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GLP-1R/GIPR agonist-1 soduim

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Catalog No. TP3645

GLP-1R/GIPR agonist-1 sodium is the sodium salt form of GLP-1R/GIPR agonist-1. It acts as a dual agonist for the glucagon-like peptide-1 receptor (GLP-1R, EC50 = 0.57 nM) and the glucose-dependent insulinotropic polypeptide receptor (GIPR, EC50 = 0.75 nM). GLP-1R/GIPR agonist-1 sodium lowers blood glucose by mimicking the effects of endogenous hormones GLP-1 and GIP, enhancing insulin secretion, and inhibiting glucagon secretion. This compound is applicable in research on metabolic disorders such as diabetes, obesity, and non-alcoholic steatohepatitis (NASH).

GLP-1R/GIPR agonist-1 soduim
Other Forms of GLP-1R/GIPR agonist-1 soduim:
GLP-1R/GIPR agonist-1TP3568
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GLP-1R/GIPR agonist-1 soduim

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Catalog No. TP3645
GLP-1R/GIPR agonist-1 sodium is the sodium salt form of GLP-1R/GIPR agonist-1. It acts as a dual agonist for the glucagon-like peptide-1 receptor (GLP-1R, EC50 = 0.57 nM) and the glucose-dependent insulinotropic polypeptide receptor (GIPR, EC50 = 0.75 nM). GLP-1R/GIPR agonist-1 sodium lowers blood glucose by mimicking the effects of endogenous hormones GLP-1 and GIP, enhancing insulin secretion, and inhibiting glucagon secretion. This compound is applicable in research on metabolic disorders such as diabetes, obesity, and non-alcoholic steatohepatitis (NASH).
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Product Introduction

Bioactivity
Description
GLP-1R/GIPR agonist-1 sodium is the sodium salt form of GLP-1R/GIPR agonist-1. It acts as a dual agonist for the glucagon-like peptide-1 receptor (GLP-1R, EC50 = 0.57 nM) and the glucose-dependent insulinotropic polypeptide receptor (GIPR, EC50 = 0.75 nM). GLP-1R/GIPR agonist-1 sodium lowers blood glucose by mimicking the effects of endogenous hormones GLP-1 and GIP, enhancing insulin secretion, and inhibiting glucagon secretion. This compound is applicable in research on metabolic disorders such as diabetes, obesity, and non-alcoholic steatohepatitis (NASH).
Chemical Properties
FormulaC220H334N55O69.xNa
SequenceHis-{Aib}-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-{Aib}-Leu-Asp-Lys-Arg-Ala-Ala-Lys(AEEA-AEEA-gammaGlu-C18 diacid)-Asp-Phe-Val-Glu-Trp-Leu-Lys-Asn-Gly-Gly-Pro-Ser-Ser-Gly-Ala-Pro-Pro-Pro-Ser-NH2
Sequence Short{Aib}-QGTFTSDYSK-{Aib}-LDKRAA-K(AEEA-AEEA-gammaGlu-C18 diacid)-DFVEWLKNGGPSSGAPPPS
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
TargetMol | Animal experiments For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent 10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.
Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSOTargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSOTargetMol | reagent stock solution to 400 μL PEG300TargetMol | reagent and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH2OTargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.
1 Enter information below:
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2 Enter the in vivo formulation:
% DMSO
%
% Tween 80
% Saline/PBS/ddH2O

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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