T13393 |
ZEN-3411
|
1952264-36-6
|
98%
|
|
ZEN-3411 is an inhibitor of BET(IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively). ZEN-3411 can be used to form PROTACs to...
|
T13412L |
ZM223 hydrochloride (2031177-48-5 free base)
|
T13412L
|
98%
|
|
ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.
|
T13567 |
BCX 1470 methanesulfonate
|
217099-44-0
|
98%
|
|
BCX 1470 methanesulfonate inhibits the esterolytic activity of factor D and C1s (IC50: 96 nM and 1.6 nM), 3.4- and 200-fold better than that of trypsin, respecti...
|
T13568 |
BCX 1470
|
217099-43-9
|
98%
|
|
BCX 1470 inhibits the esterolytic activity of factor D and C1s (IC50: 96 nM and 1.6 nM), 3.4- and 200-fold better than that of trypsin, respectively.
|
T17288 |
ZD8321
|
182073-77-4
|
98%
|
|
ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).
|
T15285 |
FK706
|
144055-55-0
|
98%
|
|
FK706 is a slow-binding and competitive human neutrophil elastase inhibitor (IC50: 83 nM; Ki: 4.2 nM). FK706 also inhibits mouse neutrophil elastase and porcine ...
|
T22451 |
UK-371804 HCl
|
256476-36-5
|
98%
|
|
UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-fol...
|
T10254 |
AE-3763
|
291778-77-3
|
98%
|
|
AE-3763 is a peptide-based human neutrophil elastase inhibitor (IC50: 29 nM).
|
T20992 |
MEGA-9
|
85261-19-4
|
98%
|
|
MEGA-9 solubilizes membrane protein and can be used as a nonionic detergent.
|
T13408 |
ZK824190
|
2254001-81-3
|
98%
|
|
ZK824190 is an orally available and selective inhibitor of urokinase plasminogen activator (uPA) as a potential treatment for multiple sclerosis(IC50s of 237, 16...
|
T3359 |
Aprotinin
|
9087-70-1
|
98%
|
|
Aprotinin a broad-spectrum serine protease inhibitor, inhibiting the activity of a number of different esterases and proteases, including trypsin, chymotrypsin, ...
|
T3990 |
AA26-9
|
1312782-34-5
|
98%
|
|
AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.
|
T8602 |
2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE
|
13947-21-2
|
98%
|
|
2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).
|
T5597 |
ZT-12-037-01
|
2328073-61-4
|
98%
|
|
Zt-12-037-01 is a ATP competitive STK19 inhibitor(IC50 values of 23.96 nM and 27.94 nM for STK19 (WT) and STK19 (D89N),respectively).
|
T6564 |
Leupeptin Hemisulfate
|
103476-89-7
|
98%
|
|
Leupeptin hemisulfate is a reversible, competitive serine/cysteine protease inhibitor. It is an orally active, antioxidant and anti-inflammatory agent.
|
TN1372 |
Alpha-Amyrin
|
638-95-9
|
98%
|
|
Alpha-Amyrin is an inhibitor of trypsin and chymotrypsin with antineoplastic effects. alpha-Amyrin can be used in studies about acting as a hepatomodulatory.
|
T25549 |
JCP174
|
126062-19-9
|
98%
|
|
JCP174 is a depalmitoylase inhibitor that enhances Toxoplasma host-cell invasion by targeting TgPPT1.
|
T8802 |
2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
|
80499-32-7
|
98%
|
|
Trypsin inhibitor (human urine urinastatin protein moiety), as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urine or...
|
T12613L |
BAY-85-8501
|
1161921-82-9
|
98%
|
|
BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of 65 pM)
|
T6285 |
GSK-690693
|
937174-76-0
|
98%
|
|
GSK690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM, also sensitive to the AGC kinase family: PKA, PrkX and PKC isozymes. Phase 1.
|