Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.

Cat. No.	Product name	CAS No.	Purity
T29663	ADL-5747	850176-30-6	98%
T29663	ADL-5747 (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletal disorders, and may be used in t...
T28453L	Propiram fumarate HCl	945013-73-0	98%
T28453L	Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
T10593	BPR1M97	2059904-66-2	98%
T10593	BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.8...
T39988	6'-GNTI dihydrochloride	2410327-94-3	98%
T39988	6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of β-aspirin 2. 6'-GNTI dihy...
T27667	JNJ-20788560	825649-28-3	98%
T27667	JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).
T12320	ORL1 antagonist 1	1174985-59-1	98%
T12320	ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).
T37610	AT-121	2099681-31-7	98%
T37610	AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively). It stimulates [35S]GTPγS binding to cell membranes exp...
T20166L	Deltorphin acetate		98%
T20166L	Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid receptor...
TP1793	Nociceptin (1-13), amide	178064-02-3	98%
TP1793	Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain memb...
T7567	Adrenorphin	88377-68-8	98%
T7567	Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
T7576	β-Casomorphin, bovine	72122-62-4	98%
T7576	β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
T4633	Asimadoline	153205-46-0	98%
T4633	Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
T7404	Dermorphin	77614-16-5	98%
T7404	Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
T11479	GSK1521498	1426543-84-1	98%
T11479	GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive consumption of food, alcohol, ...
T12168	Naloxone benzoylhydrazone	119630-94-3	98%
T12168	Naloxone benzoylhydrazone is a prototypic κ3-opioid receptor agonist, and a partial agonist at the cloned μ and δ opioid receptors, and an antagonist at opioid-l...
T11478	GSK1521498 free base (hydrochloride)	1007578-24-6	98%
T11478	GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive cons...
T13419	ROCK-IN-1	934387-35-6	98%
T13419	ROCK-IN-1 is a potent ROCK inhibitor(IC50 of 1.2 nM , ROCK2).
TP1367L	[D-Ala2]leucine-enkephalin acetate	TP1367L	98%
TP1367L	[D-Ala2]Leucine enkephalin acetate is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.
TN5017	Sideritoflavone	70360-12-2	98%
TN5017	Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
TP2036	DPDPE	88373-73-3	98%
TP2036	DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...