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Search Result

Search Results for " non-competitive "

Targets

Adrenergic Receptor

198

Compounds

27

Natural Products

2

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T8580 Bupranolol Adrenergic Receptor
Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.
T8459 DNQX disodium salt DNQX Disodium NMDAR , iGluR
DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor
T7304 DNQX FG 9041 GluR , iGluR
DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)
T1817 GNF-2 GNF2 SARS-CoV , Bcr-Abl
GNF-2 is a highly selective non-ATP competitive inhibitor of Bcr-Abl.
T23524 W-84 dibromide HDMPPA AChR
W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.
T6223 U0126-EtOH U0126 Ethanol,U0126 Mitophagy , Influenza Virus , MEK , Autophagy
U0126-EtOH (U0126 Ethanol) is a non-ATP competitive specific inhibitor of MEK1/2 (IC50: 0.07/0.06 μM).
T6893 MK-886 MK886,L 663536 Apoptosis , Leukotriene Receptor , COX , PPAR , FLAP
MK-886 (L 663536) is an inhibitor of leukotriene biosynthesis, inhibiting 5-lipoxygenase-activating protein (FLAP). It is also a moderately potent PPARα antagonist.
T10898 Samuraciclib hydrochloride ICEC0942 hydrochloride,CT7001 hydrochloride Apoptosis , CDK
Samuraciclib hydrochloride (ICEC0942 hydrochloride) is a potent, selective, ATP competitive and oral active CDK7 inhibitor with IC50 of 41 nM. The selectivity of Samuraciclib hydrochloride is 45-, 15-, 230- and 30-fold h...
T10774 CFM-2 iGluR
CFM-2, a potent and selective non-competitive antagonist of AMPAR (AMPAR), exhibits anticonvulsant activity across various seizure models.
T22346 Indomethacin sodium hydrate Indometacin Sodium COX
Indomethacin Sodium is the sodium salt of indomethacin, which is a non-selective, competitive, and reversible, inhibitor of cyclooxygenases 1 and 2 with analgesic-antipyretic, anti-inflammatory, and tocolytic effects.
TP2058L Catestatin acetate Catestatin acetate(142211-96-9 free base) Endogenous Metabolite , AChR
Catestatin acetate is a non-competitive antagonist of nAChR and inhibits catecholamine release. Catestatin acetate regulates cardiac function and blood pressure.
T26645 Aptiganel CNS 1102,CNS-1102,CNS1102 NMDAR
Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.
T2362 QNZ46 NMDAR , iGluR
QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.
T22692 CPCCOEt GluR
CPCCOEt is a low affinity, selective, non-competitive and reversible antagonist of mGluR1b
T23588 9-CP-Ade Mesylate 9-Cyclopentyladenine monomethanesulfonate,9 CP Ade Mesylate,9CPAde Mesylate AChR
9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.
T14988 CMPD1 MAPK
CMPD1 is a non-ATP-competitive p38 MAPK-mediated MK2 phosphorylation inhibitor(apparent Ki (Kiapp): 330 nM).
T8685 SP-146 Aurora Kinase
SP-146 is a selective, potent and non-ATP-competitive Aurora B inhibitor(IC50 : 0.316 nM).
T23048 N20C hydrochloride 2-((3,3-diphenylpropyl)amino)acetamide hydrochloride NMDAR
N20C hydrochloride (2-((3,3-diphenylpropyl)amino)acetamide hydrochloride) is a non-competitive NMDA receptor open-channel blocker.
T5053 Eprobemide LIS 630 MAO , Monoamine Oxidase
Eprobemide (LIS 630) is a non-competitive reversible inhibitor of monoamine oxidase A (MAO-A).
T6083 AZD8330 ARRY-424704,ARRY-704 ERK , MEK
AZD8330 (ARRY-704) is a novel, selective, non-ATP competitive MEK 1/2 inhibitor with IC50 of 7 nM. Phase 1.
T2380 BIBR 1532 Apoptosis , Telomerase
BIBR 1532 is an effective, specific and non-competitive telomerase inhibitor (IC50: 100 nM, in a cell-free assay).
T8458 CNQX disodium iGluR
CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.
T25276 Crilvastatin PMD387,PMD 387,PMD-387 HMG-CoA Reductase
Crilvastatin (PMD 387) is a novel non-competitive hydroxymethylglutaryl coenzyme A reductase inhibitor with cholesterol-lowering activity that inhibits cholesterol uptake in rats with hereditary hypercholesterolemia.
T15301 Fluspirilene Redeptin,R 6218 Calcium Channel
Fluspirilene (R 6218) is a non-competitive L-type calcium channel antagonist (IC50: 0.03 μM).Fluspirilene is a long-acting antipsychotic compound used in the treatment of schizophrenia.
T7515 MTEP hydrochloride 3-((2-Methyl-1,3-thiazol-4-yl)ethyn-yl)pyridine hydrochloride,MTEP GluR
MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)
