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Search Results for " long-acting "

Targets

174

Compounds

5

Natural Products

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T5051 Isopropamide Iodide AChR
Isopropamide iodide is a long-acting anticholinergic drug. It is used in the treatment of peptic ulcers and other gastrointestinal disorders. It also acts as a muscarinic receptor antagonist which can be applied to the t...
T4985 Neticonazole Hydrochloride Antifungal
Neticonazole Hydrochloride is an imidazole antifungal for the treatment of fungal skin infections. Neticonazole is reported as a potent exosome inhibitor which can block the activity of exosomes.
T0388 Cilnidipine FRC-8653 Calcium Channel
Cilnidipine (FRC-8653)(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity.
T2390 Cevimeline hydrochloride hemihydrate AChR
Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.
T7943 Fluphenazine decanoate Dopamine Receptor
Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.
T3716 Rolapitant SCH619734 Neurokinin receptor
Rolapitant (SCH619734) Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity. ...
T5159 Olodaterol hydrochloride BI-1744 HCl,BI 1744 hydrochloride Adrenergic Receptor
Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and activating β2-adrenergic receptors...
T20720 Norethisterone enanthate NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,NSC-9564 Estrogen/progestogen Receptor
Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.
T31716 Etidocaine Hydrochloride W-19053,Duranest,W19053,W 19053 Sodium Channel
Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel.
T0749 Succinylsulfathiazole Succinylsulphathiazole Antibacterial , Antibiotic , Autophagy
Succinylsulfathiazole (Succinylsulphathiazole) is a sulfonamide. An ultra long-acting drug.
T0364L Dibucaine hydrochloride Cinchocaine HCl,Dibucaine HCl,Cinchocaine hydrochloride Sodium Channel , AChR
Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.
T28360 PF-00489791 PF-4634817,PF 4634817,PF00489791,PF 00489791,PF4634817 PDE
PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy.
T33386 Milveterol HCl Milveterol,GSK-159797,GSK 159797,GSK159797 Adrenergic Receptor
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).
T1629 Rifapentine MDL473,Rifapentina,Rifapentinum,DL 473,Priftin,Cyclopentylrifampicin DNA/RNA Synthesis , Antibacterial , Antibiotic
Rifapentine (Rifapentinum) is a long-acting, cyclopentyl-substituted derivative of rifamycin used to treat mycobacterium infections.
T1239 Indacaterol maleate QAB149 Adrenergic Receptor
Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
T6876 Liraglutide Liraglutidum,Victoza,Liraglutida,NN2211 Glucagon Receptor
Liraglutide (Liraglutida) is a long-acting GLP-1 receptor agonist.
T11235 Estradiol 3-sulfamate ES-J 995,E2MATE,BLE 00084 Others
.Estradiol 3-sulfamate inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. Estradiol 3-sulfamate is a potent, long-acting, and orally active steroid sulfatase inhibitor.
T4499 Mequitazine Metaplexan,Virginan,Primalan,LM-209 Histamine Receptor
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
T22508 3-CPMT Chlortropbenzyl hydrochloride,3-[(4-chlorophenyl)-phenylmethoxy]-8-methyl-8-azabicyclo[3.2.1]octane hydrochloride,SL6057,Wy 2149,FC-1 Dopamine Receptor
3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.
T31716L Etidocaine Others
Etidocaine is an amino acidamide that acts as a local anesthetic with fast onset and long-acting properties.
T1446 Bambuterol hydrochloride (±)-Bambuterol hydrochloride,KWD-2183 hydrochloride,Bambuterol HCl Adrenergic Receptor , AChR
Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
T35048 Verofylline CK 0383,Verofilina,CK-0383,Verofyllinum,CK0383 PDE
Verofylline (Verofyllinum) is an orally available, long-acting, multiacting, methylxanthine-substituted bronchodilator with inhibitory effects on PDE4 for the treatment of asthma disease research obesity.
T25263 Clopimozide R-29764,NSC-335305,NSC 335305,NSC335305,R 29764 Calcium Channel
Clopimozide (R-29764) acts as a calcium channel antagonist and inhibits [3H] nilandipine binding.Clopimozide is a novel and orally available long-acting antischizophrenic psychostatic compound.
T20435L Leuphasyl TFA Opioid Receptor
Leuphasyl TFA is an amid peptide, a δ-opioid receptor agonist, is a degradation resistant long-acting Leu-enkephalin analog used to study the signaling pathway of delta opioid receptors. Leuphasyl TFA is a potent, long-a...
T16433 Pancopride LAS 30451 5-HT Receptor
Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-induced vomiting.
