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RAAS

The renin–angiotensin system (RAS), or renin–angiotensin–aldosterone system (RAAS), is a hormone system that regulates blood pressure and fluid and electrolyte balance, as well as systemic vascular resistance.

  • Angiotensin II human
    T70404474-91-3
    Angiotensin II human (Ang II) is a biologically active peptide, a vasoconstrictor. Angiotensin II interacts with AT1R and AT2R to regulate blood pressure, stimulate sympathetic nerves, and increase aldosterone biosynthesis and renal activity in humans.
    • $37
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  • Irbesartan
    T1615138402-11-6
    Irbesartan (SR-47436) is an Angiotensin 2 Receptor Blocker. The mechanism of action of irbesartan is as an Angiotensin 2 Receptor Antagonist.
    • $48
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  • Tranilast
    T269053902-12-8
    Tranilast (SB 252218), an antiallergic drug, suppresses lipid mediator and cytokine release from inflammatory cells, therefore utilized in the treatment of allergic disorders.
    • $36
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  • Sacubitril/Valsartan
    T2318936623-90-4
    Sacubitril/Valsartan (LCZ696) is an orally bioavailable, dual angiotensin II receptor and neprilysin inhibitor for the treatment of hypertension and heart failure.
    • $38
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  • Captopril
    T146262571-86-2
    Captopril (SA333) is a potent and specific inhibitor of peptidyl-dipeptidase A. It blocks the conversion of angiotensin I to angiotensin II, a vasoconstrictor and important regulator of arterial blood pressure.
    • $40
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  • [Sar1, Ile8]-Angiotensin II acetate
    T7575L1
    [Sar1, Ile8]-Angiotensin II acetate activates both the NADPH and NADH oxidases, and stimulates superoxide anion formation in vascular smooth muscle cells. [Sar1, Ile8]-Angiotensin II acetate has multiple effects on vascular smooth muscle, including contra
    • $37
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  • ANGIOTENSIN IV TFA(12676-15-2(free base))
    T7743
    ANGIOTENSIN IV TFA is a less effective agonist at the angiotensin AT1 receptor.
    • $43
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  • L-162,313
    T27762151488-11-8In house
    L-162,313 is an ANG II receptor agonist, a nonpeptide that mimics the biological actions of angiotensin II and induces an increase in MAP.
    • $350
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  • TRV-120027 acetate (1234510-46-3 free base)
    TP2158L11824712-70-0
    TRV-120027 acetate is a β-arrestin-1-biased agonist of the angiotensin II receptor type 1 (AT1 receptor) and engages -arrestins while blocking G-protein signaling.
    • $100
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  • Novokinin acetate
    T23077L
    Novokinin acetate exhibited an affinity for the AT2 receptor with Ki of 7 nM, and its antihypertensive and vasorelaxing activities were blocked by PD123319, an AT2 receptor antagonist.
    • $237
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  • Angiotensin I/II (1-5)
    TP152858442-64-1
    Angiotensin I/II (1-5) is a peptide (ASP-ARG-VAL-TYR-ILE) that contains the amino acids 1-5 and is converted from Angiotensin I/II.
    • $50
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  • FPL-62129
    T2735795445-79-7In house
    FPL-62129 is a calcium channel antagonist and a novel angiotensin-converting enzyme inhibitor with vasodilator activity for the study of cardiovascular disease.
    • $293
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  • Acein acetate
    TP1920L1
    Acein acetate is a high-affinity angiotensin-converting enzyme (ACE) ligand (Kd = 2.79 nM). Concentrations up to 500 nM had no significant effect on ACE enzyme activity. Enhanced NMDA + D-serine-induced dopamine release from striatal slices in vitro and striatum in vivo.
    • $133
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  • Ripisartan
    T28540148504-51-2In house
    Ripisartan (UP-269-6) is a potent and specific angiotensin II receptor antagonist that inhibits angiotensin II-mediated sympathetic tachycardia responses.
    • $191
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  • Pomisartan
    T28437144702-17-0In house
    Pomisartan (BIBR-363) is a small molecule angiotensin type 1 receptor (AT1R) antagonist that is used in the treatment of cardiovascular disease, studying heart failure and hypertensio
    • $143
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  • Terlakiren
    T28950119625-78-4In house
    Terlakiren (CP-80,794) is an orally active and potent renin inhibitor that inhibits the potency of human renin for the study of neurological disorders of the hypertension class.