T6546 IPA-3 IPA3,IPA 3 PAK
IPA-3 is a selective non-ATP competitive Pak1 inhibitor with IC50 of 2.5 μM, no inhibition to group II PAKs (PAKs 4-6).
T12205 Ned 19 Calcium Channel
Ned 19 is a selective membrane-permeant non competitive antagonist of NAADP and strongly inhibits tumor growth and vascularization as well as lung metastases in mice.
T21152 Ac-Phe-NH2 Ac-Phe NH2,Ac Phe NH2,Ac Phe-NH2 Others
Ac-Phe-NH2 is a non-competitive inhibitor of polyubiquitin chain elongation at Ki value of 8 ± 1.2 mM.
T2443 CI-1040 PD 184352 Apoptosis , MEK
CI-1040 (PD 184352) (PD184352) is an ATP non-competitive MEK1/2 inhibitor (IC50: 17 nM).
T0245 RS 61443 RS61443,Mycophenolate mofetil,TM-MMF Dehydrogenase
RS 61443 (Mycophenolate mofetil) is an immunosuppressant, a non-competitive, selective and reversible inhibitor of inosine monophosphate dehydrogenase (IMPDH)
T16560 Poloxin PLK
Poloxin is a non-ATP competitive Polo-like Kinase 1 inhibitor. It targets the polo-box domain (IC50: appr 4.8 μM).
T6287 Tariquidar XR9576 P-gp
Tariquidar (XR9576)(Kd=5.1 nM) is a specific and effective non-competitive inhibitor of P-glycoprotein. It can reverse drug resistance in MDR cell Lines.
T24906L Tuna AI acetate Angiotensin-converting Enzyme (ACE)
Tuna AI acetate is an inhibitor of angiotensin-converting enzyme (ACE) in non-competitive manner derived from tuna muscle.
T3067 Tideglusib NP-12,NP031112 GSK-3
Tideglusib (NP031112), a non-ATP competitive inhibitor of glycogen synthase kinase 3 (GSK-3), is with anti-inflammatory and neuroprotective activities.
T2463 ML141 CID-2950007 Apoptosis , CDK , Ras
ML141 (CID-2950007) is an effective, specific and reversible non-competitive inhibitor of Rho family GTPase cdc42 (IC50: 200 nM).
T9773 Thioquinapiperifil dihydrochloride KF-31327 PDE
Thioquinapiperifil dihydrochloride is a phosphodiesterase (PDE-5) inhibitor (IC50: 0.074 nM) that is potent, selective and non-competitive for investigational maturation.
T26520 ABP688 ABP-688,ABP 688 GluR
ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.
T7178 CNQX FG9065 GluR , iGluR
CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)
T6636 Refametinib BAY 86-97661,BAY 869766,RDEA119 MEK
Refametinib (RDEA119) (RDEA119, Bay 86-9766) is an effective, ATP non-competitive and specific inhibitor of MEK1/2 (IC50: 19/47 nM).
T26891 BPDBA GABA Receptor
BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and mouse GAT2, with IC50 values of 20 μM and 35 μM, respectivel...
T2497 MPEP hydrochloride GluR
MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).
T4354 KPT9274 KPT-9274,KPT 9274,PAK4-IN-1 NAMPT , PAK
KPT9274 (PAK4-IN-1) is a non-competitive dual inhibitor of PAK4 and NAMPT(IC50= ~120 nM). It is an orally bioavailable small molecule.
T4442 MK2-IN-1 hydrochloride MK2 Inhibitor,MK 25 MAPK
MK2-IN-1 hydrochloride (MK 25) is a highly selective, non-ATP competitive inhibitor of p38/mitogen-activated protein kinase-activated protein kinase 2 (MAPKAPK2 or MK2, IC50: 0.11 μM) [1].
T16964 SYM2206 SYM-2206,SYM 2206 Sodium Channel , iGluR
SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated sustained currents and decreasing the survival of pancreati...
T22893 L-168049 L-168,049 Glucagon Receptor
L-168049 is a selective and non-competitive antagonist of human glucagon receptor with IC50s of 3.7 nM, 63 nM, and 60 nM for human, murine, and canine, respectively.
T10066 2',5'-Dideoxyadenosine Adenylyl cyclase , Adrenergic Receptor , AChR
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
T73331 GSK3-IN-3 Mitophagy , GSK-3
GSK3-IN-3 is a mitochondrial autophagy (mitophagy) inducer and GSK-3 inhibitor (IC50: 3.01 μM) that induces parkin-dependent mitochondrial autophagy. GSK3-IN-3 is non-ATP and non-substrate competitive and neuroprotective...
T15387 GLP-1R Antagonist 1 Glucagon Receptor
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).
T77679 HPL-IN-2 Others
hPL-IN-2 is a potent, reversible and non-competitive inhibitor of Pancreatic lipase (IC50: 1.63 μM) that can be used to investigate obesity-related diseases.
T7157 XY1 Histone Methyltransferase
XY1 is a very close analogue of SGC707 (a potent, selective, and non-competitive inhibitor of PRMT3 with IC50 of 31 nM), It is intended to be used as a negative control for SGC707 in studies involving PRMT3 action.