T0127 Glimepiride Glimperide,HOE-490 Potassium Channel
Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.
T0026 Sulfalene Sulfalene(SMPZ),Sulfalen,SMP2,Butadiene sulfone,AS-18908,Sulfametopyrazine,3-Sulfolene Antibacterial , Antibiotic , Parasite , Autophagy
Sulfalene (SMP2), a long-acting sulfonamide antibiotic, is used for the therapy of chronic bronchitis, urinary tract infections, and malaria.
T4119 Octreotide Acetate SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate) Somatostatin
Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.
T6237 Trelagliptin SYR-472 Proteasome , DPP-4
Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.
T6505 Formoterol fumarate Formoterol Hemifumarate,NSC 299587,Eformoterol Hemifumarate,CGP 25827A,Eformoterol,YM 08316 Adrenergic Receptor
Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of chronic obstructive pulmonary disease(COPD) and asthma.
T1645 Ramipril HOE-498,Tritace,Altace,Carasel Apoptosis , RAAS
Ramipril (Altace) is a long-acting angiotensin-converting enzyme inhibitor. It is a prodrug that is transformed in the liver to its active metabolite ramiprilat.
T19858 Brodimoprim DHFR , Antibacterial
Brodimoprim is an inhibitor of dihydrofolate reductase(DHFR). Brodimoprim is also a long-acting broad-spectrum antibacterial agent characterized by a good pharmacokinetic profile.
T9124 Laninamivir octanoate CS-8958 Influenza Virus
Laninamivir octanoate (CS-8958) is a long acting influenza neuraminidase (NA) inhibitor which shows superior anti-influenza virus activity.
T8748 Exendin-4 acetate Glucagon Receptor
Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).
T16952 Sulfabrom Sulfabromomethazine,N 3517 Anti-infection , Antibacterial
Sulfabrom (Sulfabromomethazine) is a long-acting sulfonamide medicine for the treatment of coccidiosis and various bacterial infections in poultry, pigs, and cattle.
T4102 Goserelin acetate Fertilan,ICI-118630 acetate,Zoladex Apoptosis , GNRH Receptor
Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
T0748 Sulfameter 5-Methoxysulfadiazine,Sulfametoxydiazine DHFR , Antibacterial , Antibiotic
Sulfameter (Sulfametoxydiazine) is a long-acting sulfonamide antibacterial agent used to treat urinary tract infections and leprosy.
T15301 Fluspirilene Redeptin,R 6218 Calcium Channel
Fluspirilene (R 6218) is a non-competitive L-type calcium channel antagonist (IC50: 0.03 μM).Fluspirilene is a long-acting antipsychotic compound used in the treatment of schizophrenia.
TP1796 Albiglutide TFA (782500-75-8 free base) Albiglutide TFA Glucagon Receptor
Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
T0706 Lisinopril dihydrate Lisinopril,Renacor,MK-521 (dihydrate) RAAS , MRP
Lisinopril dihydrate (MK-521) is an orally bioavailable, long-acting angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.
T1909 L-701324 L701324 NMDAR , iGluR
L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.
T6566 Levobupivacaine hydrochloride Levobupivacaine HCl,(S)-(-)-Bupivacaine HCl,(S)-(-)-Bupivacaine monohydrochloride Sodium Channel
Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, which is the pure S(-)-enantiomer of bupivacaine. It was utilized as a long-acting local anesthetic...
T4991 Ertapenem sodium MK-826,L-749345 Antibacterial , Antibiotic
Ertapenem sodium (MK-826) is a new long-acting 1-β-methyl carbapenem antibiotic with a broad antibacterial spectrum including common aerobic and anaerobic bacteria and organisms with extended-spectrum β-lactamases.
T0699 Sulfamonomethoxine Antibacterial , Antibiotic
Sulfamonomethoxine is a long-acting sulfonamide antibacterial agent, blocks the synthesis of folic acid by inhibiting synthetase of dihydropteroate.
T6098 Cabotegravir GSK744,GSK-1265744,S/GSK1265744 HIV Protease
Cabotegravir (S/GSK1265744) (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor and inhibits the HIV-1 integrase catalyzed strand transfer reaction (IC50: 3.0 nM).
T1423 3-Methylsalicylic acid Hydroxytoluic acid,o-Cresotic acid COX
3-Methylsalicylic acid (o-Cresotic acid) is a long-acting salicylate derivative with antilipidemic properties. Hydroxytoluic acid has been shown to lower plasma free fatty acid and cholesterol levels.
T16759 Ritanserin R 55667 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
T6457 CTEP mGluR5 inhibitor,RO 4956371 GluR
CTEP (RO 4956371) (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold selectivity over other mGlu receptors.
T13106 TD-5471 hydrochloride Adrenergic Receptor
TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (COPD).
T12829 Salmeterol GR33343X Adrenergic Receptor
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.

