T10905 |
CXCR2-IN-1
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CXCR
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CXCR2-IN-1是可渗透中枢神经系统的 CXCR2拮抗剂,pIC50值为9.3。 |
T39078 |
CXCR7 antagonist-1
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CXCR7 antagonist-1 |
CXCR
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CXCR7 antagonist-1 是 SDF-1 趋化因子或 I-TAC 与趋化因子受体 CXCR7 结合的特异性拮抗剂。 CXCR7 antagonist-1 可防止肿瘤细胞增殖和肿瘤形成,可用于炎症性疾病的研究。 |
T39742 |
CXCR4 antagonist 2
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CXCR4 antagonist 2 is a CXCR4 antagonist with an IC 50 value of 47 nM. |
T36982 |
CXCR3 Antagonist 6c
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CXCR3 antagonist 6c is an antagonist of chemokine (C-X-C motif) receptor 3 (CXCR3).1It inhibits calcium mobilization ind... |
T10906 |
CXCR7 modulator 1
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Others
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CXCR7 modulator 1 is an effective and orally bioavailable peptoid hybrid CXCR7 modulator with Ki of 9 nM. |
T40786 |
CXCR4 antagonist 1
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CXCR4 antagonist 1 |
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CXCR4 antagonist 1 is a potent CXCR4 antagonist. CXCR4 antagonist 1 has anti- HIV activity. |
T10907 |
CXCR7 modulator 2
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Others
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CXCR7 modulator 2 is a 7-type C-X-C chemokine receptor (CXCR7) modulator with a Ki of 13 nM. |
T36923 |
CXCR2-IN-2
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CXCR2-IN-2 |
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CXCR2-IN-2 is a selective, brain penetrant, and orally bioavailable CXCR2 antagonist (IC50=5.2 nM/1 nM in β-arrestin ass... |
T36443 |
(R,R)-CXCR2-IN-2
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(R,R)-CXCR2-IN-2 |
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(R,R)-CXCR2-IN-2, diastereoisomer of CXCR2-IN-2 (compound 68), is a brain penetrant CXCR2 antagonist with a pIC50 of 9 a... |
T33763 |
NVP CXCR2 20
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NVP-CXCR2 20,NVP CXCR220,NVP CXCR2-20 |
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NVP CXCR2 20 is an effective selective CXCR2 antagonist (IC50 = 40 nM) with oral bioavailability. |
T61236 |
CXCR2 antagonist 7
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CXCR2 antagonist 7 (compound 19) 是一种有效的CXCR2拮抗剂。CXCR2 antagonist 7 显示出有效的CXCR2结合亲和力 (IC50=0.044 μM) 和钙动员 (IC50=0.66 μM)。 |
T63369 |
CXCR4 antagonist 4
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CXCR4 antagonist 4 是口服具有活力的、有效的CXCR4拮抗剂,IC50 值为 24 nM。CXCR4 antagonist 4能够抑制 CYP 2D6 的活性,增加 PAMPA 的通透性,有效阻碍人类免疫缺陷病毒的进入 (... |
T61356 |
CXCR2 antagonist 3
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CXCR2 antagonist 3 (compound 11h) is a highly effective antagonist of CXC chemokine receptor 2 (CXCR2). It displays pote... |
T60811 |
CXCR4 antagonist 7
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CXCR4 antagonist 7 (Compound PARA-B) 是可用于研究HIV 感染、炎症性疾病、癌症和 WHIM 综合症的CXCR4拮抗剂 (IC50 = 9.3 nM)。 |
T62352 |
CXCR4 modulator-2
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CXCR4 modulator-2 (compound Z7R) 是一种 CXCR4 的高效调节剂 (IC50: 1.25 nM)。CXCR4 modulator-2 在小鼠血清中表现出较好的稳定性 (t1/2= 77.1 min),在小鼠... |
T61363 |
CXCR4 antagonist 8
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CXCR4 antagonist 8 (Compound 3) is a potent inhibitor of CXCR4. It demonstrates an IC50 value of 57 nM in CXCR4 antagoni... |
T61420 |
CXCR4 antagonist 6
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CXCR4 antagonist 6 (compound 46) is a highly potent inhibitor of CXCR4 with an IC50 value of 79 nM. It effectively inhib... |
T61419 |
CXCR4 antagonist 5
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CXCR4 antagonist 5 (compound 23), a potent CXCR4 antagonist, exhibits high inhibition efficacy against CXCR4 with an IC5... |
T61650 |
CXCR4 antagonist 9
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CXCR4 antagonist 9 (Compound 2) is a potent CXCR4 antagonist displaying an IC50 of 15 nM. It effectively inhibits the cy... |
TMPY-06553 |
CXCR4/CD184 Protein, Human, Recombinant, VLP
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