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6β-Naltrexol
🥰Excellent
Catalog No. T85517Cas No. 49625-89-0
Alias 6β-Hydroxynaltrexone
6β-Naltrexol functions as a potent and peripherally selective opioid receptor antagonist. Unlike central-acting opioid antagonists, 6β-Naltrexol is restricted primarily to peripheral tissues, which allows it to counteract opioid-mediated side effects such as opioid-induced constipation while minimizing central nervous system interactions. 6β-Naltrexol is therefore relevant in reseaches in peripheral opioid effects.
6β-Naltrexol
🥰Excellent
Purity: 99.933%
Catalog No. T85517Alias 6β-HydroxynaltrexoneCas No. 49625-89-0
6β-Naltrexol functions as a potent and peripherally selective opioid receptor antagonist. Unlike central-acting opioid antagonists, 6β-Naltrexol is restricted primarily to peripheral tissues, which allows it to counteract opioid-mediated side effects such as opioid-induced constipation while minimizing central nervous system interactions. 6β-Naltrexol is therefore relevant in reseaches in peripheral opioid effects.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $83 | - | In Stock | |
| 5 mg | $290 | - | In Stock | |
| 10 mg | $464 | - | In Stock | |
| 25 mg | $789 | - | In Stock | |
| 50 mg | $1,180 | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.933%
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Product Introduction
Bioactivity
Chemical Properties
| Description | 6β-Naltrexol functions as a potent and peripherally selective opioid receptor antagonist. Unlike central-acting opioid antagonists, 6β-Naltrexol is restricted primarily to peripheral tissues, which allows it to counteract opioid-mediated side effects such as opioid-induced constipation while minimizing central nervous system interactions. 6β-Naltrexol is therefore relevant in reseaches in peripheral opioid effects. |
| Targets&IC50 | CHO cells:1.2 nM (EC50) |
| Synonyms | 6β-Hydroxynaltrexone |
| Molecular Weight | 343.42 |
| Formula | C20H25NO4 |
| Cas No. | 49625-89-0 |
| Smiles | O[C@]12[C@@]34C=5C(O[C@]3([C@H](O)CC1)[H])=C(O)C=CC5C[C@]2(N(CC6CC6)CC4)[H] |
| Color | White |
| Appearance | Solid |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 80 mg/mL (232.95 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
Dose Conversion
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Tech Support
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