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Search Results for "insulin receptor"

Compounds

Cat No. Product Name
TMPY-04395 Insulin Receptor Protein, Human, Recombinant (His & GST Tag)
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to t...
TMPY-01149 Insulin Receptor Protein, Human, Recombinant (ECD, short isoform, His Tag)
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to t...
TMPY-05283 Insulin Receptor Protein, Human, Recombinant (long isoform, His Tag), Biotinylated
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to t...
TMPY-01146 Insulin Receptor Protein, Human, Recombinant (ECD, long isoform, His Tag)
INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to t...
TP1259 [pTyr1146][pTyr1150][pTyr1151]Insulin Receptor (1142-1153) [pTyr1146][pTyr1150][pTyr1151]Insulin Receptor 1142-1153,Insulin Receptor 1142-1153
[pTyr1146][pTyr1150][pTyr1151]Insulin Receptor (1142-1153) functions as a substrate for insulin receptor tyrosine kinase...
T2349 BMS-754807 IGF-1R , Trk receptor , c-Met/HGFR
BMS754807 是一种可逆的IGF-1R 抑制剂 (IC50:1.8 nM,Ki<2 nM),也是一种可逆的IR 抑制剂 (IC50:7 nM,Ki<2 nM)。它也抑制 Met (IC50:6 nM),RON (IC50:44 nM)...
T21761 HNMPA IGF-1R
HNMPA 是膜不可渗透的胰岛素受体酪氨酸激酶 (insulin receptor tyrosine kinase) 抑制剂。HNMPA 可以抑制人胰岛素受体的酪氨酸和丝氨酸自磷酸化。HNMPA 对环 AMP 依赖性蛋白激酶或蛋白激酶 C ...
T8773 MID-1 IGF-1R , Others
MID-1 是 MG53-IRS-1 相互作用的抑制剂,能够破坏 MG53 与 IRS-1 的分子缔合,并消除 MG53 诱导的 IRS-1 泛素化和骨骼肌降解,升高 IRS-1 表达水平,增加胰岛素信号传导和葡萄糖摄取。
T8221 Insulin (human) Insulin(human),INSULIN,甘精胰岛素,胰岛素 IGF-1R
Insulin 是一种能够调节血液中的葡萄糖水平的多肽激素。
T6017 Linsitinib 林西替尼,OSI-906 IGF-1R
Linsitinib 是选择性的、有效的、具有口服活性的IGF-1和胰岛素受体(IR)的双重抑制剂,IC50分别为 35 和 75 nM。
TP1125 Insulin(cattle) Insulin from bovine pancreas,牛胰岛素,胰岛素 IGF-1R
Insulin cattle 是一种在胰腺 β 细胞中产生的两链多肽激素,在很多哺乳动物细胞培养体系中用作生长因子。
T9609 GRK5-IN-2 GRK
GRK5-IN-2 是基于吡啶的双环化合物,抑制 G 蛋白偶联受体激酶 5 。它调节胰岛素的表达和/或释放,在代谢疾病中有研究价值。
T8348 Phentolamine Adrenergic Receptor
Phentolamine 是一种 alpha-1 和 alpha-2 选择性肾上腺素能受体拮抗剂。
T22967 MEDICA16 MEDICA 16 GPR , ATP Citrate Lyase , Others
MEDICA16 是 GPR40 的特异性激动剂以及 GPR120 的部分激动剂。 MEDICA16 是一种 ATP-柠檬酸裂解酶抑制剂,可显着降低腓肠肌中的细胞内 TG 含量,同时增加胰岛素敏感性。
T9030 SU4984 FGFR , IGF-1R , PDGFR
SU4984 是蛋白质酪氨酸激酶抑制剂,能够抑制成纤维细胞生长因子受体 1 (FGFR1) (IC50:10-20 μM),还能够抑制血小板衍生的生长因子受体和胰岛素受体的活性。它可用于研究癌症。
