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Picrasidine Q

Name: Picrasidine Q
Brand: TargetMol
SKU: TN6651
Rating: 4.5 (1 reviews)

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Catalog No. TN6651Cas No. 101219-61-8

Picrasidine Q is an anticancer natural alkaloid that targets FGFR2, inducing apoptosis and G1 arrest in oesophageal squamous cell carcinoma (ESCC) cells.

Picrasidine Q

😃Good

Catalog No. TN6651Cas No. 101219-61-8

Picrasidine Q is an anticancer natural alkaloid that targets FGFR2, inducing apoptosis and G1 arrest in oesophageal squamous cell carcinoma (ESCC) cells.

Pack Size	Price	Availability	Quantity
10 mg	$422	Backorder

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Product Introduction

Bioactivity

Description	Picrasidine Q is an anticancer natural alkaloid that targets FGFR2, inducing apoptosis and G1 arrest in oesophageal squamous cell carcinoma (ESCC) cells.
Targets&IC50	A549 cells:16.2 μg/mL (ED50), MCF7:18.1 μg/mL (ED50)
In vitro	Methods: Picrasidine Q (0-60 μM) was used to treat the human esophageal cancer cell lines (including KYSE30, KYSE410, and KYSE450). Cell proliferation was measured by MTT assay; flow cytometry was employed to analyze cell cycle distribution and apoptosis; and changes in related protein expression levels were examined through Western blotting. Results: Picrasidine Q effectively inhibited the proliferation of ESCC cells and significantly induced their apoptosis.[1]

Chemical Properties

Molecular Weight	266.25
Formula	C₁₅H₁₀N₂O₃
Cas No.	101219-61-8
Smiles	O=C1C(OC)=C(O)C2=NC=CC=3C4=CC=CC=C4N1C23
Relative Density.	1.51 g/cm3 (Predicted)
Color	Yellow
Appearance	Solid

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