Compounds

Bupranolol
T8580
Synonym:
Target: Adrenergic Receptor
DNQX disodium salt
T8459
Synonym: DNQX Disodium
Target: NMDAR, iGluR
DNQX
T7304
Synonym: FG 9041
Target: GluR, iGluR
GNF-2
T1817
Synonym: GNF2
Target: SARS-CoV, Bcr-Abl
W-84 dibromide
T23524
Synonym: HDMPPA
Target: AChR
U0126-EtOH
T6223
Synonym: U0126 Ethanol,U0126
Target: Mitophagy, Influenza Virus, MEK, Autophagy
MK-886
T6893
Synonym: MK886,L 663536
Target: Apoptosis, Leukotriene Receptor, COX, PPAR, FLAP
Samuraciclib hydrochloride
T10898
Synonym: ICEC0942 hydrochloride,CT7001 hydrochloride
Target: Apoptosis, CDK
CFM-2
T10774
Synonym:
Target: iGluR
Indomethacin sodium hydrate
T22346
Synonym: Indometacin Sodium
Target: COX
Catestatin acetate
TP2058L
Synonym: Catestatin acetate(142211-96-9 free base)
Target: Endogenous Metabolite, AChR
Aptiganel
T26645
Synonym: CNS 1102,CNS-1102,CNS1102
Target: NMDAR
QNZ46
T2362
Synonym:
Target: NMDAR, iGluR
CPCCOEt
T22692
Synonym:
Target: GluR
9-CP-Ade Mesylate
T23588
Synonym: 9-Cyclopentyladenine monomethanesulfonate,9 CP Ade Mesylate,9CPAde Mesylate
Target: AChR
CMPD1
T14988
Synonym:
Target: MAPK
SP-146
T8685
Synonym:
Target: Aurora Kinase
N20C hydrochloride
T23048
Synonym: 2-((3,3-diphenylpropyl)amino)acetamide hydrochloride
Target: NMDAR
Eprobemide
T5053
Synonym: LIS 630
Target: MAO, Monoamine Oxidase
AZD8330
T6083
Synonym: ARRY-424704,ARRY-704
Target: ERK, MEK
BIBR 1532
T2380
Synonym:
Target: Apoptosis, Telomerase
CNQX disodium
T8458
Synonym:
Target: iGluR
Crilvastatin
T25276
Synonym: PMD387,PMD 387,PMD-387
Target: HMG-CoA Reductase
Fluspirilene
T15301
Synonym: Redeptin,R 6218
Target: Calcium Channel
MTEP hydrochloride
T7515
Synonym: 3-((2-Methyl-1,3-thiazol-4-yl)ethyn-yl)pyridine hydrochloride,MTEP
Target: GluR
IPA-3
T6546
Synonym: IPA3,IPA 3
Target: PAK
Ned 19
T12205
Synonym:
Target: Calcium Channel
Ac-Phe-NH2
T21152
Synonym: Ac-Phe NH2,Ac Phe NH2,Ac Phe-NH2
Target: Others
CI-1040
T2443
Synonym: PD 184352
Target: Apoptosis, MEK
RS 61443
T0245
Synonym: RS61443,Mycophenolate mofetil,TM-MMF
Target: Dehydrogenase
Poloxin
T16560
Synonym:
Target: PLK
Tariquidar
T6287
Synonym: XR9576
Target: P-gp
Tuna AI acetate
T24906L
Synonym:
Target: Angiotensin-converting Enzyme (ACE)
Tideglusib
T3067
Synonym: NP-12,NP031112
Target: GSK-3
ML141
T2463
Synonym: CID-2950007
Target: Apoptosis, CDK, Ras
Thioquinapiperifil dihydrochloride
T9773
Synonym: KF-31327
Target: PDE
ABP688
T26520
Synonym: ABP-688,ABP 688
Target: GluR
CNQX
T7178
Synonym: FG9065
Target: GluR, iGluR
Refametinib
T6636
Synonym: BAY 86-97661,BAY 869766,RDEA119
Target: MEK
BPDBA
T26891
Synonym:
Target: GABA Receptor
MPEP hydrochloride
T2497
Synonym:
Target: GluR
KPT9274
T4354
Synonym: KPT-9274,KPT 9274,PAK4-IN-1
Target: NAMPT, PAK
MK2-IN-1 hydrochloride
T4442
Synonym: MK2 Inhibitor,MK 25
Target: MAPK
SYM2206
T16964
Synonym: SYM-2206,SYM 2206
Target: Sodium Channel, iGluR
L-168049
T22893
Synonym: L-168,049
Target: Glucagon Receptor
2',5'-Dideoxyadenosine
T10066
Synonym:
Target: Adenylyl cyclase, Adrenergic Receptor, AChR
GSK3-IN-3
T73331
Synonym:
Target: Mitophagy, GSK-3
GLP-1R Antagonist 1
T15387
Synonym:
Target: Glucagon Receptor
hPL-IN-2
T77679
Synonym:
Target: Others
XY1
T7157
Synonym:
Target: Histone Methyltransferase
1 2 3 4
Cat No. Product Name Synonyms Targets
T11054 DL-Norvaline 2-Aminopentanoic acid Arginase , Endogenous Metabolite
