Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
Applied FilterClear all
TargetMol | Tags By Target
  • Histamine Receptor
    (121)
  • 5-HT Receptor
    (31)
  • Adrenergic Receptor
    (21)
  • Dopamine Receptor
    (21)
  • AChR
    (14)
  • Norepinephrine
    (11)
  • Apoptosis
    (6)
  • Antibacterial
    (4)
  • Autophagy
    (4)
  • Others
    (48)
Filter
Search Result
Results for "

h1 receptor

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    192
    TargetMol | Inhibitors_Agonists
  • Peptide Products
    1
    TargetMol | Peptide_Products
  • Natural Products
    6
    TargetMol | Natural_Products
  • Recombinant Protein
    5
    TargetMol | Recombinant_Protein
  • Isotope Products
    13
    TargetMol | Isotope_Products
  • Disease Modeling
    2
    TargetMol | Disease_Modeling_Products
DF-1111301
DF1111301, DF 1111301
T27159160665-99-6In house
DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.
  • Inquiry Price
6-8 weeks
Size
QTY
TargetMol
ReN-1869
ReN1869, ReN 1869, NNC05-1869, NNC-05-1869, NNC 05-1869
T28516170149-99-2In house
ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseases.
  • Inquiry Price
6-8 weeks
Size
QTY
vapitadine dihydrochloride
Vapitadine 2HCl, R-129160 dihydrochloride, R129160 dihydrochloride, R-129160 2HCl, R129160 2HCl, R 129160 2HCl
T29096279253-83-7In house
Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.
  • Inquiry Price
6-8weeks
Size
QTY
Dimethindene
Z-2001, Z2001, Z 2001, Dimetindeno, Dimetindene
T314885636-83-9In house
Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.
  • Inquiry Price
6-8 weeks
Size
QTY
TargetMol | Inhibitor Sale
Fenclozine Maleate
S 1429
T8397576823-82-0In house
Fenclozine Maleate (S 1429) is a potential histamine H1 receptor antagonist , which can be used to study fever, inflammation and pain.
  • Inquiry Price
Size
QTY
Chlorprothixene
Truxal, Taractan, Clorprotixeno
T0074113-59-7
Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.
  • Inquiry Price
Size
QTY
Paliperidone
9-hydroxyrisperidone
T0076144598-75-4
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the primary active metabolite of the older atypical antipsychotic risperidone.
  • Inquiry Price
Size
QTY
Diphenhydramine hydrochloride
DPH, Diphenhydramine HCl
T0330147-24-0
Diphenhydramine hydrochloride (DPH) is a histamine H1 antagonist used as an antitussive and antiemetic. It is also used for pruritus and dermatoses, for hypersensitivity reactions, as an antiparkinson, a hypnotic, and as an ingredient in common cold preparations.
  • Inquiry Price
Size
QTY
Trimipramine maleate
Surmontil maleate
T1045521-78-8
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Maleate is the maleate salt form of trimipramine, a tricyclic secondary amine of the dibenzazepine class, with an antidepressant property.
  • Inquiry Price
Size
QTY
Levocarnitine propionate hydrochloride
ST-261, Propionyl-L-carnitine hydrochloride, L-Propionylcarnitine chloride
T1182119793-66-7
Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, intermittent claudication, and other diseases.
  • Inquiry Price
Size
QTY
Orphenadrine hydrochloride
Mephenamin, Mebedrol
T1308341-69-5
Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.
  • Inquiry Price
Size
QTY
Sodium butanoate
Sodium Butyrate, Butanoic acid sodium salt
T1393156-54-7
Sodium butanoate (Sodium Butyrate) is the sodium salt of butyrate with potential antineoplastic activity. Butyrate, a short chain fatty acid, competitively binds to the zinc sites of class I and II histone deacetylases (HDACs).