    • $628
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  • Ceronapril
    T25226111223-26-8In house
    Ceronapril (SQ 29852) is an orally active and potent angiotensin-converting enzyme (ACE) inhibitor (IC50 : 36 nM) for the study of dementia and hypertension.
    • $628
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  • Alamandine TFA
    T37496L
    Alamandine TFA , a member of the renin-angiotensin system (RAS), a vasoactive peptide, is an endogenous ligand of the G protein-coupled receptor MrgD. Alamandine TFA targets to protect the kidney and heart through anti-hypertensive actions[1][2].
    • $55
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  • Enalapril
    T160575847-73-3
    Enalapril is a dicarbocyl-containing peptide and angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.
    • $30
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  • Azilsartan Methyl Ester
    T66580147403-52-9
    Azilsartan Methyl Ester is an angiotensin II receptor antagonist. Azilsartan Methyl Ester inhibits specific binding of [125I]AII (0.2 nM) to bovine adrenal cortex with IC50 value is 0.44uM.
    • $62
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  • A 779 TFA(159432-28-7 free base)
    T7616L
    A 779 TFA is a potent antagonist of angiotensin-(1-7) receptor.
    • $50
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  • N-Acetyl-Ser-Asp-Lys-Pro
    TP1828127103-11-1
    Acetyl Ser-Asp-Lys-Pro is formed in bone marrow cells by enzymatic processing of thymosin β4. It inhibits the entry of pluripotent hemopoietic stem cells into S-phase of the cell cycle and protects against Ara-C lethality in mice.
    • $50
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  • Pomisartan 2HCl
    T28437L In house
    Pomisartan 2HCl (BIBR363 2HCL) is a small molecule AT1R antagonist used to study heart failure and hypertension.
    • $195
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  • ME-3221
    T28009139958-16-0
    ME-3221 is an angiotensin AT1 receptor antagonist that prevents hypertensive complications in aged stroke-prone hypertensive rats.
    • $293
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  • Angiotensin II 5-valine TFA
    TP1017L
    Angiotensin II 5-valine TFA is an agonist of angiotensin receptor.
    • $53
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  • Leucylarginylproline
    T7510133943-59-6
    Leucylarginylproline is an inhibitor of angiotensin-converting enzyme (ACE) (IC50 : 0.27μM).
    • $89
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  • Methyl candesartan
    T65739139481-69-9
    Methyl candesartan (Candesartan Methyl Ester) is a potent angiotensin 2 receptor antagonist used in the study of hypertension.
    • $43
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  • TRV055 acetate
    T40220L
    TRV055 acetate is a ligand of angiotensin II type 1 receptor and stimulates cellular Gq-mediated signaling.
    • $195
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  • Valsartan Methyl Ester
    T67848137863-17-3
    Valsartan Methyl Ester is a potent angiotensin II receptor antagonist, IC50= 0.06uM.
    • $80
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  • CGP-42112 acetate
    T14939L
    CGP-42112 acetate is a potent angiotensin receptor AT2 agonist that inhibits the increase in protein kinase A activity produced by LPS.
    • $127
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  • (Sar¹)-Angiotensin II acetate
    T35834L
    (Sar¹)-Angiotensin II acetate, an analogue of Angiotensin II, is a specific agonist of angiotensin AT1 receptor. It binds to brain membrane-rich particles, with a Kd of 2.7 nM. It can stimulate protein synthesis and cell growth in embryonic chick myocytes.
    • $148
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  • Angiotensin 1/2 (5-7) acetate
    T22574L
    Angiotensin 1/2 (5-7) acetate is a peptide with the sequence H2N-Ile-His-Pro-OH. Angiotensin is an oligopeptide and is a hormone and a powerful dipsogen. It is derived from the precursor molecule angiotensinogen, a serum globulin produced in the liver. It
    • $37
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  • Angiotensin I/II (1-6)
    TP157947896-63-9
    Angiotensin I/II (1-6) is a peptide (ASP-ARG-VAL-TYR-ILE-HIS) that contains the amino acids 1-6 and is converted from Angiotensin I/II peptide.
