rs-1

RS-1 is a RAD51 activator. RS-1 also increases CRISPR/Cas9-mediated knock-in efficiencies.

RS1-PDK1 inhibitor (RS 1) is a selective inhibitor of the protein kinase PDK1 that can be used to treat and prevent disease or disorders.

ARS-1323 is the racemate of ARS-1620 and a mutant K-ras G12C inhibitor.

ARS-1630 is a mutant K-ras G12C inhibitor. It is a less active enantiomer of ARS-1620.

(RS)-G12Di-1 is a selective covalent inhibitor of K-Ras-G12D.

RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.

ARS-1323-alkyne is a switch-II pocket (S-IIP) inhibitor and a conformational specific chemical reporter of KRASG12C nucleotide state in living cells.

MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).

MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist.

Compound 2, known as KCC2 potentiators-1, acts as an enhancer of the potassium chloride cotransporter-2 (KCC2). It holds potential for applications in studies related to neurological disorders.

MRS-1477 is used as a TRPV1 positive allosteric modulator (PAM).

RS-136270 is a bioactive chemical.

RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.

RS-102221 is a selective antagonist of the 5-HT2C receptor with a K i of 10 nM, demonstrating nearly 100-fold more selectivity for the 5-HT2C receptor over the 5-HT2A and 5-HT2B receptors. This compound not only has the potential to promote the differentiation of new nerve cells but also increases food intake and weight gain in rats.

RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).

'(2α,3β,4α)-2,3,19-Trihydroxyurs-12-ene-23,28-dioic acid, a saponin isolated from Rubus ellipticus var. obcordatus, inhibits α-Glucosidase with an IC 50 of 1.68 mM [1].'

ARS-1620 is a covalent inhibitor of K-RASG12C.

2α,3β,24-Trihydroxyurs-12-en-28-oic acid, a natural product, is isolated from *Salvia palaestina* [1].

2a,3a,23-Trihydroxyurs-12,20(30)-dien-28-oic acid (compound 3), a triterpenoid, markedly reduces fibronectin levels by 27.66% at a 10 μM concentration in HK-2 cells subjected to high-glucose and TGF-b1 induction [1].

RS-127445 maleate is a chemically selective antagonist with a high affinity for the 5-HT2B receptor, boasting an oral bioavailability and a pKi of 9.5.

2alpha,19alpha-Dihydroxy-3-oxo-urs-12-en-28-oic acid has anti-HIV activity. It shows an inhibitory effect on the activation of Epstein-Barr virus early antigen (EBV-EA) induced by 12-O-tetradecanoylphorbol-13-acetate (TPA) and causes a significant delay o

6,19-Dihydroxyurs-12-en-3-oxo-28-oic acid is a natural product for research related to life sciences. The catalog number is TN3143 and the CAS number is 194027-11-7.

3β-Acetoxyurs-12-en-11-one (11-Ketoamyrinacetate) is an ursane triterpene natural product present in the stem bark of Morus mesozygia and the leaves of Ficus hirta Vahl (Moraceae).

3β-Hydroxy-27-p-Z-coumaroyloxyurs-12-en-28-oic acid (compound 8) is a triterpene ester HIV-1 protease inhibitor with potential for use in antiretroviral combination therapy for AIDS.