Compounds

Isopropamide Iodide
T5051
Synonym:
Target: AChR
Neticonazole Hydrochloride
T4985
Synonym:
Target: Antifungal
Cilnidipine
T0388
Synonym: FRC-8653
Target: Calcium Channel
Cevimeline hydrochloride hemihydrate
T2390
Synonym:
Target: AChR
Fluphenazine decanoate
T7943
Synonym:
Target: Dopamine Receptor
Rolapitant
T3716
Synonym: SCH619734
Target: Neurokinin receptor
Olodaterol hydrochloride
T5159
Synonym: BI-1744 HCl,BI 1744 hydrochloride
Target: Adrenergic Receptor
Norethisterone enanthate
T20720
Synonym: NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,NSC-9564
Target: Estrogen/progestogen Receptor
Etidocaine Hydrochloride
T31716
Synonym: W-19053,Duranest,W19053,W 19053
Target: Sodium Channel
Succinylsulfathiazole
T0749
Synonym: Succinylsulphathiazole
Target: Antibacterial, Antibiotic, Autophagy
Dibucaine hydrochloride
T0364L
Synonym: Cinchocaine HCl,Dibucaine HCl,Cinchocaine hydrochloride
Target: Sodium Channel, AChR
PF-00489791
T28360
Synonym: PF-4634817,PF 4634817,PF00489791,PF 00489791,PF4634817
Target: PDE
Milveterol HCl
T33386
Synonym: Milveterol,GSK-159797,GSK 159797,GSK159797
Target: Adrenergic Receptor
Rifapentine
T1629
Synonym: MDL473,Rifapentina,Rifapentinum,DL 473,Priftin,Cyclopentylrifampicin
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Indacaterol maleate
T1239
Synonym: QAB149
Target: Adrenergic Receptor
Liraglutide
T6876
Synonym: Liraglutidum,Victoza,Liraglutida,NN2211
Target: Glucagon Receptor
Estradiol 3-sulfamate
T11235
Synonym: ES-J 995,E2MATE,BLE 00084
Target: Others
Mequitazine
T4499
Synonym: Metaplexan,Virginan,Primalan,LM-209
Target: Histamine Receptor
3-CPMT
T22508
Synonym: Chlortropbenzyl hydrochloride,3-[(4-chlorophenyl)-phenylmethoxy]-8-methyl-8-azabicyclo[3.2.1]octane hydrochloride,SL6057,Wy 2149,FC-1
Target: Dopamine Receptor
Etidocaine
T31716L
Synonym:
Target: Others
Bambuterol hydrochloride
T1446
Synonym: (±)-Bambuterol hydrochloride,KWD-2183 hydrochloride,Bambuterol HCl
Target: Adrenergic Receptor, AChR
Verofylline
T35048
Synonym: CK 0383,Verofilina,CK-0383,Verofyllinum,CK0383
Target: PDE
Clopimozide
T25263
Synonym: R-29764,NSC-335305,NSC 335305,NSC335305,R 29764
Target: Calcium Channel
Leuphasyl TFA
T20435L
Synonym:
Target: Opioid Receptor
Pancopride
T16433
Synonym: LAS 30451
Target: 5-HT Receptor
Glimepiride
T0127
Synonym: Glimperide,HOE-490
Target: Potassium Channel
Sulfalene
T0026
Synonym: Sulfalene(SMPZ),Sulfalen,SMP2,Butadiene sulfone,AS-18908,Sulfametopyrazine,3-Sulfolene
Target: Antibacterial, Antibiotic, Parasite, Autophagy
Octreotide Acetate
T4119
Synonym: SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)
Target: Somatostatin
Trelagliptin
T6237
Synonym: SYR-472
Target: Proteasome, DPP-4
Formoterol fumarate
T6505
Synonym: Formoterol Hemifumarate,NSC 299587,Eformoterol Hemifumarate,CGP 25827A,Eformoterol,YM 08316
Target: Adrenergic Receptor
Ramipril
T1645
Synonym: HOE-498,Tritace,Altace,Carasel
Target: Apoptosis, RAAS
Brodimoprim
T19858
Synonym:
Target: DHFR, Antibacterial
Laninamivir octanoate
T9124
Synonym: CS-8958
Target: Influenza Virus
Exendin-4 acetate
T8748
Synonym:
Target: Glucagon Receptor
Sulfabrom
T16952
