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Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.
Cat. No. Product name CAS No. Purity Chemical Structure
T11198 Endomorphin 2 TFA 1276124-00-5 98%
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the...
T12241 Norbinaltorphimine dihydrochloride 113158-34-2 98%
Norbinaltorphimine dihydrochloride is a potent and selective antagonist of κ opioid receptor.
T11478L GSK1521498 free base 1007573-18-3 98%
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor. GSK1521498 free base also has the potential for disorders of compulsive consu...
T7404 Dermorphin 77614-16-5 98%
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
T15165 DPI-3290 182417-73-8 98%
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent antinocicepti...
T12314 Opioid receptor modulator 1 77514-44-4 98%
Opioid receptor modulator 1 is a modulator of opioid receptor.
T13438 (R,S)-Ivosidenib 2070009-31-1 98%
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
T7173 [Leu5]-Enkephalin 58822-25-6 98%
[Leu5]-Enkephalin is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and µ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively)
TN3367 Akuammidine 639-36-1 98%
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki va...
T4633 Asimadoline 153205-46-0 98%
Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
TP1793 Nociceptin (1-13), amide 178064-02-3 98%
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain memb...
T7306 Valorphin 144313-54-2 98%
Valorphin has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
T7576 β-Casomorphin, bovine 72122-62-4 98%
β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
TN3368 Akuammigine 642-17-1 98%
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
TP2036 DPDPE 88373-73-3 98%
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
T7567 Adrenorphin 88377-68-8 98%
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
TN5017 Sideritoflavone 70360-12-2 98%
Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
TP1367L [D-Ala2]leucine-enkephalin acetate TP1367L 98%
[D-Ala2]Leucine enkephalin acetate is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.
T13419 ROCK-IN-1 934387-35-6 98%
ROCK-IN-1 is a potent ROCK inhibitor(IC50 of 1.2 nM , ROCK2).
T11478 GSK1521498 free base (hydrochloride) 1007578-24-6 98%
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive cons...
Endomorphin 2 TFA
T11198
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the...
Norbinaltorphimine dihydrochloride
T12241
Norbinaltorphimine dihydrochloride is a potent and selective antagonist of κ opioid receptor.
GSK1521498 free base
T11478L
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor. GSK1521498 free base also has the potential for disorders of compulsive consu...
Dermorphin
T7404
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
DPI-3290
T15165
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent antinocicepti...
Opioid receptor modulator 1
T12314
Opioid receptor modulator 1 is a modulator of opioid receptor.
(R,S)-Ivosidenib
T13438
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
[Leu5]-Enkephalin
T7173
[Leu5]-Enkephalin is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and µ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively)
Akuammidine
TN3367
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki va...
Asimadoline
T4633
Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
Nociceptin (1-13), amide
TP1793
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain memb...
Valorphin
T7306
Valorphin has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
β-Casomorphin, bovine
T7576
β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
Akuammigine
TN3368
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
DPDPE
TP2036
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
Adrenorphin
T7567
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
Sideritoflavone
TN5017
Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
[D-Ala2]leucine-enkephalin acetate
TP1367L
[D-Ala2]Leucine enkephalin acetate is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.
ROCK-IN-1
T13419
ROCK-IN-1 is a potent ROCK inhibitor(IC50 of 1.2 nM , ROCK2).
GSK1521498 free base (hydrochloride)
T11478
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive cons...
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