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Bremelanotide Acetate

Name: Bremelanotide Acetate
Brand: TargetMol
SKU: T7608
Price: 46 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T7608Cas No. 1607799-13-2

Alias PT-141 Acetate

Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .

Bremelanotide Acetate

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Purity: 96.72%

Catalog No. T7608Alias PT-141 AcetateCas No. 1607799-13-2

Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .

Pack Size	Price	USA Warehouse	Global Warehouse
10 mg	$46	In Stock	In Stock
25 mg	$83	In Stock	In Stock
50 mg	$139	In Stock	In Stock
100 mg	$207	-	In Stock
1 mL x 10 mM (in DMSO)	$65	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

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Batch Information

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Purity:96.72%

Appearance:Solid

Color:White to Yellow

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COA HPLC MS

Product Introduction

Bioactivity

Description	Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
In vivo	Treatment with Bremelanotide?(100 or 200 μg/kg) significantly increased proceptive solicitations in females primed with E+Por E alone (E+O) in bilevel chambers[1]
Animal Research	Bremelanotide(PT-141), a cyclic heptapeptide melanocortin analogue (Palatin Technologies, Cranbury, NJ), was dissolved in saline to obtain doses of 50, 100, and 200 μg/kg/ml, and injected s.c. 5 min before each behavioral test. An equal volume of saline was administered to control animals[1].
Synonyms	PT-141 Acetate

Chemical Properties

Molecular Weight	1085.22
Formula	C₅₂H₇₂N₁₄O₁₂
Cas No.	1607799-13-2
Smiles	CC(O)=O.[H][C@]1(CCCCNC(=O)C[C@H](NC(=O)[C@H](CCCC)NC(C)=O)C(=O)N[C@@H](Cc2cnc[nH]2)C(=O)N[C@]([H])(Cc2ccccc2)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1)C(O)=O
Relative Density.	no data available
Sequence	Ac-Nle-Asp(1)-His-D-Phe-Arg-Trp-Lys(1)-OH.CH3CO2H
Sequence Short	XDHFRWK

Storage & Solubility Information

Storage

keep away from moisture,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 122.5 mg/mL (112.88 mM), Sonication is recommended.

In Vivo Formulation

10% DMSO+40% PEG300+5% Tween 80+45% Saline: 2 mg/mL (1.84 mM), Sonication is recommended.

Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	0.9215 mL	4.6074 mL	9.2147 mL	46.0736 mL
5 mM	0.1843 mL	0.9215 mL	1.8429 mL	9.2147 mL
10 mM	0.0921 mL	0.4607 mL	0.9215 mL	4.6074 mL
20 mM	0.0461 mL	0.2304 mL	0.4607 mL	2.3037 mL
50 mM	0.0184 mL	0.0921 mL	0.1843 mL	0.9215 mL
100 mM	0.0092 mL	0.0461 mL	0.0921 mL	0.4607 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc