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GABA Receptor

The GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels (also known as ionotropic receptors); whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors.
Cat. No. Product name CAS No. Purity Chemical Structure
T10456 Bamaluzole 87034-87-5 98%
Bamaluzole is an agonist of GABA receptor extracted from patent WO 2012064642 A1.
T4S1616 Sanggenon D 81422-93-7 98%
Sanggenone D represents a new scaffold of positive GABAA receptor modulators, it also inhibits COX-2 activity (IC 50 = 73-100 μM). Sanggenone D has anti-inflamma...
T0128L Vigabatrin Hydrochloride 1391054-02-6 98%
Vigabatrin HCl is a structural analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA), which irreversibly inhibits the catabolism of GABA by GABA t...
TN1591 DL-Menthol 15356-70-4 98%
DL-Menthol has short term toxicity in rats, it plays a role in the induction of surgical anesthesia in fishes, related at least in part to the activation of GABA...
TN4440 Limonexic acid 99026-99-0 98%
Limonexic acid shows antinociceptive actions , it produces dose-related inhibition of glutamate- and capsaicin-induced pain. Limonexic acid can effectively prote...
T12044 (-)-Bicuculline methochloride 53552-05-9 98%
(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.
T15737 Lesogaberan 344413-67-8 98%
Lesogaberan is an effective and selective GABAB receptor agonist (EC50: 8.6 nM for human recombinant GABAB receptors). For rat brain GABAB and GABAA receptors, t...
TN1202 (-)-α-Pinene 7785-26-4 98%

(1S)-(-)-Alpha-Pinene is a natural product

T40659L γ-Acetylenic GABA hydrochloride 103451-26-9 98%
γ-Acetylenic GABA hydrochloride is a GABA transaminase inhibitor.
T12867L SCH 50911 733717-87-8 98%
SCH 50911 is (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid and is a selective, orally-active and competitive γ-Aminobutyric acid B GABA(B) receptor antagonist, b...
T15380 Gidazepam 129186-29-4 98%
Gidazepam is an GABA receptor channels agonist.
T11686 Isotanshinone I 20958-17-2 98%
Isotanshinone I with IC50s of 1.13 μM and 0.432 μM for α-glucosidase and AGE, respectively. Isotanshinone I has inhibitory activity against α-glucosidase and for...
T3173 DAA-1106 220551-92-8 98%
DAA1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR), acting as a potent and selective agonist at the peripheral benzodiazepine ...
T12867 SCH 50911 hydrochloride 160415-07-6 98%
SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).
T9424 Temgicoluril 10095-06-4 98%
Temgicoluril acts on GABA Receptor.
T12043 (-)-Bicuculline methobromide 73604-30-5 98%
(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .
T13150 THIP 64603-91-4 98%
THIP is a selective agonist of δ-aminobutyric acid type A receptor (δ-GABAAR),and exhibits agonism at α4β1δ, α4β3δ and weak antagonism at αβγ and α4β2δ GABAARs.
TN4322 Isopulegol 7786-67-6 98%
Isopulegol presents depressant- and anxiolytic-like effects, it also has anticonvulsant and bioprotective effects against PTZ-induced convulsions are possibly re...
T11061 DMCM hydrochloride 1215833-62-7 98%
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine. DMCM showed significant differences in human recombinant GABAA zaerxep3 receptor s...
T17306 (R)-Baclofen hydrochloride 63701-55-3 98%
Arbaclofen hydrochloride, a Gamma-Aminobutyric Acid derivative, is a specific agonist of GABA-B receptors, it is used to treat spasticity, especially that due to...
Bamaluzole
T10456
Bamaluzole is an agonist of GABA receptor extracted from patent WO 2012064642 A1.
Sanggenon D
T4S1616
Sanggenone D represents a new scaffold of positive GABAA receptor modulators, it also inhibits COX-2 activity (IC 50 = 73-100 μM). Sanggenone D has anti-inflamma...
Vigabatrin Hydrochloride
T0128L
Vigabatrin HCl is a structural analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA), which irreversibly inhibits the catabolism of GABA by GABA t...
DL-Menthol
TN1591
DL-Menthol has short term toxicity in rats, it plays a role in the induction of surgical anesthesia in fishes, related at least in part to the activation of GABA...
Limonexic acid
TN4440
Limonexic acid shows antinociceptive actions , it produces dose-related inhibition of glutamate- and capsaicin-induced pain. Limonexic acid can effectively prote...
(-)-Bicuculline methochloride
T12044
(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.
Lesogaberan
T15737
Lesogaberan is an effective and selective GABAB receptor agonist (EC50: 8.6 nM for human recombinant GABAB receptors). For rat brain GABAB and GABAA receptors, t...
(-)-α-Pinene
TN1202
<p>(1S)-(-)-Alpha-Pinene is a natural product</p>
γ-Acetylenic GABA hydrochloride
T40659L
γ-Acetylenic GABA hydrochloride is a GABA transaminase inhibitor.
SCH 50911
T12867L
SCH 50911 is (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid and is a selective, orally-active and competitive γ-Aminobutyric acid B GABA(B) receptor antagonist, b...
Gidazepam
T15380
Gidazepam is an GABA receptor channels agonist.
Isotanshinone I
T11686
Isotanshinone I with IC50s of 1.13 μM and 0.432 μM for α-glucosidase and AGE, respectively. Isotanshinone I has inhibitory activity against α-glucosidase and for...
DAA-1106
T3173
DAA1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR), acting as a potent and selective agonist at the peripheral benzodiazepine ...
SCH 50911 hydrochloride
T12867
SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).
Temgicoluril
T9424
Temgicoluril acts on GABA Receptor.
(-)-Bicuculline methobromide
T12043
(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .
THIP
T13150
THIP is a selective agonist of δ-aminobutyric acid type A receptor (δ-GABAAR),and exhibits agonism at α4β1δ, α4β3δ and weak antagonism at αβγ and α4β2δ GABAARs.
Isopulegol
TN4322
Isopulegol presents depressant- and anxiolytic-like effects, it also has anticonvulsant and bioprotective effects against PTZ-induced convulsions are possibly re...
DMCM hydrochloride
T11061
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine. DMCM showed significant differences in human recombinant GABAA zaerxep3 receptor s...
(R)-Baclofen hydrochloride
T17306
Arbaclofen hydrochloride, a Gamma-Aminobutyric Acid derivative, is a specific agonist of GABA-B receptors, it is used to treat spasticity, especially that due to...
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