: AChR
VU0467154
T17244
Synonym:
Target: AChR
Irsogladine
T6548
Synonym: Dicloguamine
Target: PDE, AChR
Piperidolate
T7405
Synonym:
Target: AChR
VU 0365114
T13325
Synonym:
Target: AChR
prifinium bromide
T9420
Synonym:
Target: Others
W-84 dibromide
T23524
Synonym: HDMPPA
Target: AChR
Mepenzolate Bromide
T0794
Synonym: Colibantil,Cantil,Cantilaque
Target: AChR
Umeclidinium bromide
T4997
Synonym: GSK573719A
Target: AChR
BQCA
T3993
Synonym: benzylquinolone carboxylic acid
Target: AChR
Zamifenacin fumarate
T13385
Synonym: UK-76654 fumarate
Target: AChR
VU0119498
T8224
Synonym:
Target: AChR
CLOZAPINE N-OXIDE
T4494
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, AChR, Drug Metabolite
Tolterodine tartrate
T0099
Synonym: Detrol LA,PNU-200583E,Kabi-2234
Target: AChR
Cyclopentolate Hydrochloride
T8383
Synonym:
Target: AChR
Dicyclomine hydrochloride
T1460
Synonym:
Target: AChR
OXOMEMAZINE
T9353
Synonym:
Target: AChR, Histamine Receptor
Trihexyphenidyl hydrochloride
T7002
Synonym: Triesifenidile,Benzhexol hydrochloride,Tremin,Artane hydrochloride
Target: AChR
JHU37152
T9019
Synonym: JHU 37152
Target: AChR
VU 0255035
T23508
Synonym:
Target: AChR
VU 0238429
T8007
Synonym: SCR-1481B1,VU0238429
Target: AChR
Homatropine Methylbromide
T0427
Synonym: Homatropine methobromide
Target: AChR
Otenzepad
T16411
Synonym: AF-DX 116
Target: AChR
VU0152099
T29123
Synonym: VU 0152099,VU-0152099
Target: AChR
JHU37160
T9018
Synonym: JHU 37160
Target: AChR
Tiotropium bromide
T1179
Synonym: Tiopropium,BA679 BR
Target: AChR
MK-7622
T15942
Synonym: M1 receptor modulator
Target: AChR
VU0357017 hydrochloride
T3619
Synonym: ML071 hydrochloride,CID-25010775,VU 0357017 hydrochloride
Target: AChR
Nor-benzetimide
T22380
Synonym:
Target: Others, AChR
ML380
T28069
Synonym: ML 380,ML-380
Target: AChR
Gallamine triethiodide
T0720
Synonym: Benzkurin,Flaxedil
Target: AChR
1 2 3 4 5 6
Cat No. Product Name Synonyms Targets
T0962 L-Hyoscyamine Daturine,Hyoscyamine AChR
L-Hyoscyamine (Daturine) functions as a non-selective, competitive antagonist of muscarinic receptors, thereby inhibiting the parasympathetic activities of acetylcholine on the salivary, bronchial, and sweat glands, as w...
T8304 Anisodamine Hydrobromide 6-Hydroxyhyoscyamine Adrenergic Receptor , AChR
Anisodamine Hydrobromide (6-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T8196 Arborine Arborin Others , AChR
Arborine (Arborin) is a larval growth inhibitor from glycoslnis pentaphylla.
T2198 Arecoline hydrobromide Arecoline HBr,Arecoline bromide AChR
Arecoline hydrobromide (Arecoline HBr) is a muscarinic acetylcholine receptor agonist.
T5S0106 Peimisine Ebeiensine RAAS , AChR
1. Peimisine (Ebeiensine) can affect M-receptor, excit β-receptor, restrain the release of internal calcium, and promote to releaseing nitrogen monoxidum in order to relax tracheal smooth muscle and relieve asthma. 2. Pe...
T1285 Anethole trithione Anetholtrithion Others , AChR
Anethole trithione (Anetholtrithion) is a bile secretion-stimulating drug that restores salivation and relieves the discomfort of dry mouth in chemotherapy-induced xerostomia.
T4S1619 L-Hyoscyamine sulfate Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate AChR
L-Hyoscyamine sulfate (Levsin Sulfate) is the sulfate salt of a belladonna alkaloid derivative and the levorotatory form of racemic atropine isolated from the plants Hyoscyamus niger or Atropa belladonna, which exhibits ...
T1231 Pilocarpine nitrate Pilagan,Pilofrin AChR
Pilocarpine nitrate (Pilagan) is a slowly hydrolyzed muscarinic agonist with no nicotinic effects. Pilocarpine is used as a miotic and in the treatment of glaucoma.