DL-Norvaline (2-Aminopentanoic acid) is a non-competitive inhibitor of arginase.
T3419 Chelerythrine chloride Apoptosis , BCL , PKC , Autophagy
Chelerythrine Chloride is a cell-permeable inhibitor of protein kinase C, competitive with respect to the phosphate acceptor and non-competitive with respect to ATP.
T1680 Tolazoline hydrochloride Imidaline hydrochloride,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride) Adrenergic Receptor
Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn.
T3379 Decanoic Acid Decoic acid,CAPRIC ACID,Caprynic acid GluR , iGluR
Decanoic Acid (Caprynic acid) acts as a non-competitive AMPA receptor antagonist.
TJS0851 Plantagoside Others
Plantagoside is a specific non-competitive inhibitor for jack bean alpha-mannosidase (IC50: 5 μM). It also is a potent inhibitor of the Maillard reaction.
T8319 Butyl isobutyl phthalate ButylIsobutylPhthalate Glucosidase
Butyl isobutyl phthalate (ButylIsobutylPhthalate) is a non-competitive α-glucosidase inhibitor(IC50 :38 μM),it shows a hypoglycemic effect
T8044 Ajmalicine Lamuran,Delta-Yohimbine,Raubasine,Ajmalicin Adrenergic Receptor
Ajmalicine (Raubasine) (Raubasine) is a potent adrenolytic agent which preferentially blocks α1-adrenoceptor. Ajmalicine is an reversible but non-competitive nicotine receptor full inhibitor, IC50 = 72.3 μM. Ajmalicine a...
T25192 Butyrolactone I Olomoucin CDK
Butyrolactone I (Olomoucin) is an ATP-competitive inhibitor of CDK and cdc2 kinase family. Butyrolactone I shows antitumor effects in non-small cell lung, small cell lung, and prostate cancer cell lines.
T6680 Staurosporine Antibiotic AM-2282,AM-2282,CGP 41251 Apoptosis , PKA , Antibacterial , Antibiotic , Src , PKC , Antifungal
Staurosporine (AM-2282) is a protein kinase inhibitor with ATP-competitive and non-selective inhibitory activity (IC50=6/15/2/3/3000 nM) against PKC, PKA, c-Fgr, phosphorylase kinase and TAOK2. Staurosporine also induces...
TN1343 8-Geranyloxypsoralen Anti-infection , P450 , BACE
8-Geranyloxypsoralen inhibits α2-secretase (BACE1) activity in non-competitive manner, with the IC(50) values <25.0 μM, it can induce vasorelaxation on rat arterial tissues. 8-Geranyloxypsoralen possesses nematicidal act...
TN4660 Niranthin Anti-infection , HBV , PAFR , Topoisomerase
Niranthin is a potent anti-leishmanial agent, inhibits the relaxation activity of heterodimeric type IB topoisomerase of L. donovani and acts as a non-competitive inhibitor interacting with both subunits of the enzyme. N...
T6S0659 Rhynchophylline Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin Calcium Channel , NF-κB
1. Rhynchophylline (Mitrinermine) can protect against ischemic damage, probably via regulating the Akt/mTOR pathway. 2. Rhynchophylline can protect against glutamate-induced neuronal death, can inhibit MA impairment in c...
T4S1619 L-Hyoscyamine sulfate Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate AChR
L-Hyoscyamine sulfate (Levsin Sulfate) is the sulfate salt of a belladonna alkaloid derivative and the levorotatory form of racemic atropine isolated from the plants Hyoscyamus niger or Atropa belladonna, which exhibits ...
T0962 L-Hyoscyamine Daturine,Hyoscyamine AChR
