Shopping Cart

Remove All
Your shopping cart is currently empty

Aptiganel hydrochloride

Name: Aptiganel hydrochloride
Brand: TargetMol
SKU: T38068
Price: 30 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T38068Cas No. 137160-11-3

Alias CNS 1102, Cerestat

Aptiganel hydrochloride（Cerestat） is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.

Aptiganel hydrochloride

🥰Excellent

Purity: 99.89%

Catalog No. T38068Alias CNS 1102, CerestatCas No. 137160-11-3

Pack Size	Price	Availability
1 mg	$30	In Stock
5 mg	$64	In Stock
10 mg	$113	In Stock
25 mg	$247	In Stock
50 mg	$428	In Stock
100 mg	$691	In Stock
200 mg	$983	In Stock
1 mL x 10 mM (in DMSO)	$71	In Stock

Add to Cart

Add to Quotation

Bulk & Custom

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

Select Batch

Purity:99.89%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	Aptiganel hydrochloride（Cerestat） is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.
Synonyms	CNS 1102, Cerestat

Chemical Properties

Molecular Weight	339.86
Formula	C₂₀H₂₂ClN₃
Cas No.	137160-11-3
Smiles	Cl.N=C(NC1=CC=CC=2C=CC=CC21)N(C3=CC=CC(=C3)CC)C

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 80.00 mg/mL (235.39 mM), Sonication is recommended.

H2O: 5.00 mg/mL (14.71 mM), Sonication is recommended.

Solution Preparation Table

H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	2.9424 mL	14.7119 mL	29.4239 mL	147.1194 mL
5 mM	0.5885 mL	2.9424 mL	5.8848 mL	29.4239 mL
10 mM	0.2942 mL	1.4712 mL	2.9424 mL	14.7119 mL

DMSO

	1mg	5mg	10mg	50mg
20 mM	0.1471 mL	0.7356 mL	1.4712 mL	7.3560 mL
50 mM	0.0588 mL	0.2942 mL	0.5885 mL	2.9424 mL
100 mM	0.0294 mL	0.1471 mL	0.2942 mL	1.4712 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc