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Acyltransferase

Acyltransferase is a type of transferase enzyme that acts upon acyl groups.
Cat. No. Product name CAS No. Purity Chemical Structure
T6937 PF-04620110 1109276-89-2 98%
PF-04620110 is an orally active, selective and potent diglyceride acyltransferase-1 (DGAT1) inhibitor with IC50 of 19 nM.
T12426 PF-06424439 1469284-78-3 98%
PF-06424439 is an oral and selective inhibitor of imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) (IC50 of 14 nM).
T13373 YM17E 124900-72-7 98%
YM17E is an inhibitor of ACAT with IC50 of 44 nM in rabbit liver microsomes in vitro.
T23521 VULM 1457 228544-65-8 98%
Acyl-CoA: cholesterol acyltransferase (ACAT) inhibitor
T10035 10,12-Tricosadiynoic acid 66990-30-5 98%
10,12-Tricosadiynoic acid is a highly selective and orally active inhibitor of acyl-CoA oxidase-1 (ACOX1). It can treat the high-fat diet- or obesity-induced met...
T5544 2-Furoic acid 88-14-2 98%
2-Furoic acid, an orally active selective human cathepsin K inhibitor, may have the therapeutic potential for the treatment of diseases characterized by excessiv...
T6365 A 922500 959122-11-3 98%
A922500 is an inhibitor for human and mouse DGAT-1 with IC50 of 7 nM and 24 nM, respectively, good selectivity over related acyltransferases, hERG, and a panel o...
T8236 RHC 80267 83654-05-1 98%
RHC 80267 is a selective inhibitor of DAGL (IC50 : 4 µM in canine platelets)
T31611 Eldacimibe 141993-70-6 98%
Eldacimibe is an ACAT2 inhibitor for the treatment of cardiovascular disease and endocrine and metabolic disorders, study of atherosclerosis and hypercholesterol...
T27245L Eflucimibe 202340-45-2 98%
Eflucimibe is an acyl coenzyme A: cholesterol acyltransferase inhibitor for the treatment of cardiovascular disease and endocrine and metabolic disorders, and ca...
T12767 RP 70676 136609-26-2 98%
RP 70676 is a potent ACAT inhibitor(rat and rabbit ACAT with IC50 of 25 and 44 nM ).
T8314 RP-64477 135239-65-5 98%
RP64477 is the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT) inhibitor.
T0504 Cyclandelate 456-59-7 98%
Cyclandelate, a direct-acting smooth muscle relaxant, is used to dilate blood vessels.
T25635 Lateritin 65454-13-9 98%
Lateritin is An Acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor and a platelet aggregation inhibitor from the mycelial cake of Gibberella lateritium. Bassi...
T12225L Nevanimibe hydrochloride 133825-81-7 98%
Nevanimibe hydrochloride is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM).
T3342 Xanthohumol 6754-58-1 98%
Xanthohumol, also known as 2', 4, 4'-trihydroxy-6'-methoxy-3'-prenylchalcone or desmethylxanthohumol, is a member of the class of compounds known as 3-prenylated...
T22665 PD 128042 114289-47-3 98%
acyl-coenzyme A:cholesterol acyltransferase (ACAT) inhibitor
T25651 Lecimibide 130804-35-2 98%
Lecimibide is a potent and selective inhibitor of acyl coenzyme A: cholesterol acyltransferase (ACAT), which can be used to study diseases due to high lipids.
T23550 YM-750 138046-43-2 98%
Acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor
TN1691 Glabrol 59870-65-4 98%
Glabrol is a PTP1B inhibitor, it is also a CYP1B1 inhibitor, it shows inhibition of CYP1B1 in live cell assay with the IC50 value of 15uM.
PF-04620110
T6937
PF-04620110 is an orally active, selective and potent diglyceride acyltransferase-1 (DGAT1) inhibitor with IC50 of 19 nM.
PF-06424439
T12426
PF-06424439 is an oral and selective inhibitor of imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) (IC50 of 14 nM).
YM17E
T13373
YM17E is an inhibitor of ACAT with IC50 of 44 nM in rabbit liver microsomes in vitro.
VULM 1457
T23521
Acyl-CoA: cholesterol acyltransferase (ACAT) inhibitor
10,12-Tricosadiynoic acid
T10035
10,12-Tricosadiynoic acid is a highly selective and orally active inhibitor of acyl-CoA oxidase-1 (ACOX1). It can treat the high-fat diet- or obesity-induced met...
2-Furoic acid
T5544
2-Furoic acid, an orally active selective human cathepsin K inhibitor, may have the therapeutic potential for the treatment of diseases characterized by excessiv...
A 922500
T6365
A922500 is an inhibitor for human and mouse DGAT-1 with IC50 of 7 nM and 24 nM, respectively, good selectivity over related acyltransferases, hERG, and a panel o...
RHC 80267
T8236
RHC 80267 is a selective inhibitor of DAGL (IC50 : 4 µM in canine platelets)
Eldacimibe
T31611
Eldacimibe is an ACAT2 inhibitor for the treatment of cardiovascular disease and endocrine and metabolic disorders, study of atherosclerosis and hypercholesterol...
Eflucimibe
T27245L
Eflucimibe is an acyl coenzyme A: cholesterol acyltransferase inhibitor for the treatment of cardiovascular disease and endocrine and metabolic disorders, and ca...
RP 70676
T12767
RP 70676 is a potent ACAT inhibitor(rat and rabbit ACAT with IC50 of 25 and 44 nM ).
RP-64477
T8314
RP64477 is the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT) inhibitor.
Cyclandelate
T0504
Cyclandelate, a direct-acting smooth muscle relaxant, is used to dilate blood vessels.
Lateritin
T25635
Lateritin is An Acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor and a platelet aggregation inhibitor from the mycelial cake of Gibberella lateritium. Bassi...
Nevanimibe hydrochloride
T12225L
Nevanimibe hydrochloride is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM).
Xanthohumol
T3342
Xanthohumol, also known as 2', 4, 4'-trihydroxy-6'-methoxy-3'-prenylchalcone or desmethylxanthohumol, is a member of the class of compounds known as 3-prenylated...
PD 128042
T22665
acyl-coenzyme A:cholesterol acyltransferase (ACAT) inhibitor
Lecimibide
T25651
Lecimibide is a potent and selective inhibitor of acyl coenzyme A: cholesterol acyltransferase (ACAT), which can be used to study diseases due to high lipids.
YM-750
T23550
Acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor
Glabrol
TN1691
Glabrol is a PTP1B inhibitor, it is also a CYP1B1 inhibitor, it shows inhibition of CYP1B1 in live cell assay with the IC50 value of 15uM.
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