  • Inquiry Price
Size
QTY
Diphenhydramine
Syntedril, PM-255, PM255, PM 255, Debendrin, Dabylen
T2141958-73-1
Diphenhydramine (Syntedril), a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the treatment of allergies. Diphenhydramine is also used in the management of drug-induced parkinsonism and other extrapyramidal symptoms.
  • Inquiry Price
Size
QTY
Desloratadine
Sch34117, NSC 675447
T2520100643-71-8
Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typical histaminergic effects on H1-receptors in bronchial smooth muscle, capillaries and gastrointestinal smooth muscle, including vasodilation, bronchoconstriction, increased vascular permeability, pain, itching and spasmodic contractions of gastrointestinal smooth muscle. Desloratadine is used to provide symptomatic relieve of allergic symptoms.
  • Inquiry Price
Size
QTY
Osthole
Ostol, Osthol, NSC 31868
T2848484-12-8
Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.
  • Inquiry Price
Size
QTY
Mebhydrolin
Mebhydroline
T7085524-81-2
Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.
  • Inquiry Price
Size
QTY
Escitalopram
Seroplex, S-(+)-Citalopram, (S)-Citalopram
T0185128196-01-0
Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing ethanol uptake in alcoholics and is used in depressed patients who also suffer from tardive dyskinesia in preference to tricyclic antidepressants, which aggravate this condition.
  • Inquiry Price
1-2 weeks
Size
QTY
Perphenazine
Trilafon, Perphenazin, Etaperazine
T109058-39-9
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
  • Inquiry Price
Size
QTY
Emedastine
LY188695, Emadine
T397987233-61-2
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blocks histamine by binding to H1 receptors, thus blocking its downstream activity. As a result this agent interferes with mediator release from mast cells either by inhibiting calcium ion influx across mast cell basophil plasma membrane or by inhibiting intracellular calcium ion release within the cells. In addition, emedastine may also inhibit the late-phase allergic reaction mediated through leukotrienes or prostaglandins, or by producing an anti-platelet activating factor effect. Upon ocular administration, emedastine causes a dose-dependent inhibition of histamine-stimulated vascular permeability in the conjunctiva. Emedastine does not affect adrenergic, dopamine, or serotonin receptors.
  • Inquiry Price
Size
QTY
Quetiapine
Quetiapin, ICI204636
T0162111974-69-7
Quetiapine (ICI204636) is used for the therapy of schizophrenia, and for the treatment of acute manic episodes associated with bipolar I disorder. The mechanism of quetiapine' action is thought by mediated through antagonist activity at serotonin and dopamine receptors. Specifically, the D1 and D2 dopamine, the α1 adrenoreceptor and α2 adrenoreceptor, and 5-HT1A and 5-HT2 serotonin receptor subtypes are antagonized. Quetiapine also can inhibit the histamine H1 receptor.
  • Inquiry Price
Size
QTY
Hydroxyzine
Hydroxyzine free base
T2088468-88-2
Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
  • Inquiry Price
Size
QTY
(s)-(+)-dimethindene maleate
T23297136152-65-3
(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that also inhibits muscarinic M1, M3, and M4 receptors.
  • Inquiry Price
7-10 days
Size
QTY
AVN-101
T266901061354-48-0
AVN-101 is a highly potent 5-HT7 receptor antagonist with a Ki value of 153 pM. AVN-101 also exhibits considerable affinity for histamine H1 (Ki value of 0.58 nM) and adrenergic α2A, α2B and α2C (Ki values ​​of 0.41-3.6 nM) receptors. AVN-101 has shown good oral bioavailability and brain-blood barrier permeability, low toxicity and reasonable efficacy in animal models of central nervous system diseases.
  • Inquiry Price
Size
QTY
Betahistine
Vasomotal, Serc base, PT 9 base
T41955638-76-6
Betahistine (Vasomotal) is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may exacerbate bronchial asthma and peptic ulcers. Betahistine dihydrochloride is an anti-vertigo drug. It is commonly prescribed for balance disorders or to alleviate vertigo symptoms associated with Ménière's disease.
  • Inquiry Price
Size
QTY