L-Hyoscyamine (Daturine) functions as a non-selective, competitive antagonist of muscarinic receptors, thereby inhibiting the parasympathetic activities of acetylcholine on the salivary, bronchial, and sweat glands, as w...
T13752 L-(+)-Arabinose Endogenous Metabolite
L-(+)-Arabinose selectively inhibits intestinal sucrase activity in a non-competitive manner, inhibiting glucose elevation caused by sucrose intake.
TN3013 4,5-Dimethoxycanthin-6-one Methylnigakinone P450 , Antibacterial , PDE
4,5-Dimethoxycanthin-6-one is an alkaloid isolated from Picrasma quassioides BENNET (Simaroubaceae).4,5-Dimethoxycanthin-6-one was isolated from Picrasma quassioides BENNET (Simaroubaceae) with antimicrobial activity.4,5...
T39025 Adenosine 2',5'-diphosphate sodium
Adenosine 2',5'-diphosphate sodium is a competitive P2Y1 antagonist with non-selective antagonism at recombinant and human platelet P2X1 receptors.
TN4571 Mirabijalone D Beta Amyloid
Mirabijalone D is a non-competitive inhibitor based on the Dixon plot.It inhibits Aβ1-42 production by 43.7% in APPSW-N2a cells.
T2S0118 Daurinoline Calcium Channel , 5-HT Receptor , Histamine Receptor
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a protective function on microcirculation of cerebral pia mat...
T8214 Kushenol E Flemiphilippinin D IDO , Indoleamine 2,3-Dioxygenase (IDO)
Kushenol E (Flemiphilippinin D) is a class of flavonoids isolated from Sophora flavescens. It is a non-competitive IDO1 inhibitor (IC50: 7.7 μM, Ki: 9.5 μM), has anti-tumor activity.
TN3383 α-Amyrin palmitate alpha-Amyrin palmitate PKA
alpha-Amyrin palmitate is antiarthritic in the adjuvant model of arthritis in rats. alpha-Amyrin palmitate is a potent non-competitive inhibitor of chymotrypsin (Ki=6 microM), it also shows weak cytotoxicity against the ...
T8306 Epiberberine chloride Epiberberine (chloride) Reactive Oxygen Species , Beta-Secretase , BACE , AChR , AChE
Epiberberine chloride (Epiberberine (chloride)) is an alkaloid isolated from Coptis chinensis, acts as a potent AChE and BChE inhibitor, and a non-competitive BACE1 inhibitor (IC50s: 1.07, 6.03 and 8.55 μM).
TN2517 1,7-Dihydroxy-2,3-dimethoxyxanthone Others
1,7-Dihydroxy-2,3-dimethoxyxanthone may have medicinal use in the management of inflammation, asthma and allergy, it antagonises in a non competitive but, reversible manner the contractions induced by chemical inflammato...
T73202 BChE-IN-11
BChE-IN-11, a selective and non-competitive inhibitor of butyrylcholinesterase (BChE), demonstrates potent activity with an inhibitory concentration (IC50) of 2.1 μM. This compound is applicable in Alzheimer's disease (A...
T75513 BChE-IN-12
BChE-IN-12, also known as compound 12, is a potent non-competitive inhibitor of butyrylcholinesterase (BChE) with an IC50 value of 2.3 μM. Derived from Bletilla striata, it is utilised in research related to Alzheimer's ...
T37774 Thielavin A
Thielavin A is a fungal metabolite originally isolated from T. terricola that is related to thielavin B . Thielavin A inhibits COX, blocking both the conversion of arachidonic acid to prostaglandin H2 and the conversion ...
T69254 Ajmalicine hydrochloride Raubasine hydrochloride
Ajmalicine (Raubasine) hydrochloride, a potent adrenolytic compound, selectively inhibits α1-adrenoceptors and acts as a reversible, non-competitive full inhibitor of nicotine receptors with an IC50 of 72.3 μM. This chem...

