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Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.
Cat. No. Product name CAS No. Purity Chemical Structure
T29663 ADL-5747 850176-30-6 98%
ADL-5747 (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletal disorders, and may be used in t...
T28453L Propiram fumarate HCl 945013-73-0 98%
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
T10593 BPR1M97 2059904-66-2 98%
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.8...
T39988 6'-GNTI dihydrochloride 2410327-94-3 98%
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of β-aspirin 2. 6'-GNTI dihy...
T27667 JNJ-20788560 825649-28-3 98%
JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).
T12320 ORL1 antagonist 1 1174985-59-1 98%
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).
T37610 AT-121 2099681-31-7 98%
AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively). It stimulates [35S]GTPγS binding to cell membranes exp...
T20166L Deltorphin acetate 98%
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid receptor...
TP1793 Nociceptin (1-13), amide 178064-02-3 98%
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain memb...
T7567 Adrenorphin 88377-68-8 98%
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
T7576 β-Casomorphin, bovine 72122-62-4 98%
β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
T4633 Asimadoline 153205-46-0 98%
Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
T7404 Dermorphin 77614-16-5 98%
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
T11479 GSK1521498 1426543-84-1 98%
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive consumption of food, alcohol, ...
T12168 Naloxone benzoylhydrazone 119630-94-3 98%
Naloxone benzoylhydrazone is a prototypic κ3-opioid receptor agonist, and a partial agonist at the cloned μ and δ opioid receptors, and an antagonist at opioid-l...
T11478 GSK1521498 free base (hydrochloride) 1007578-24-6 98%
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive cons...
T13419 ROCK-IN-1 934387-35-6 98%
ROCK-IN-1 is a potent ROCK inhibitor(IC50 of 1.2 nM , ROCK2).
TP1367L [D-Ala2]leucine-enkephalin acetate TP1367L 98%
[D-Ala2]Leucine enkephalin acetate is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.
TN5017 Sideritoflavone 70360-12-2 98%
Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
TP2036 DPDPE 88373-73-3 98%
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
ADL-5747
T29663
ADL-5747 (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletal disorders, and may be used in t...
Propiram fumarate HCl
T28453L
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
BPR1M97
T10593
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.8...
6'-GNTI dihydrochloride
T39988
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of β-aspirin 2. 6'-GNTI dihy...
JNJ-20788560
T27667
JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).
ORL1 antagonist 1
T12320
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).
AT-121
T37610
AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively). It stimulates [35S]GTPγS binding to cell membranes exp...
Deltorphin acetate
T20166L
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid receptor...
Nociceptin (1-13), amide
TP1793
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain memb...
Adrenorphin
T7567
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
β-Casomorphin, bovine
T7576
β-Casomorphin, bovine(2TFA) is an opioid peptide isolated from casein peptone
Asimadoline
T4633
Asimadoline is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally developed to treat...
Dermorphin
T7404
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
GSK1521498
T11479
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive consumption of food, alcohol, ...
Naloxone benzoylhydrazone
T12168
Naloxone benzoylhydrazone is a prototypic κ3-opioid receptor agonist, and a partial agonist at the cloned μ and δ opioid receptors, and an antagonist at opioid-l...
GSK1521498 free base (hydrochloride)
T11478
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive cons...
ROCK-IN-1
T13419
ROCK-IN-1 is a potent ROCK inhibitor(IC50 of 1.2 nM , ROCK2).
[D-Ala2]leucine-enkephalin acetate
TP1367L
[D-Ala2]Leucine enkephalin acetate is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.
Sideritoflavone
TN5017
Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
DPDPE
TP2036
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
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