T11198 |
Endomorphin 2 TFA
|
1276124-00-5
|
98%
|
|
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the...
|
T12241 |
Norbinaltorphimine dihydrochloride
|
113158-34-2
|
98%
|
|
Norbinaltorphimine dihydrochloride is a potent and selective antagonist of κ opioid receptor.
|
T11478L |
GSK1521498 free base
|
1007573-18-3
|
98%
|
|
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor. GSK1521498 free base also has the potential for disorders of compulsive consu...
|
T7404 |
Dermorphin
|
77614-16-5
|
98%
|
|
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
|
T15165 |
DPI-3290
|
182417-73-8
|
98%
|
|
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent antinocicepti...
|
T12314 |
Opioid receptor modulator 1
|
77514-44-4
|
98%
|
|
Opioid receptor modulator 1 is a modulator of opioid receptor.
|
T13438 |
(R,S)-Ivosidenib
|
2070009-31-1
|
98%
|
|
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
|
T7173 |
[Leu5]-Enkephalin
|
58822-25-6
|
98%
|
|
[Leu5]-Enkephalin is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and µ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively)
|
TN3367 |
Akuammidine
|
639-36-1
|
98%
|
|
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki va...
|
T4633 |
Asimadoline
|
153205-46-0
|
98%
|
|
Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
|
TP1793 |
Nociceptin (1-13), amide
|
178064-02-3
|
98%
|
|
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain memb...
|
T7306 |
Valorphin
|
144313-54-2
|
98%
|
|
Valorphin has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
|
T7576 |
β-Casomorphin, bovine
|
72122-62-4
|
98%
|
|
β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
|
TN3368 |
Akuammigine
|
642-17-1
|
98%
|
|
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
|
TP2036 |
DPDPE
|
88373-73-3
|
98%
|
|
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
|
T7567 |
Adrenorphin
|
88377-68-8
|
98%
|
|
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
|
TN5017 |
Sideritoflavone
|
70360-12-2
|
98%
|
|
Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
|
TP1367L |
[D-Ala2]leucine-enkephalin acetate
|
TP1367L
|
98%
|
|
[D-Ala2]Leucine enkephalin acetate is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.
|
T13419 |
ROCK-IN-1
|
934387-35-6
|
98%
|
|
ROCK-IN-1 is a potent ROCK inhibitor(IC50 of 1.2 nM , ROCK2).
|
T11478 |
GSK1521498 free base (hydrochloride)
|
1007578-24-6
|
98%
|
|
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive cons...
|