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GR 89696 fumarate

Name: GR 89696 fumarate
Brand: TargetMol
SKU: T22810
Price: 58 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T22810Cas No. 126766-32-3

GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.

GR 89696 fumarate

🥰Excellent

Purity: 99.84%

Catalog No. T22810Cas No. 126766-32-3

GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.

Pack Size	Price	Availability
5 mg	$58	In Stock
10 mg	$97	In Stock
25 mg	$165	In Stock
50 mg	$238	In Stock
100 mg	$352	In Stock
1 mL x 10 mM (in DMSO)	$71	In Stock

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Batch Information

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Purity:99.84%

Resource Download

COA HNMR HPLC LCMS

Product Introduction

Bioactivity

Description

GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.

Chemical Properties

Molecular Weight	530.4
Formula	C₂₃H₂₉Cl₂N₃O₇
Cas No.	126766-32-3
Smiles	C(=C/C(O)=O)\C(O)=O.C(CC1=CC(Cl)=C(Cl)C=C1)(=O)N2C(CN3CCCC3)CN(C(OC)=O)CC2
Relative Density.	no data available
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

Ethanol: 3.6 mg/mL (6.79 mM), Sonication is recommended.

DMSO: 45 mg/mL (84.84 mM), Sonication is recommended.

H2O: 7.7 mg/mL (14.52 mM), Sonication is recommended.

Solution Preparation Table

Ethanol/H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	1.8854 mL	9.4268 mL	18.8537 mL	94.2685 mL
5 mM	0.3771 mL	1.8854 mL	3.7707 mL	18.8537 mL

H2O/DMSO

	1mg	5mg	10mg	50mg
10 mM	0.1885 mL	0.9427 mL	1.8854 mL	9.4268 mL

DMSO

	1mg	5mg	10mg	50mg
20 mM	0.0943 mL	0.4713 mL	0.9427 mL	4.7134 mL
50 mM	0.0377 mL	0.1885 mL	0.3771 mL	1.8854 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc