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Lomefloxacin hydrochloride (Okacyn) inhibits DNA gyrase, a type II topoisomerase involved in the induction or relaxation of supercoiling during DNA replication. This inhibition leads to a decrease in DNA synthesis during bacterial replication, resulting in cell growth inhibition and eventually cell lysis. Lomefloxacin Hydrochloride is the hydrochloride salt form of lomefloxacin, a synthetic broad-spectrum fluoroquinolone with antibacterial activity.

Lomefloxacin (SC47111A) is a synthetic broad-spectrum fluoroquinolone with antibacterial activity.

Dolutegravir intermediate-1 (1-(2,2-dimethoxyethyl)-5-methoxy-6-(methoxycarbonyl)-4-oxo-1,4-dihydropyridine-3-carboxylic acid) is a new synthetic Dolutegravir intermediate. Dolutegravir is an integrase inhibitor developed for the treatment of human immunodeficiency virus (HIV)-1 infection.

Sitagliptin Intermediate 2 is a useful organic compound that has been used in life science related research.

cholesterol-absorption inhibitor Intermediate 2 is a potent and orally active cholesterol absorption inhibitor that reduces blood cholesterol levels.

Ketoconazole Intermediate 1e ((cis-2-((1H-Imidazol-1-yl)methyl)-2-(2,4-dichlorophenyl)-1,3-dioxolan-4-yl)methyl 4- methylbenzenesulfonate) is a ketoconazole intermediate.

Nivocasan Intermediate is an intermediate of Nivocasan. Nivocasan (GS-9450) is a pan-caspase inhibitor used in the study of HCV infection and non-alcoholic steatohepatitis.

Type III-Intermediate 8 is a useful organic compound for research related to life sciences and the catalog number is T9562.

Type III-Intermediate7 is a useful organic compound for research related to life sciences and the catalog number is T9563.

Intermediate of Pregabalin.

CRAC intermediate 1 is a key intermediate used in the synthesis of the CRAC ion channel series of compounds, details from patent WO 2010122089.

CRAC intermediate 2 is used as an intermediate compound in the synthesis of CRAC inhibitors.

Dacomitinib Intermediate 2 (N-(3-Chloro-4-fluorophenyl)-7-methoxy-6-nitroquinazolin-4-amine) has anticancer activity and can be used to study lung cancer.

LX-4211 intermediate is a synthetic intermediate of LX-4211, a potent SGLT1/2 inhibitor used as an antidiabetic agent.

PDE4 inhibitor intermediate 1 is a PDE4 inhibitor synthesis intermediate.

P62-mediated mitophagy inducer (PMI) is a regulator of mitophagy.

Doxapram intermediate-1 (Compound II) is a pyrrolidone derivative that significantly stimulates the central nervous system (CXS) and respiratory system in dogs, usually accompanied by varying degrees of blood pressure activity.

Exatecanintermediate 8 serves as an intermediate in the synthesis of Exatecan. Exatecan (DX-8951) is a commonly used cytotoxin component in ADC (Antibody-Drug Conjugate) preparation, and it functions as an inhibitor of DNA topoisomerase I (IC50=2.2 μM).

Tubulysin Aintermediate-1 is an intermediate in the synthesis of the cytotoxic peptide Tubulysin A. Tubulysin A (TubA) acts as an antibiotic (antibiotic), anti-microtubule toxins (anti-microtubule toxins), and apoptosis (apoptosis) inducer, which can be isolated from myxobacteria. It exhibits anti-angiogenic, anti-microtubule, anti-mitotic, and anti-proliferative properties, effectively blocking cells in the G2/M phase, inhibiting tubulin polymerization, and inducing depolymerization of isolated microtubules. Tubulysin A serves as an ADC Cytotoxin (ADC Cytotoxin) in the synthesis of ADCs.

The compound '(6R)-Taltobulin intermediate-9' serves as an intermediate in the synthesis of Taltobulin. Taltobulin is a common cytotoxic component (ADC Cytotoxin) in the preparation of antibody-drug conjugates (ADCs) and acts as a potent inhibitor of microtubule/tubulin. It disrupts tubulin polymerization, induces mitotic arrest, and triggers apoptosis (apoptosis).

Taltobulinintermediate-6 serves as an intermediate in the synthesis of Taltobulin. Taltobulin is a common cytotoxic component in the preparation of antibody-drug conjugates (ADC Cytotoxin) and acts as a potent inhibitor of microtubules/tubulin (Microtubule/Tubulin). It disrupts microtubule polymerization, induces mitotic arrest, and triggers apoptosis (apoptosis).

Taltobulinintermediate-7 is an intermediate in the synthesis of Taltobulin. Taltobulin is a commonly used toxin component in ADC preparation (ADC Cytotoxin) and serves as a potent inhibitor of microtubule/tubulin. It disrupts microtubule polymerization, induces mitotic arrest, and triggers apoptosis [apoptosis].

Exatecanintermediate 10 serves as an intermediate in synthesizing Exatecan. Exatecan (DX-8951) is a DNA topoisomerase I inhibitor with an IC50 value of 2.2 μM (0.975 μg/mL), utilized for cancer research.

(4R,5S)-MonomethylauristatinE intermediate-6 is an intermediate reactant in the synthesis of MonomethylauristatinE. MonomethylauristatinE (MMAE) is a microtubule/tubulin inhibitor with anticancer activity and is widely utilized as the cytotoxic component in antibody-drug conjugates (ADC Cytotoxin).