Natural Products

DL-Norvaline
T11054
Synonym: 2-Aminopentanoic acid
Target: Arginase, Endogenous Metabolite
Chelerythrine chloride
T3419
Synonym:
Target: Apoptosis, BCL, PKC, Autophagy
Tolazoline hydrochloride
T1680
Synonym: Imidaline hydrochloride,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)
Target: Adrenergic Receptor
Decanoic Acid
T3379
Synonym: Decoic acid,CAPRIC ACID,Caprynic acid
Target: GluR, iGluR
Plantagoside
TJS0851
Synonym:
Target: Others
Butyl isobutyl phthalate
T8319
Synonym: ButylIsobutylPhthalate
Target: Glucosidase
Ajmalicine
T8044
Synonym: Lamuran,Delta-Yohimbine,Raubasine,Ajmalicin
Target: Adrenergic Receptor
Butyrolactone I
T25192
Synonym: Olomoucin
Target: CDK
Staurosporine
T6680
Synonym: Antibiotic AM-2282,AM-2282,CGP 41251
Target: Apoptosis, PKA, Antibacterial, Antibiotic, Src, PKC, Antifungal
8-Geranyloxypsoralen
TN1343
Synonym:
Target: Anti-infection, P450, BACE
Niranthin
TN4660
Synonym:
Target: Anti-infection, HBV, PAFR, Topoisomerase
Rhynchophylline
T6S0659
Synonym: Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin
Target: Calcium Channel, NF-κB
L-Hyoscyamine sulfate
T4S1619
Synonym: Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate
Target: AChR
L-Hyoscyamine
T0962
Synonym: Daturine,Hyoscyamine
Target: AChR
L-(+)-Arabinose
T13752
Synonym:
Target: Endogenous Metabolite
4,5-Dimethoxycanthin-6-one
TN3013
Synonym: Methylnigakinone
Target: P450, Antibacterial, PDE
Adenosine 2',5'-diphosphate sodium
T39025
Synonym:
Target:
Mirabijalone D
TN4571
Synonym:
Target: Beta Amyloid
Daurinoline
T2S0118
Synonym:
Target: Calcium Channel, 5-HT Receptor, Histamine Receptor
Kushenol E
T8214
Synonym: Flemiphilippinin D
Target: IDO, Indoleamine 2,3-Dioxygenase (IDO)
α-Amyrin palmitate
TN3383
Synonym: alpha-Amyrin palmitate
Target: PKA
Epiberberine chloride
T8306
Synonym: Epiberberine (chloride)
Target: Reactive Oxygen Species, Beta-Secretase, BACE, AChR, AChE
1,7-Dihydroxy-2,3-dimethoxyxanthone
TN2517
Synonym:
Target: Others
BChE-IN-11
T73202
Synonym:
Target:
BChE-IN-12
T75513
Synonym:
Target:
Thielavin A
T37774
Synonym:
Target:
Ajmalicine hydrochloride
T69254
Synonym: Raubasine hydrochloride
Target:

Recombinant Proteins

Species：
Human (2)
Expression System：
E. coli (1)
Yeast (1)
Tag：
N-6His (1)
N-terminal 6xHis-tagged (1)
Cat No. Product Name Species Expression System
TMPJ-00473 QPRTase Protein, Human, Recombinant (His) Human E. coli
Nicotinate-Nucleotide Pyrophosphorylase (QPRT) belongs to the nadC/modD family. QPRT plays an improtant role in catabolism of quinolinate which acts as a potent endogenous exitotoxin to neurons. In addition, QPRT serves ...
TMPH-01092 CHGA Protein, Human, Recombinant (His) Human Yeast
Strongly inhibits glucose induced insulin release from the pancreas.; Inhibits catecholamine release from chromaffin cells and noradrenergic neurons by acting as a non-competitive nicotinic cholinergic antagonist. Displa...
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