Home Tools
Log in
Products Inhibitors Libraries Kits Services Contact Us
Cart
Peptides Monoclonal Antibodies Dye Reagents PROTAC Virtual Screening Targetmol Kits Cell Counting Kit-8 (CCK-8) Inhibitor Cocktails Natural Products Phenols Alkaloids Flavonoids
Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling
MAPK Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination Others
Compound Libraries Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD Drug-like Compound Libraries Fragment Libraries Custom Compound Library
Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library

Search Result

Search Results for "insulin receptor"

Compounds

Cat No. Product Name
TMPY-04395 Insulin Receptor Protein, Human, Recombinant (His & GST Tag)
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to t...
TMPY-01149 Insulin Receptor Protein, Human, Recombinant (ECD, short isoform, His Tag)
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to t...
TMPY-05283 Insulin Receptor Protein, Human, Recombinant (long isoform, His Tag), Biotinylated
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to t...
TMPY-01146 Insulin Receptor Protein, Human, Recombinant (ECD, long isoform, His Tag)
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to t...
TP1259 [pTyr1146][pTyr1150][pTyr1151]Insulin Receptor (1142-1153) [pTyr1146][pTyr1150][pTyr1151]Insulin Receptor 1142-1153,Insulin Receptor 1142-1153
[pTyr1146][pTyr1150][pTyr1151]Insulin Receptor (1142-1153) functions as a substrate for insulin receptor tyrosine kinase...
T2349 BMS-754807 IGF-1R , Trk receptor , c-Met/HGFR
BMS754807 是一种可逆的IGF-1R 抑制剂 (IC50:1.8 nM，Ki<2 nM)，也是一种可逆的IR 抑制剂 (IC50:7 nM，Ki<2 nM)。它也抑制 Met (IC50:6 nM)，RON (IC50:44 nM)...
T21761 HNMPA IGF-1R
HNMPA 是膜不可渗透的胰岛素受体酪氨酸激酶 (insulin receptor tyrosine kinase) 抑制剂。HNMPA 可以抑制人胰岛素受体的酪氨酸和丝氨酸自磷酸化。HNMPA 对环 AMP 依赖性蛋白激酶或蛋白激酶 C ...
T8773 MID-1 IGF-1R , Others
MID-1 是 MG53-IRS-1 相互作用的抑制剂，能够破坏 MG53 与 IRS-1 的分子缔合，并消除 MG53 诱导的 IRS-1 泛素化和骨骼肌降解，升高 IRS-1 表达水平，增加胰岛素信号传导和葡萄糖摄取。
T8221 Insulin (human) Insulin(human),INSULIN,甘精胰岛素,胰岛素 IGF-1R
Insulin 是一种能够调节血液中的葡萄糖水平的多肽激素。
T6017 Linsitinib 林西替尼,OSI-906 IGF-1R
Linsitinib 是选择性的、有效的、具有口服活性的IGF-1和胰岛素受体(IR)的双重抑制剂，IC50分别为 35 和 75 nM。
TP1125 Insulin(cattle) Insulin from bovine pancreas,牛胰岛素,胰岛素 IGF-1R
Insulin cattle 是一种在胰腺 β 细胞中产生的两链多肽激素，在很多哺乳动物细胞培养体系中用作生长因子。
T9609 GRK5-IN-2 GRK
GRK5-IN-2 是基于吡啶的双环化合物，抑制 G 蛋白偶联受体激酶 5 。它调节胰岛素的表达和/或释放，在代谢疾病中有研究价值。
T8348 Phentolamine Adrenergic Receptor
Phentolamine 是一种 alpha-1 和 alpha-2 选择性肾上腺素能受体拮抗剂。
T22967 MEDICA16 MEDICA 16 GPR , ATP Citrate Lyase , Others
MEDICA16 是 GPR40 的特异性激动剂以及 GPR120 的部分激动剂。 MEDICA16 是一种 ATP-柠檬酸裂解酶抑制剂，可显着降低腓肠肌中的细胞内 TG 含量，同时增加胰岛素敏感性。
T9030 SU4984 FGFR , IGF-1R , PDGFR
SU4984 是蛋白质酪氨酸激酶抑制剂，能够抑制成纤维细胞生长因子受体 1 (FGFR1) (IC50:10-20 μM)，还能够抑制血小板衍生的生长因子受体和胰岛素受体的活性。它可用于研究癌症。
