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Sampatrilat is an effecive and orally active vasopeptidase inhibitor of ACE and neutral endopeptidase. Sampatrilat inhibits C-domain ACE (Ki=13.8 nM) 12.4-fold more potent than that for the N-domain (Ki=171.9 nM).

Acacetin (5,7-Dihydroxy-4'-methoxyflavone) is an O-methylated flavone found in various plants, exhibiting antinociceptive, anti-inflammatory, and antioxidant activities in different research models.

Acacetin-7-glucuronide is a glucuronic acid glycoside that can be isolated from the methanol leaf extract of the purple bead. It may be used in the development of nutritional health products and pharmaceutical preparations.

Acacetin 7-O-β-sophoroside, a flavonoid glycoside, has been isolated from the rhizomes and roots of valerian (Valeriana officinalis) [1].

Acacetin 7-O-β-D-xylopyranosyl-(1→2)[α-L-rhamnopyranosyl-(1→6)]-β-D-glucopyranoside (Compound 10), a flavone glycoside, is extractable from Robinia pseudoacacia leaf preparations [1].

Acacetin 7-O-β-D-glucuronopyranosyl-(1→2)[α-L-rhamnopyranosyl-(1→6)]-β-D-glucopyranoside, also known as compound 8, is a flavonoid glycoside isolated from the leaf extract of the black locust (Leguminosae) [1].

Acacetin 7-O-(6″-O-α-L-rhamnopyranosyl-β-sophoroside), a flavonoid glycoside, has been isolated from Valeriana jatamansi Jones [1].

Acacetin 7-O-(6-O-malonylglucoside) is a reversible inhibitor of hMAO-A and hMAO-B (IC₅₀ = 2.34 and 1.87 μM), respectively, and can be used in the study of neurodegenerative diseases.

Acacetin (Standard) is a reference standard for research and analysis in studies involving Acacetin. Acacetin (5,7-Dihydroxy-4'-methoxyflavone) is an O-methylated flavone found in various plants, shows antinociceptive, anti-inflammatory, and antioxidant activity in various research models.

Norplicacetin exhibits activity against Gram-positive bacteria and mycobacteria.

Plicacetin is a crystalline antibiotic that can be isolated from the fermentation broth of actinobacteria (Streptomyces), and it has a structure similar to Amicetin and Bamicetin.

Acacetin-7-O-beta-D-galactopyranoside is a natural product found in Chrysanthemum indicum.

Acacetin 7-[rhamnosyl-(1->2)-galacturonide] is a natural product that can be used as a reference standard. The CAS number of Acacetin 7-[rhamnosyl-(1->2)-galacturonide] is 38722-95-1.

Acacetin-7-O-(3-O-malonyl)-β-D-glucopyranoside (compound 13) is a compound extractable from the plant D. foetidum.

Clozapine N-oxide is the major metabolite of Clozapine and is blood-brain barrier permeable. Clozapine N-oxide is an agonist of DREADDs and activates the DREADD receptors hM3Dq and hM4Di. Clozapine N-oxide is also a dopamine antagonist and selective muscarinic M4 receptor agonist.

Adiphenine hydrochloride (Patrovina), a nicotinic receptor inhibitor, can be used as an antispasmodic drug.

Galanthamine hydrobromide (Galantamine hydrobromide), a long-acting and centrally active AChE inhibitor (IC50:410 nM), is an allosteric potentiator at neuronal nicotinic ACh receptors.

Ipratropium bromide monohydrate (Ipratropium bromide hydrate) is a muscarinic antagonist structurally related to ATROPINE but often considered safer and more effective for inhalation use. It is used for various bronchial disorders, in rhinitis, and as an antiarrhythmic.

Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.

Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 MUSCARINIC ANTAGONIST. It is used as a UROLOGIC AGENT in the treatment of URINARY INCONTINENCE.

Pancuronium dibromide (Pavulon), a competitive AChR antagonist (IC50 = 5.5 nM), acts as a skeletal muscle relaxant. Pancuronium dibromide(Pancuronium bromide) blocking neuromuscular transmission is achieved by competing with acetylcholine for receptor sites on the motor end-plate.

Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.

Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.

Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.