TN2144 |
Resveratroloside
|
38963-95-0
|
|
|
Resveratroloside has cardioprotective effect, it exhibits α±-glucosidase inhibitory activity, it also can inhibit hydroxylation of testosterone by CYP3A4.
|
TN4800 |
Pisatin
|
20186-22-5
|
98%
|
|
Pisatin is an isoflavonoid phytoalexin synthesized by pea (Pisum sativum L.).
|
TN3294 |
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate
|
67667-71-4
|
98%
|
|
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes.
|
TQ0109 |
Cephaeline dihydrochloride
|
5853-29-2
|
98%
|
|
(-)-Cephaeline (dihydrochloride) is an enantiomer of Cephaeline. Cephaeline is a selective CYP2D6 inhibitor (IC50: 121 μM).
|
T10535 |
BI 653048
|
1198784-72-3
|
98%
|
|
BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor.
|
TN4424 |
Lecanoric acid
|
480-56-8
|
98%
|
|
Lecanoric acid shows antioxidant activity with an IC50 value of 79-95 ug/ml, it at 100 ug/ml conc. shows high growth stimulating activity in terms of increased d...
|
TN4277 |
Isocupressic acid
|
1909-91-7
|
98%
|
|
Isocupressic acid induces abortion in pregnant cows when ingested primarily during the last trimester, it decrease affects the angiogenesis of the female reprodu...
|
TMA2106 |
(-)-Sparteine
|
24915-04-6
|
98%
|
|
Sparteine is a class 1a antiarrhythmic agent, a sodium channel blocker. The deficient debrisoquine hydroxylation of Sparteine is due to the absence of P-450IID1 ...
|
TN5278 |
Zederone
|
7727-79-9
|
98%
|
|
Zederone has anti-bacterial activity,it inhibits gram-positive bacteria activity. Zederone induces hepatotoxicity implicated the induction of Cyps, which leads t...
|
TN3300 |
8alpha-Tigloyloxyhirsutinolide 13-O-acetate
|
83182-58-5
|
98%
|
|
8alpha-Tigloyloxyhirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. 8alpha-Tigloyloxyhirsutinolide 13-O-acetate has ...
|
TMA0164 |
15-Hydroxydehydroabietic acid
|
54113-95-0
|
98%
|
|
15-Hydroxydehydroabietic acid exhibits a promising alpha-glucosidase inhibitory activity, it also shows significant antibacterial activities.
|
TN2147 |
Retrorsine
|
480-54-6
|
98%
|
|
Retrorsine selectively inhibits hepatocyte proliferation and following liver injury evokes small hepatocyte-like progenitor cells. Retrorsine can be used for the...
|
T10891 |
CRTH2-IN-1
|
926661-54-3
|
98%
|
|
CRTH2-IN-1 is a selective prostaglandin D2 receptor DP2 (CRTH2) antagonist, a Ramatroban analog, with an IC50 of 6 nM in the human DP2 binding assay.
|
TN1378 |
α-Viniferin
|
62218-13-7
|
98%
|
|
α-Viniferin belongs to a class of organic compounds, also known as 2-arylbenzofuran flavonoids, that are inhibitors of prostaglandin H2 synthetase. α-Viniferin h...
|
TN3080 |
5,6,7-Trimethoxycoumarin
|
55085-47-7
|
98%
|
|
5,6,7-Trimethoxycoumarin shows moderate inhibitory activity against Micrococcus luteus, it also displays an intermediate cytotoxic effects against brine shrimp l...
|
T6051 |
Orteronel
|
566939-85-3
|
98%
|
|
Orteronel ((S)-Orteronel)(TAK-700) was selected as a candidate for clinical evaluation. orteronel (TAK-700) is currently in phase III clinical trials for the tre...
|
T11964 |
MCH-1 antagonist 1
|
1039825-68-7
|
98%
|
|
MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).
|
TQ0296 |
N-Nornuciferine
|
4846-19-9
|
98%
|
|
N-Nornuciferine, an aporphine alkaloid in lotus leaf, significantly inhibits CYP2D6 (IC50: 3.76 μM, Ki: 2.34 μM).
|
TN4928 |
Rutacridone
|
17948-33-3
|
98%
|
|
Rutacridone has mutagenicity.
|
TN2687 |
2,3',4,6-Tetrahydroxybenzophenone
|
26271-33-0
|
98%
|
|
2,3',4,6-Tetrahydroxybenzophenone possesses significant antioxidant activity.
|