T6080 NVP-AEW541 AEW541 Tyrosine Kinases , FLT , IGF-1R , Autophagy
NVP-AEW541 是一种IGF-1R 抑制剂,IC50为 0.15 μM。它也抑制InsR,IC50为 0.14 μM。
T6419 BMS-536924 胰岛素样生长因子-1 受体拮抗剂,HY-10262,BMS 536924,CS-0117 MEK , FAK , Apoptosis , IGF-1R , Src
BMS-536924 是一种具有口服活性,竞争性和选择性的胰岛素样生长因子受体激酶和胰岛素受体抑制剂,IC50分别为 100 nM 和 73 nM。它具有抗癌活性。
T3079 GSK1838705A S6 Kinase , IGF-1R , JNK , ALK
GSK1838705A 是一种高效的、可逆的IGF-IR (IC50:2.0 nM) 和胰岛素受体 (IC50:1.6 nM)抑制剂,也可抑制ALK (IC50:0.5 nM)。
T3386 Kaempferitrin 山奈苷,Lespenefril,Kaempferol 3,7-dirhamnoside,Kaempferol,Lespedin,Lespenephryl cell cycle arrest , Glucokinase , IGF-1R
Kaempferitrin 是天然黄酮苷类化合物,具有缓解疼痛、抗糖尿病、消炎、抗肿瘤和化疗作用,可激活胰岛素信号传导。
T2607 MSDC 0160 MSDC-0160,Mitoglitazone,CAY10415,MSDC0160 Mitochondrial Metabolism , IGF-1R , Others
MSDC 0160 是一种线粒体丙酮酸载体 (MPC) 的调节剂,也是调节噻唑烷二酮的线粒体靶标 (mTOT) 的胰岛素增敏剂。它是一种噻唑烷二酮 (TZD),具有抗糖尿病和神经保护活性作用。它具有用于阿尔茨海默氏病的潜力。
Insulin Receptor Protein, Human, Recombinant (His & GST Tag)
TMPY-04395
synonym:
Target:
Insulin Receptor Protein, Human, Recombinant (ECD, short isoform, His Tag)
TMPY-01149
synonym:
Target:
Insulin Receptor Protein, Human, Recombinant (long isoform, His Tag), Biotinylated
TMPY-05283
synonym:
Target:
Insulin Receptor Protein, Human, Recombinant (ECD, long isoform, His Tag)
TMPY-01146
synonym:
Target:
[pTyr1146][pTyr1150][pTyr1151]Insulin Receptor (1142-1153)
TP1259
synonym: [pTyr1146][pTyr1150][pTyr1151]Insulin Receptor 1142-1153,Insulin Receptor 1142-1153
Target:
BMS-754807
T2349
synonym:
Target:
HNMPA
T21761
synonym:
Target:
MID-1
T8773
synonym:
Target:
Insulin (human)
T8221
synonym: Insulin(human),INSULIN,甘精胰岛素,胰岛素
Target:
Linsitinib
T6017
synonym: 林西替尼,OSI-906
Target:
Insulin(cattle)
TP1125
synonym: Insulin from bovine pancreas,牛胰岛素,胰岛素
Target:
GRK5-IN-2
T9609
synonym:
Target:
Phentolamine
T8348
synonym:
Target:
MEDICA16
T22967
synonym: MEDICA 16
Target:
SU4984
T9030
synonym:
Target:
NVP-AEW541
T6080
synonym: AEW541
Target:
BMS-536924
T6419
synonym: 胰岛素样生长因子-1 受体拮抗剂,HY-10262,BMS 536924,CS-0117
Target:
GSK1838705A
T3079
synonym:
Target:
Kaempferitrin
T3386
synonym: 山奈苷,Lespenefril,Kaempferol 3,7-dirhamnoside,Kaempferol,Lespedin,Lespenephryl
Target:
MSDC 0160
T2607
synonym: MSDC-0160,Mitoglitazone,CAY10415,MSDC0160
Target:
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