T32810 |
LL-C 10037alpha
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LL-c10037alpha,LLC 10037alpha |
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LL-C 10037alpha is a gamma-aminoepoxysemiquinone isolated from Streptomyces. |
TN1040 |
Skullcapflavone II
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COX
,
Antibacterial
,
TGF-beta/Smad
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Skullcapflavone II 是从黄芩中提取的黄酮,具有抗炎作用。它对 M. aurum 和 M. bovisBCG 具有较强的抗菌活性。它还调节破骨细胞的分化、存活和功能。 |
TN5033 |
Skullcapflavone I
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IL Receptor
,
Caspase
,
Prostaglandin Receptor
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Skullcapflavone I has anti-inflammatory and anti-allergic potential, it can significantly inhibit LPS stimulated NO and ... |
T3S1967 |
(S)-Indoximod
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相思子碱;相思豆碱,红豆,Abrine,N-ME-Tryptophan,L-Abrine |
Others
,
Indoleamine 2,3-Dioxygenase (IDO)
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|
Abrine 是一种吲哚胺-2,3-双加氧酶 (IDO) 抑制剂,可用于研究癌症。 |
T12580 |
PTUPB
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Epoxide Hydrolase
,
COX
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PTUPB 是强效的sEH(IC50:0.9 μM)和COX-2(IC50:1.26 μM)的双向抑制剂。 |
T0463 |
Loxoprofen
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Koloxo,Loxoprofene,Loxoprofeno,洛索洛芬 |
COX
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|
Loxoprofen 是一种非甾体类抗炎药,具有解热作用,可用于缓解疼痛的研究。它是非选择性COX 抑制剂,对 COX-1 和 COX-2 的IC50分别为 6.5 和 13.5 μM。 |
T11719 |
JMV 2959 hydrochloride (925238-89-7 free base)
|
JMV 2959 hydrochloride |
GHSR
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|
JMV 2959 hydrochloride (925238-89-7 free base) 是一种生长激素促分泌素受体 1a 型 (GHS-R1a) 拮抗剂,在 LLC-PK1 细胞中的 IC50 为 32±3 nM。 |
T9616 |
PD-1/PD-L1-IN-10
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PD-1/PD-L1
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PD-1/PD-L1-IN-10 是一种口服有效的PD-1/PD-L1抑制剂 (IC50of 2.7 nM),显示出抗肿瘤活性。 |
T5S0106 |
Peimisine
|
贝母辛,Ebeiensine |
AChR
,
RAAS
|
|
Peimisine 非竞争性拮抗气管平滑肌 M 受体,抑制 Ach 引起的平滑肌收缩。它兴奋 β 受体和拮抗内钙释放,促进一氧化氮释放,可舒张气管平滑肌,有平喘作用。 |
T6835 |
Fenoldopam mesylate
|
mesylate,Corlopam mesylate,Fenoldopam methanesulfonate,SKF 82526,SKF-82526 mesylate,非诺多泮甲磺酸盐 |
Dopamine Receptor
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Fenoldopam mesylate 是一种多巴胺受体D1选择性激动剂。 |
TN4455 |
Lucialdehyde B
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Integrase
,
HSV
|
|
Lucialdehyde B exhibits potent inhibitory activity against herpes simplex virus. It shows cytotoxic effects on Lewis lun... |
TN4457 |
Lucidal
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|
Others
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Lucialdehyde C (Lucidal) exhibits potent cytotoxicity against LLC, T-47D, Sarcoma 180, and Meth-A tumor cells with ED(50... |
T38281 |
C22 Galactosylceramide (d18:1/22:0)
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|
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C22 Galactosylceramide is a sphingolipid that has been found in the central nervous system.1,2C22 Galactosylceramide lev... |
T39195 |
YM-244769 dihydrochloride
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Calcium Channel
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|
YM-244769 dihydrochloride 是一种有效的 Na+/Ca2+ exchange 3 (NCX3) 抑制剂,IC50 为 18 nM。 YM-244769 dihydrochloride 对神经元和肾脏具有有效的保护作用... |
T35483 |
19,20-Epoxycytochalasin D
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|
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19,20-Epoxycytochalasin D is a fungal metabolite that has been found in the endophytic fungus Nemania sp. UM10M. It is a... |
T38286 |
C26 Sphingomyelin (d18:1/26:0)
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C26 Sphingomyelin (d18:1/26:0) |
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C26 Sphingomyelin is a sphingolipid that has been found in serum and cell or brain extracts.1,2,3C26 sphingomyelin level... |
T9888 |
YM-244769
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3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]- |
Calcium Channel
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YM-244769 是一种有效的 Na+/Ca2+ exchange 3 (NCX3) 抑制剂,IC50 为 18 nM。 YM-244769 对神经元和肾脏具有有效的保护作用。 |
TN4108 |
Ganoderic acid Z
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Antifection
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The binding affinities of ganoderic acid DM and ganoderic acid Z (ÎGbind, -16.83 and-10.99 kcal mol-1) are comparable t... |
T37455 |
C18 D-threo Ceramide (d18:1/18:0)
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C18 D-threo Ceramide (d18:1/18:0) |
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C18 D-threoCeramide (d18:1/18:0) is a synthetic ceramide and stereoisomer of C18 ceramide .1It inhibits rat brain mitoch... |
T36695 |
TAS-103
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|
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TAS-103 is a dual inhibitor of DNA topoisomerase I/II, used for cancer research.
TAS-103 is a dual inhibitor of DNA topo... |