T29663 |
ADL-5747
|
850176-30-6
|
98%
|
|
ADL-5747 (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletal disorders, and may be used in t...
|
T28453L |
Propiram fumarate HCl
|
945013-73-0
|
98%
|
|
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
|
T10593 |
BPR1M97
|
2059904-66-2
|
98%
|
|
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.8...
|
T39988 |
6'-GNTI dihydrochloride
|
2410327-94-3
|
98%
|
|
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of β-aspirin 2. 6'-GNTI dihy...
|
T27667 |
JNJ-20788560
|
825649-28-3
|
98%
|
|
JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).
|
T12320 |
ORL1 antagonist 1
|
1174985-59-1
|
98%
|
|
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).
|
T37610 |
AT-121
|
2099681-31-7
|
98%
|
|
AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively). It stimulates [35S]GTPγS binding to cell membranes exp...
|
T20166L |
Deltorphin acetate
|
|
98%
|
|
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid receptor...
|
TP1793 |
Nociceptin (1-13), amide
|
178064-02-3
|
98%
|
|
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain memb...
|
T7567 |
Adrenorphin
|
88377-68-8
|
98%
|
|
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
|
T7576 |
β-Casomorphin, bovine
|
72122-62-4
|
98%
|
|
β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
|
T4633 |
Asimadoline
|
153205-46-0
|
98%
|
|
Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
|
T7404 |
Dermorphin
|
77614-16-5
|
98%
|
|
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
|
T11479 |
GSK1521498
|
1426543-84-1
|
98%
|
|
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive consumption of food, alcohol, ...
|
T12168 |
Naloxone benzoylhydrazone
|
119630-94-3
|
98%
|
|
Naloxone benzoylhydrazone is a prototypic κ3-opioid receptor agonist, and a partial agonist at the cloned μ and δ opioid receptors, and an antagonist at opioid-l...
|
T11478 |
GSK1521498 free base (hydrochloride)
|
1007578-24-6
|
98%
|
|
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive cons...
|
T13419 |
ROCK-IN-1
|
934387-35-6
|
98%
|
|
ROCK-IN-1 is a potent ROCK inhibitor(IC50 of 1.2 nM , ROCK2).
|
TP1367L |
[D-Ala2]leucine-enkephalin acetate
|
TP1367L
|
98%
|
|
[D-Ala2]Leucine enkephalin acetate is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.
|
TN5017 |
Sideritoflavone
|
70360-12-2
|
98%
|
|
Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
|
TP2036 |
DPDPE
|
88373-73-3
|
98%
|
|
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
|