Home Tools
Log in
Cart

Search Result

Search Results for " rem "

20

Compounds

Cat No. Product Name Synonyms Targets
T7413 JNJ-5207852 Histamine Receptor
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
T8822 JNJ-5207852 dihydrochloride Histamine Receptor
JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.
T12612 (R)-Apremilast (R)-CC-10004 Others
(R)-Apremilast ((R)-CC-10004) is the enantiomer of Apremilast and one of the isoindoline derivatives.
T16991 Targapremir-210 TGP-210 Apoptosis
Targapremir-210 (TGP-210) is a selective and potent miRNA-210 (miRNA-210) inhibitor that inhibits pre-miR-210 processing and induces apoptosis in breast cancer cells.
T16730 Remibrutinib BTK
Remibrutinib inhibits BTK activity with an IC50 value of 0.023 μM in blood. Remibrutinib is an effective and orally active Bruton tyrosine kinase inhibitor (IC50: 1 nM). Remibrutinib has the potential for Chronic urticar...
T23232 Remoxipride hydrochloride Remoxipride Hydrochloride Anhydrous,Roxiam,(S)-Remoxipride Hydrochloride Dopamine Receptor
Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoceptor.
T5555 Siremadlin NVP-HDM 201 E1/E2/E3 Enzyme
Siremadlin (NVP-HDM 201) is a potent, orally bioavailable and highly specific p53-MDM2 interaction inhibitor.
T77466 Tremelimumab Ticilimumab,CP-675206 Others
Tremelimumab is a cytotoxic T-lymphocyte-associated antigen-4 (CTLA-4) blocking antibody.Tremelimumab is often used in combination with Durvalumab for the treatment of solid cancers such as hepatocellular carcinoma and l...
T36857L Premarin Estrone 3-sulfate,Estrone sulfate Estrogen Receptor/ERR
Premarin (Estrone 3-sulfate) is an an estrogen sulfate with neuroprotective actions during traumatic brain injury.
T3499 Remodelin Histone Acetyltransferase
Remodelin is an effective and specific inhibitor of the acetyl-transferase protein NAT10.
T12339 Oxotremorine M iodide Oxotremorine methiodide AChR
Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.
T2923 Apremilast CC-10004 Apoptosis , TNF , PDE
Apremilast (CC-10004) (CC-10004) is a potent and orally active PDE4 (IC50=74 nM) with anti-inflammation activities.
T6133 Remodelin hydrobromide Remodelin,Remodelin HBR RAAS , Histone Acetyltransferase
Remodelin hydrobromide (Remodelin HBR) is a novel potent and selective inhibitor of the acetyl-transferase protein NAT10.
T7766 Remdesivir GS-5734 SARS-CoV , DNA/RNA Synthesis
Remdesivir (GS-5734) is a nucleoside analog, a broad-spectrum antiviral compound that exerts its activity by inhibiting the RNA-dependent RNA polymerase of viruses. Remdesivir is active against Ebola, SARS, and MERS viru...
T2429 Olverembatinib dimesylate GZD824 Dimesylate,HQP1351 Bcr-Abl
Olverembatinib dimesylate (GZD824 Dimesylate) is a novel orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT) and Bcr-Abl(T315I).
T16729 Remetinostat SHP-141 HDAC
Remetinostat (SHP-141), a hydroxamic acid-based inhibitor of histone deacetylase enzymes, is currently being developed for the treatment of cutaneous T-cell lymphoma.
T34286 Remogliflozin etabonate GSK189075,GSK 189075,GSK-189075A,GSK189075A,GSK-189075,GSK 189075A SGLT
Remogliflozin etabonate (GSK189075A) is a prodrug of regaliflozin and an inhibitor SGLT2 with Ki values of 1.95, 2.14, 8.57, and 43.1μM for hSGLT2, rSGLT2, rSGLT1, and hSGLT1, respectively.
T23116 Oxotremorine sesquifumarate AChR
Oxotremorine sesquifumarate is a muscarinic agonist.
T3071 Olverembatinib GZD 824 Bcr-Abl
Olverembatinib (GZD 824) is an orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT, IC50: 0.34 nM) and Bcr-Abl(T315I, IC50: 0.68 nM).
T7608 Bremelanotide Acetate bremelanotide,PT-141 Acetate Melanocortin Receptor
Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
1 2 3 4 5 6
TargetMol