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CP-866087 (Synonyms: UNII-MDH21334PI, CP866087, CP-866,087, CP 866087)
Catalog No. T31081 Copy Product Info
Purity: 99.56%
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CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.
CP-866087
Copy Product Info😃Good
Catalog No. T31081
Synonyms UNII-MDH21334PI, CP866087, CP-866,087, CP 866087
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.
Cas No. 519052-04-1
| Pack Size | Price | USA Stock | Global Stock | Quantity |
|---|---|---|---|---|
| 1 mg | $762 | In Stock | In Stock | |
| 5 mg | $1,590 | In Stock | In Stock | |
| 25 mg | $2,130 | In Stock | In Stock | |
| 50 mg | $2,580 | In Stock | In Stock |
For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)
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For research use only—not for human use. No sales to individuals. Use as intended only.
Batch Information
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Purity:99.56%
ee:100%
Appearance:Solid
Color:White to Yellow
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Product Introduction
CP-866087 AI Summary
CP-866087 exhibits significant bioactivity related to opioid receptors, showing high affinity as an antagonist at the human mu opioid receptor (Ki = 0.16 nM). It also binds to the human delta opioid receptor (Ki = 108.0 nM) and human kappa opioid receptor (Ki = 60.0 nM), demonstrating higher selectivity towards the mu receptor over delta (selectivity ratio = 31.0) and kappa (selectivity ratio = 17.0) receptors. Additionally, the compound inhibits the human ERG channel (IC50 = 2200.0 nM) and CYP2D6 enzyme activity (17% inhibition). It exhibits an efflux ratio that suggests potential interactions with the human MDR1 transporter. Metabolically, CP-866087 has an intrinsic clearance rate in human liver microsomes of 11.0 mL.min-1.kg-1..
Note: Summary generated by AI. Data source: ChEMBL 
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction. |
| Synonyms | UNII-MDH21334PI, CP866087, CP-866,087, CP 866087 |
| Molecular Weight | 376.49 |
| Formula | C24H28N2O2 |
| Cas No. | 519052-04-1 |
| Smiles | C(C)[C@]1([C@@]2([C@]1(CN(CC3(O)CC=4C(C3)=CC=CC4)C2)[H])[H])C5=CC(C(N)=O)=CC=C5 |
| Relative Density. | no data available |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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