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Search Results for "llc"

Compounds

Cat No. Product Name
T32810 LL-C 10037alpha LL-c10037alpha,LLC 10037alpha
LL-C 10037alpha is a gamma-aminoepoxysemiquinone isolated from Streptomyces.
TN1040 Skullcapflavone II COX , Antibacterial , TGF-beta/Smad
Skullcapflavone II 是从黄芩中提取的黄酮,具有抗炎作用。它对 M. aurum 和 M. bovisBCG 具有较强的抗菌活性。它还调节破骨细胞的分化、存活和功能。
TN5033 Skullcapflavone I IL Receptor , Caspase , Prostaglandin Receptor
Skullcapflavone I has anti-inflammatory and anti-allergic potential, it can significantly inhibit LPS stimulated NO and ...
T3S1967 (S)-Indoximod 相思子碱;相思豆碱,红豆,Abrine,N-ME-Tryptophan,L-Abrine Others , Indoleamine 2,3-Dioxygenase (IDO)
Abrine 是一种吲哚胺-2,3-双加氧酶 (IDO) 抑制剂,可用于研究癌症。
T12580 PTUPB Epoxide Hydrolase , COX
PTUPB 是强效的sEH(IC50:0.9 μM)和COX-2(IC50:1.26 μM)的双向抑制剂。
T0463 Loxoprofen Koloxo,Loxoprofene,Loxoprofeno,洛索洛芬 COX
Loxoprofen 是一种非甾体类抗炎药,具有解热作用,可用于缓解疼痛的研究。它是非选择性COX 抑制剂,对 COX-1 和 COX-2 的IC50分别为 6.5 和 13.5 μM。
T11719 JMV 2959 hydrochloride (925238-89-7 free base) JMV 2959 hydrochloride GHSR
JMV 2959 hydrochloride (925238-89-7 free base) 是一种生长激素促分泌素受体 1a 型 (GHS-R1a) 拮抗剂,在 LLC-PK1 细胞中的 IC50 为 32±3 nM。
T9616 PD-1/PD-L1-IN-10 PD-1/PD-L1
PD-1/PD-L1-IN-10 是一种口服有效的PD-1/PD-L1抑制剂 (IC50of 2.7 nM),显示出抗肿瘤活性。
T5S0106 Peimisine 贝母辛,Ebeiensine AChR , RAAS
Peimisine 非竞争性拮抗气管平滑肌 M 受体,抑制 Ach 引起的平滑肌收缩。它兴奋 β 受体和拮抗内钙释放,促进一氧化氮释放,可舒张气管平滑肌,有平喘作用。
T6835 Fenoldopam mesylate mesylate,Corlopam mesylate,Fenoldopam methanesulfonate,SKF 82526,SKF-82526 mesylate,非诺多泮甲磺酸盐 Dopamine Receptor
Fenoldopam mesylate 是一种多巴胺受体D1选择性激动剂。
TN4455 Lucialdehyde B Integrase , HSV
Lucialdehyde B exhibits potent inhibitory activity against herpes simplex virus. It shows cytotoxic effects on Lewis lun...
TN4457 Lucidal Others
Lucialdehyde C (Lucidal) exhibits potent cytotoxicity against LLC, T-47D, Sarcoma 180, and Meth-A tumor cells with ED(50...
T38281 C22 Galactosylceramide (d18:1/22:0)
C22 Galactosylceramide is a sphingolipid that has been found in the central nervous system.1,2C22 Galactosylceramide lev...
T39195 YM-244769 dihydrochloride Calcium Channel
YM-244769 dihydrochloride 是一种有效的 Na+/Ca2+ exchange 3 (NCX3) 抑制剂,IC50 为 18 nM。 YM-244769 dihydrochloride 对神经元和肾脏具有有效的保护作用...
T35483 19,20-Epoxycytochalasin D
19,20-Epoxycytochalasin D is a fungal metabolite that has been found in the endophytic fungus Nemania sp. UM10M. It is a...
T38286 C26 Sphingomyelin (d18:1/26:0) C26 Sphingomyelin (d18:1/26:0)
C26 Sphingomyelin is a sphingolipid that has been found in serum and cell or brain extracts.1,2,3C26 sphingomyelin level...
T9888 YM-244769 3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]- Calcium Channel
YM-244769 是一种有效的 Na+/Ca2+ exchange 3 (NCX3) 抑制剂,IC50 为 18 nM。 YM-244769 对神经元和肾脏具有有效的保护作用。
TN4108 Ganoderic acid Z Antifection
The binding affinities of ganoderic acid DM and ganoderic acid Z (ΔGbind, -16.83 and-10.99 kcal mol-1) are comparable t...
T37455 C18 D-threo Ceramide (d18:1/18:0) C18 D-threo Ceramide (d18:1/18:0)
C18 D-threoCeramide (d18:1/18:0) is a synthetic ceramide and stereoisomer of C18 ceramide .1It inhibits rat brain mitoch...
T36695 TAS-103
TAS-103 is a dual inhibitor of DNA topoisomerase I/II, used for cancer research. TAS-103 is a dual inhibitor of DNA topo...
LL-C 10037alpha
T32810
synonym: LL-c10037alpha,LLC 10037alpha
Target:
Skullcapflavone II
TN1040
synonym:
Target:
Skullcapflavone I
TN5033
synonym:
Target:
(S)-Indoximod
T3S1967
synonym: 相思子碱;相思豆碱,红豆,Abrine,N-ME-Tryptophan,L-Abrine
Target:
PTUPB
T12580
synonym:
Target:
Loxoprofen
T0463
synonym: Koloxo,Loxoprofene,Loxoprofeno,洛索洛芬
Target:
JMV 2959 hydrochloride (925238-89-7 free base)
T11719
synonym: JMV 2959 hydrochloride
Target:
PD-1/PD-L1-IN-10
T9616
synonym:
Target:
Peimisine
T5S0106
synonym: 贝母辛,Ebeiensine
Target:
Fenoldopam mesylate
T6835
synonym: mesylate,Corlopam mesylate,Fenoldopam methanesulfonate,SKF 82526,SKF-82526 mesylate,非诺多泮甲磺酸盐
Target:
Lucialdehyde B
TN4455
synonym:
Target:
Lucidal
TN4457
synonym:
Target:
C22 Galactosylceramide (d18:1/22:0)
T38281
synonym:
Target:
YM-244769 dihydrochloride
T39195
synonym:
Target:
19,20-Epoxycytochalasin D
T35483
synonym:
Target:
C26 Sphingomyelin (d18:1/26:0)
T38286
synonym: C26 Sphingomyelin (d18:1/26:0)
Target:
YM-244769
T9888
synonym: 3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]-
Target:
Ganoderic acid Z
TN4108
synonym:
Target:
C18 D-threo Ceramide (d18:1/18:0)
T37455
synonym: C18 D-threo Ceramide (d18:1/18:0)
Target:
TAS-103
T36695
synonym:
Target:
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