Synonym: Sulfabromomethazine,N 3517
Target: Anti-infection, Antibacterial
Goserelin acetate
T4102
Synonym: Fertilan,ICI-118630 acetate,Zoladex
Target: Apoptosis, GNRH Receptor
Sulfameter
T0748
Synonym: 5-Methoxysulfadiazine,Sulfametoxydiazine
Target: DHFR, Antibacterial, Antibiotic
Fluspirilene
T15301
Synonym: Redeptin,R 6218
Target: Calcium Channel
Albiglutide TFA (782500-75-8 free base)
TP1796
Synonym: Albiglutide TFA
Target: Glucagon Receptor
Lisinopril dihydrate
T0706
Synonym: Lisinopril,Renacor,MK-521 (dihydrate)
Target: RAAS, MRP
L-701324
T1909
Synonym: L701324
Target: NMDAR, iGluR
Levobupivacaine hydrochloride
T6566
Synonym: Levobupivacaine HCl,(S)-(-)-Bupivacaine HCl,(S)-(-)-Bupivacaine monohydrochloride
Target: Sodium Channel
Ertapenem sodium
T4991
Synonym: MK-826,L-749345
Target: Antibacterial, Antibiotic
Sulfamonomethoxine
T0699
Synonym:
Target: Antibacterial, Antibiotic
Cabotegravir
T6098
Synonym: GSK744,GSK-1265744,S/GSK1265744
Target: HIV Protease
3-Methylsalicylic acid
T1423
Synonym: Hydroxytoluic acid,o-Cresotic acid
Target: COX
Ritanserin
T16759
Synonym: R 55667
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
CTEP
T6457
Synonym: mGluR5 inhibitor,RO 4956371
Target: GluR
TD-5471 hydrochloride
T13106
Synonym:
Target: Adrenergic Receptor
Salmeterol
T12829
Synonym: GR33343X
Target: Adrenergic Receptor
1 2 3 4
Cat No. Product Name Synonyms Targets
T1261 Medroxyprogesterone Acetate Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,Farlutin,Medroxyprogesterone (acetate) Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , Androgen Receptor , Endogenous Metabolite
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally or by intramuscular injection and has also been...
T0086 Galanthamine hydrobromide Galantamine hydrobromide,Galanthamine HBr AChR , AChE
Galanthamine hydrobromide (Galantamine hydrobromide), a long-acting and centrally active AChE inhibitor (IC50:410 nM), is an allosteric potentiator at neuronal nicotinic ACh receptors.
T3S2007 MRE-269 MRE 269,ACT-333679,MRE269 Prostaglandin Receptor
MRE-269 (ACT-333679) is an orally available and long-acting prostacyclin receptor agonist prodrug. MRE-269(ACT-333679) is used for the treatment of pulmonary arterial hypertension. MRE-269(ACT-333679) is an active metabo...
T0012 Cinchonine LA40221,(8R,9S)-Cinchonine Apoptosis , P-gp , Parasite
Cinchonine (LA40221), a local anesthetic of the amide type, now generally used for surface anesthesia. It is one of the most potent and toxic of the long-acting local narcotics and its parenteral use is restricted to spi...
T2520 Desloratadine Sch34117,NSC 675447 Endogenous Metabolite , Histamine Receptor
Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typical histaminergic effects on H1-receptors in bronchial smoot...

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-01816 Pentraxin 3 Protein, Human, Recombinant (His) Human HEK293
Pentraxin-related protein PTX3, also known as Tumor necrosis factor alpha-induced protein 5, Tumor necrosis factor-inducible gene 14 protein, TSG-14, PTX3 and TNFAIP5, is a secreted protein that contains one pentaxin dom...
TargetMol