T6080 NVP-AEW541 AEW541 Tyrosine Kinases , FLT , IGF-1R , Autophagy
NVP-AEW541 是一种IGF-1R 抑制剂，IC50为 0.15 μM。它也抑制InsR，IC50为 0.14 μM。
T6419 BMS-536924 胰岛素样生长因子-1 受体拮抗剂,HY-10262,BMS 536924,CS-0117 MEK , FAK , Apoptosis , IGF-1R , Src
BMS-536924 是一种具有口服活性，竞争性和选择性的胰岛素样生长因子受体激酶和胰岛素受体抑制剂，IC50分别为 100 nM 和 73 nM。它具有抗癌活性。
T3079 GSK1838705A S6 Kinase , IGF-1R , JNK , ALK
GSK1838705A 是一种高效的、可逆的IGF-IR (IC50:2.0 nM) 和胰岛素受体 (IC50:1.6 nM)抑制剂，也可抑制ALK (IC50:0.5 nM)。
T3386 Kaempferitrin 山奈苷,Lespenefril,Kaempferol 3,7-dirhamnoside,Kaempferol,Lespedin,Lespenephryl cell cycle arrest , Glucokinase , IGF-1R
Kaempferitrin 是天然黄酮苷类化合物，具有缓解疼痛、抗糖尿病、消炎、抗肿瘤和化疗作用，可激活胰岛素信号传导。
T2607 MSDC 0160 MSDC-0160,Mitoglitazone,CAY10415,MSDC0160 Mitochondrial Metabolism , IGF-1R , Others
MSDC 0160 是一种线粒体丙酮酸载体 (MPC) 的调节剂，也是调节噻唑烷二酮的线粒体靶标 (mTOT) 的胰岛素增敏剂。它是一种噻唑烷二酮 (TZD)，具有抗糖尿病和神经保护活性作用。它具有用于阿尔茨海默氏病的潜力。
Insulin Receptor Protein, Human, Recombinant (His & GST Tag)
TMPY-04395
synonym:
Target:
Insulin Receptor Protein, Human, Recombinant (ECD, short isoform, His Tag)
TMPY-01149
synonym:
Target:
Insulin Receptor Protein, Human, Recombinant (long isoform, His Tag), Biotinylated
TMPY-05283
synonym:
Target:
Insulin Receptor Protein, Human, Recombinant (ECD, long isoform, His Tag)
TMPY-01146
synonym:
Target:
[pTyr1146][pTyr1150][pTyr1151]Insulin Receptor (1142-1153)
TP1259
synonym: [pTyr1146][pTyr1150][pTyr1151]Insulin Receptor 1142-1153,Insulin Receptor 1142-1153
Target:
BMS-754807
T2349
synonym:
Target:
HNMPA
T21761
synonym:
Target:
MID-1
T8773
synonym:
Target:
Insulin (human)
T8221
synonym: Insulin(human),INSULIN,甘精胰岛素,胰岛素
Target:
Linsitinib
T6017
synonym: 林西替尼,OSI-906
Target:
Insulin(cattle)
TP1125
synonym: Insulin from bovine pancreas,牛胰岛素,胰岛素
Target:
GRK5-IN-2
T9609
synonym:
Target:
Phentolamine
T8348
synonym:
Target:
MEDICA16
T22967
synonym: MEDICA 16
Target:
SU4984
T9030
synonym:
Target:
NVP-AEW541
T6080
synonym: AEW541
Target:
BMS-536924
T6419
synonym: 胰岛素样生长因子-1 受体拮抗剂,HY-10262,BMS 536924,CS-0117
Target:
GSK1838705A
T3079
synonym:
Target:
Kaempferitrin
T3386
synonym: 山奈苷,Lespenefril,Kaempferol 3,7-dirhamnoside,Kaempferol,Lespedin,Lespenephryl
Target:
MSDC 0160
T2607
synonym: MSDC-0160,Mitoglitazone,CAY10415,MSDC0160
Target:
1 2 3 4 5 6 7 8 9 10
CORPORATE
About Us Privacy Notice Events & News Terms & Conditions
SUPPORT
Contact Us Worldwide Distributors Quality Control Technical Support
RESOURCE
Product Catalog Product Citations Signaling Pathways Solution Calculators
FOLLOW OUR
Social Network
Newsletter Subscription
Subscribe to receive our lastest product updates and special offers!
Corporate
Support
Resource
Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.
Copyright © 2015-2022 TargetMol Chemicals Inc. All rights reserved.