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ATN-658

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Catalog No. T9901A-1238

ATN-658 is a humanized monoclonal antibody target the Domain 3 region of the urokinase-type plasminogen activator receptor, inhibition of cellular migration and invasion by disrupting the functional interaction between the receptor and various integrin signaling partners within designated preclinical oncology models.

ATN-658

ATN-658

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Catalog No. T9901A-1238
ATN-658 is a humanized monoclonal antibody target the Domain 3 region of the urokinase-type plasminogen activator receptor, inhibition of cellular migration and invasion by disrupting the functional interaction between the receptor and various integrin signaling partners within designated preclinical oncology models.
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Product Introduction

Bioactivity
Description
ATN-658 is a humanized monoclonal antibody target the Domain 3 region of the urokinase-type plasminogen activator receptor, inhibition of cellular migration and invasion by disrupting the functional interaction between the receptor and various integrin signaling partners within designated preclinical oncology models.
In vitro
In PC-3 prostate cancer cell assays, ATN-658 caused a significant dose-dependent decrease in cell motility without affecting doubling time [1].
In vivo
In intratibial PC-3 xenograft models, systemic administration of ATN-658 resulted in a significant decrease in tumor volume and skeletal lesions [1].
Reactivity
Human
Application
FACS
Functional assay
Antibody Type
Monoclonal
FormulationSupplied as a sterile solution in a buffered formulation system (e.g., phosphate-, citrate-, or amino acid-based). Please refer to the CoA for lot-specific composition.
Endotoxin<1.0 EU/mg
Related Conjugates and Formulations
Conjucates
Unconjugated
Antigen Details
Uniprot ID
TargetPLAUR/uPAR/CD87
Chemical Properties
Antibody Information
IsotypeIgG1
Storage & Solubility Information
Storagestore at low temperature | -20°C for 2 years, 4°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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