    • $50
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  • Moveltipril
    T2583285856-54-8In house
    Moveltipril (Moveltipril calcium) is a potent angiotensin-converting enzyme (ACE) inhibitor.Moveltipril is converted to captopril in the body for action.
    • $83
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  • Allisartan Isoproxil
    T26594947331-05-7In house
    Allisartan Isoproxil is a nonpeptide antagonist of angiotensin II receptor and can be used in studies about hypertension and heart diseases.
    • $195
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  • Cilazapril Monohydrate
    T644492077-78-6In house
    Cilazapril Monohydrate (Justor) is an angiotensin-converting enzyme (ACE) inhibitor used for the treatment of hypertension and congestive heart failure.
    • $58
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  • Losartan
    T0215L114798-26-4
    Losartan (DuP-753) is an angiotensin II receptor antagonist.
    • $50
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  • PD 123319
    T6067130663-39-7
    PD 123319 ((S)-(+)-PD 123319) is a potent, selective AT2 angiotensin II receptor antagonist.
    • $45
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  • Valsartan
    T6716137862-53-4
    Valsartan (CGP 48933) is a tetrazole derivative and angiotensin II type 1 receptor blocker that is used to treat hypertension.
    • $46
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  • A 779
    T7616159432-28-7
    A 779 is a potent antagonist of the G-protein-coupled receptor Mas, the Ang1-7 receptor, which is distinct from conventional AngII.
    • $268
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  • Azilsartan Medoxomil
    T6219863031-21-4
    Azilsartan Medoxomil (TAK-491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.
    • $34
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  • DX600 TFA
    TP1622
    DX600 TFA is a specific inhibitor of ACE2 and does not cross-react with ACE.
    • $163
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  • Perindoprilat
    T148495153-31-4
    Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.
    • $37
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  • Camellianin A
    TN1464109232-77-1
    Camellianin A is a flavonoid series of compounds derived from A. nitida and tea that exhibits anticancer activity, inhibits angiotensin-converting enzyme (ACE) activity, and promotes apoptosis in Hep G2 and MCF-7 cells.Camellianin A prevents CCl4-induced liver injury by exerting anti-oxidative stress, anti-inflammatory, and anti-apoptotic properties.
    • $400
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  • Cyanidin 3-sambubioside chloride
    TN110433012-73-6
    Cyanidin 3-sambubioside chloride (Cyanidin-3-O-sambubioside chloride) is a plant-derived anthocyanin, an inhibitor of NO and H274Y mutations, and an inhibitor of influenza neuraminidase.Cyanidin 3- sambubioside chloride has anti-inflammatory properties. sambubioside chloride has antioxidant, antiangiogenic and antiviral activities and inhibits angiotensin-converting enzyme (ACE) activity, which can be used in the study of viral infections and cardiovascular diseases.
    • $630
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  • [Sar1, Ile8]-Angiotensin II
    T757537827-06-8
    [Sar1, Ile8]-Angiotensin II(3TFA) is a peptide that has multiple effects on vascular smooth muscle.
    • $48
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  • Leucosceptoside A
    TN443183529-62-8
    Leucosceptoside A shows inhibitory activity against PKCalpha with the IC50 value of 19.0 microM; it also exhibits strong inhibitory capacity against α-glucosidase. Leucosceptoside A has antihypertensive effect, it shows angiotensin converting enzyme (ACE)
    • $698
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  • Olodanrigan
    T44311316755-16-4
    Olodanrigan (EMA401), a highly selective AT2R antagonist, inhibition of augmented AngII/AT2R induced p38 and p42/p44 MAPK activation, and hence inhibition of DRG neuron hyperexcitability and sprouting of DRG neurons. EMA401 blocks p38, p42/p44 mitogen-activated protein kinase (MAPK) activation, neurite outgrowth in adult rat DRG neurons, and sensitization of adult rat and human DRG neurons induced by AngII. It inhibits capsaicin responses in cultured hDRG neurons.
    • $42
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  • BIBS 39
    T3178133085-33-3
    BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist.
    • $36
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  • Tasosartan
    T7797145733-36-4
    Tasosartan (WAY-ANA 756) is an antagonist of angiotensin II type 2 (AT2) receptor (IC50 = 1.2 nM).
    • $51
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