T0970 Racanisodamine Anisodamine,7β-Hydroxyhyoscyamine,Raceanisodamine Adrenergic Receptor , AChR
Racanisodamine (7β-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T5805 Guvacoline hydrochloride Norarecoline hydrochloride AChR
Guvacoline hydrochloride (Norarecoline hydrochloride) is a muscarinic agonist.
T0804 Pilocarpine Hydrochloride NSC 5746 HCl,Pilocarpine HCl,(+)-Pilocarpine hydrochloride AChR
Pilocarpine Hydrochloride (NSC 5746 HCl) , a nonselective muscarinic acetylcholine receptor agonist, is utilized to produce an experimental model of epilepsy.
TN1653 Fustin ERK , Beta Amyloid , AChR
Fustin is the phytogenic flavanol component of the plant Rhus verniciflua Stokes. Fustin shows protective effects on 6-hydroxydopamine-induced neuronal cell death.
T6805 Choline bitartrate 2,3,4-trihydroxy-4-oxobutanoate,2-hydroxyethyl(trimethyl)azanium Others , AChR
Choline bitartrate (2-hydroxyethyl(trimethyl)azanium) is a form of the nutrient choline which is found in foods. Choline is necessary for normal liver and kidney function and a component of the neurotransmitter acetylcho...
T7056 Dronedarone SR 33589 P450 , Potassium Channel , Calcium Channel , Sodium Channel , Adrenergic Receptor , AChR , Autophagy
Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
T1341 Nortropine Nortropenol AChR
Nortropine (Nortropenol) is used as muscarinic receptor antagonists.
T21532 Anisodamine 6-Hydroxyhyoscyamine,6-beta-Hydroxyhyoscyamine AChR
Anisodamine (6-beta-Hydroxyhyoscyamine) is an antagonist of muscarinic and nicotinic cholinoceptor with similar affinities at the muscarinic receptor as scopolamine and atropine. Anisodamine improve the microcirculation ...
T4727 Taurolithocholic acid sodium salt Sodium taurolithocholate Others , Calcium Channel
Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but not to M2 or M3 receptors.
T4S0111 Hupehenine AChR
Hupehenine is a steriodal alkaloid extracted from the bulbs of Fritillaria Hupehensis, with the potential for inhibiting acetylcholine, antagonism for muscarinic receptors and cholinesterase inhibition.
T68953 Arecoline Reactive Oxygen Species , AChR
Arecoline is a natural alkaloid derived from areca nut in the palm family and is a potent nicotine and partial agonist of muscarinic acetylcholine receptors. Arecoline has anti-anxiety and anti-parasitic activity, can in...
T0266 Quinidine hydrochloride monohydrate Quinidine hydrochloride Potassium Channel , Sodium Channel , Parasite
Quinidine hydrochloride monohydrate is an optical isomer of quinine, extracted from the bark of the Cinchona tree and similar plant species. It prolongs cellular action potential and decreases automaticity. This alkaloid...
T6S0659 Rhynchophylline Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin Calcium Channel , NF-κB
1. Rhynchophylline (Mitrinermine) can protect against ischemic damage, probably via regulating the Akt/mTOR pathway. 2. Rhynchophylline can protect against glutamate-induced neuronal death, can inhibit MA impairment in c...
TN2116 Pteropodine BCL , Calcium Channel , 5-HT Receptor
Pteropodine acts as a positive modulator of muscarinic M(1) and 5-HT(2) receptors. Pteropodine shows antigenotoxic, antioxidant and lymphocyte induction effects, it also shows strong apoptotic effect on acute leukaemic l...
TN4342 Izalpinine Others
Izalpinin exhibits potent antioxidant activities in the 1,1-diphenyl-2-picrylhydrazyl (DPPH) assay. Izalpinin exhibits inhibitory role of muscarinic receptor-related detrusor contractile activity, and it may be a promisi...
TN1790 Isopteropodine Uncarine E 5-HT Receptor , Antibacterial , AChR
Isopteropodine (Uncarine E) is an isoyohimbine-type octindole alkaloid isolated from Hamelia patens micropropagated and has antimicrobial activity and stimulates the immune system. Isopteropodine has antimicrobial activi...
T73856 Anagyrine hydrochloride
Anagyrine hydrochloride ((-)-Anagyrine hydrochloride), a quinolizidine alkaloid discovered in Lupinus albus, interacts with both muscarinic and nicotinic acetylcholine receptors, demonstrating IC50 values of 132 and 2096...

