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Nalmefene hydrochloride

Name: Nalmefene hydrochloride
Brand: TargetMol
SKU: T6221
Rating: 4.5 (1 reviews)

😃Good

Catalog No. T6221Cas No. 58895-64-0

Alias Nalmefene HCl

Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.

Nalmefene hydrochloride

😃Good

Purity: 99.85%

Catalog No. T6221Alias Nalmefene HClCas No. 58895-64-0

Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.

Pack Size	Price	USA Warehouse	Global Warehouse
2 mg	$50	Backorder	Backorder
5 mg	$68	Backorder	Backorder
10 mg	$99	Backorder	Backorder
25 mg	$194	Backorder	Backorder
50 mg	$334	Backorder	Backorder
100 mg	$603	Backorder	Backorder

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.85%

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COA

Product Introduction

Bioactivity

Description	Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.
Synonyms	Nalmefene HCl

Chemical Properties

Molecular Weight	375.89
Formula	C₂₁H₂₆ClNO₃
Cas No.	58895-64-0
Smiles	C1(CC1)CN1[C@@H]2Cc3c4c(O[C@@H]5[C@]4([C@]2(CCC5=C)O)CC1)c(cc3)O.Cl
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: >10 mM, Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.6604 mL	13.3018 mL	26.6035 mL	133.0176 mL
5 mM	0.5321 mL	2.6604 mL	5.3207 mL	26.6035 mL
10 mM	0.2660 mL	1.3302 mL	2.6604 mL	13.3018 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc