TMA0164 |
15-Hydroxydehydroabietic acid
|
54113-95-0
|
98%
|
|
15-Hydroxydehydroabietic acid exhibits a promising alpha-glucosidase inhibitory activity, it also shows significant antibacterial activities.
|
TN2687 |
2,3',4,6-Tetrahydroxybenzophenone
|
26271-33-0
|
98%
|
|
2,3',4,6-Tetrahydroxybenzophenone possesses significant antioxidant activity.
|
TN3379 |
Allocryptopine
|
24240-04-8
|
98%
|
|
Allocryptopine has certain effects on anti-injury for hepatocyte, ameliorating liver function, and prohibiting hepatic fibrosis; it increases mRNA levels of cyto...
|
TN1378 |
Alpha-Viniferin
|
62218-13-7
|
98%
|
|
Alpha-viniferin is a prostaglandin H2 synthase inhibitor, which has anti-inflammatory, anti-oxidant, anti-arthritis, and anti-tumor activities.
|
TN3294 |
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate
|
67667-71-4
|
98%
|
|
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes.
|
TN3147 |
6',7'-Dihydroxybergamottin
|
264234-05-1
|
98%
|
|
6',7'-Dihydroxybergamottin(DHB), a well-known inhibitor of CYP3A4, the inhibition of CYP3A4 activity by DHB includes the inhibition of POR activity, DHB can inhi...
|
TN3300 |
8alpha-Tigloyloxyhirsutinolide 13-O-acetate
|
83182-58-5
|
98%
|
|
8alpha-Tigloyloxyhirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. 8alpha-Tigloyloxyhirsutinolide 13-O-acetate has ...
|
TN3875 |
Dipterocarpol
|
471-69-2
|
98%
|
|
Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng. Dipterocarpol A shows moderate acetylcholinesterase inhibitory a...
|
TN4130 |
Germacrone 4,5-epoxide
|
92691-35-5
|
98%
|
|
(4S,5S)-(+)-Germacrone-4,5-epoxide inhibits certain subtypes of cytochrome P450 (CYP).
|
TN3627 |
Chalepensin
|
13164-03-9
|
98%
|
|
Chalepensin behaves as an energy transfer inhibitor at low concentration, it inhibits multiple P450s and that epoxidation activity is crucial for the potential d...
|
T10688 |
Casopitant mesylate
|
414910-30-8
|
98%
|
|
Casopitant mesylate (GW679769B) is a selective, brain permeable, and orally active antagonist of neurokinin 1 (NK1) receptor. It is a second in the class of anti...
|
TQ0296 |
N-Nornuciferine
|
4846-19-9
|
98%
|
|
N-Nornuciferine, an aporphine alkaloid in lotus leaf, significantly inhibits CYP2D6 (IC50: 3.76 μM, Ki: 2.34 μM).
|
T10535L |
BI 653048 phosphate
|
1198784-97-2
|
98%
|
|
BI 653048 phosphate is a selective and orally active agonist of nonsteroidal glucocorticoid (GC)(IC50 : 55 nM).
|
TN2144 |
Resveratroloside
|
38963-95-0
|
98%
|
|
Resveratroloside has cardioprotective effect, it exhibits α±-glucosidase inhibitory activity, it also can inhibit hydroxylation of testosterone by CYP3A4.
|
TN1748 |
Humantenirine
|
82375-30-2
|
98%
|
|
Standard reference
|
TN1210 |
2-Hydroxy-1-Methoxyaporphine
|
33770-27-3
|
98%
|
|
2-Hydroxy-1-Methoxyaporphine can inhibit CYP2D6 activity, it also increase the glucose consumption significantly as rosiglitazone.
|
TN3080 |
5,6,7-Trimethoxycoumarin
|
55085-47-7
|
98%
|
|
5,6,7-Trimethoxycoumarin shows moderate inhibitory activity against Micrococcus luteus, it also displays an intermediate cytotoxic effects against brine shrimp l...
|
TN4928 |
Rutacridone
|
17948-33-3
|
98%
|
|
Rutacridone has mutagenicity.
|
T16739 |
RG-12525
|
120128-20-3
|
98%
|
|
RG-12525 is a PPAR-gamma agonist (IC50: appr 60 nM) and a potent inhibitor of CYP3A4 (Ki: 0.5 µM). RG-12525 is a specific and competitive antagonist of the pepti...
|
TQ0276 |
Methysticin
|
20697-20-5
|
98%
|
|
Methysticin, a major kavalactone extracted from kava, can induce CYP1A1.
|