Natural Products

L-Hyoscyamine
T0962
Synonym: Daturine,Hyoscyamine
Target: AChR
Anisodamine Hydrobromide
T8304
Synonym: 6-Hydroxyhyoscyamine
Target: Adrenergic Receptor, AChR
Arborine
T8196
Synonym: Arborin
Target: Others, AChR
Arecoline hydrobromide
T2198
Synonym: Arecoline HBr,Arecoline bromide
Target: AChR
Peimisine
T5S0106
Synonym: Ebeiensine
Target: RAAS, AChR
Anethole trithione
T1285
Synonym: Anetholtrithion
Target: Others, AChR
L-Hyoscyamine sulfate
T4S1619
Synonym: Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate
Target: AChR
Pilocarpine nitrate
T1231
Synonym: Pilagan,Pilofrin
Target: AChR
Racanisodamine
T0970
Synonym: Anisodamine,7β-Hydroxyhyoscyamine,Raceanisodamine
Target: Adrenergic Receptor, AChR
Guvacoline hydrochloride
T5805
Synonym: Norarecoline hydrochloride
Target: AChR
Pilocarpine Hydrochloride
T0804
Synonym: NSC 5746 HCl,Pilocarpine HCl,(+)-Pilocarpine hydrochloride
Target: AChR
Fustin
TN1653
Synonym:
Target: ERK, Beta Amyloid, AChR
Choline bitartrate
T6805
Synonym: 2,3,4-trihydroxy-4-oxobutanoate,2-hydroxyethyl(trimethyl)azanium
Target: Others, AChR
Dronedarone
T7056
Synonym: SR 33589
Target: P450, Potassium Channel, Calcium Channel, Sodium Channel, Adrenergic Receptor, AChR, Autophagy
Nortropine
T1341
Synonym: Nortropenol
Target: AChR
Anisodamine
T21532
Synonym: 6-Hydroxyhyoscyamine,6-beta-Hydroxyhyoscyamine
Target: AChR
Taurolithocholic acid sodium salt
T4727
Synonym: Sodium taurolithocholate
Target: Others, Calcium Channel
Hupehenine
T4S0111
Synonym:
Target: AChR
Arecoline
T68953
Synonym:
Target: Reactive Oxygen Species, AChR
Quinidine hydrochloride monohydrate
T0266
Synonym: Quinidine hydrochloride
Target: Potassium Channel, Sodium Channel, Parasite
Rhynchophylline
T6S0659
Synonym: Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin
Target: Calcium Channel, NF-κB
Pteropodine
TN2116
Synonym:
Target: BCL, Calcium Channel, 5-HT Receptor
Izalpinine
TN4342
Synonym:
Target: Others
Isopteropodine
TN1790
Synonym: Uncarine E
Target: 5-HT Receptor, Antibacterial, AChR
Anagyrine hydrochloride
T73856
Synonym:
Target:

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-02286 Influenza A H1N1 (A/Puerto Rico/8/34/Mount Sinai) Matrix protein 1/M1 Protein (His) H1N1 E. coli
The Influenza virus matrix protein 1 (M1) is a matrix protein of the influenza virus. M1 protein has been shown to play a crucial role in virus replication, assembly, and budding. It forms a coat inside the viral envelop...
TMPY-00496 Influenza A H1N1 (A/Brevig Mission/1/1918) Matrix protein 1/M1 Protein (His) H1N1 E. coli
The Influenza virus matrix protein 1 (M1) is a matrix protein of the influenza virus. M1 protein has been shown to play a crucial role in virus replication, assembly, and budding. It forms a coat inside the viral envelop...
TMPY-03844 Influenza A H7N9 (A/Anhui/1/2013) Matrix protein 1/M1 Protein (His) H7N9 E. coli
The Influenza virus matrix protein 1 (M1) is a matrix protein of the influenza virus. M1 protein has been shown to play a crucial role in virus replication, assembly, and budding. It forms a coat inside the viral envelop...
TMPY-00498 Influenza A H3N2 (A/Aichi/2/1968) Matrix protein 1/M1 Protein (His) H3N2 E. coli
The Influenza virus matrix protein 1 (M1) is a matrix protein of the influenza virus. M1 protein has been shown to play a crucial role in virus replication, assembly, and budding. It forms a coat inside the viral envelop...
TMPH-01714 CHRM1 Protein, Human, Recombinant (His) Human E. coli
The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. ...
TMPH-03338 CHRM1 Protein, Rat, Recombinant (His) Rat E. coli
CHRM1 Protein, Rat, Recombinant (His) is expressed in E. coli.
TMPH-01715 CHRM2 Protein, Human, Recombinant (His) Human E. coli
The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. ...
TMPH-01716 CHRM3 Protein, Human, Recombinant (B2M & His) Human E. coli
The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. ...
TMPH-01717 CHRM5 Protein, Human, Recombinant (His) Human E. coli
The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. ...
Cat No. Product Name
L9830 Anti-Parkinson's Disease Compound Library

908 compounds
A unique collection of 908 compounds with anti-PD activities or acting on main drug targets of PD can be used for HTS and HCS.
TargetMol