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Cat No. | Product Name | Synonyms | Targets |
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T5051 | Isopropamide Iodide | AChR | |
Isopropamide iodide is a long-acting anticholinergic drug. It is used in the treatment of peptic ulcers and other gastrointestinal disorders. It also acts as a muscarinic receptor antagonist which can be applied to the t... | |||
T4985 | Neticonazole Hydrochloride | Antifungal | |
Neticonazole Hydrochloride is an imidazole antifungal for the treatment of fungal skin infections. Neticonazole is reported as a potent exosome inhibitor which can block the activity of exosomes. | |||
T0388 | Cilnidipine | FRC-8653 | Calcium Channel |
Cilnidipine (FRC-8653)(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity. | |||
T2390 | Cevimeline hydrochloride hemihydrate | AChR | |
Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome. | |||
T7943 | Fluphenazine decanoate | Dopamine Receptor | |
Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia. | |||
T3716 | Rolapitant | SCH619734 | Neurokinin receptor |
Rolapitant (SCH619734) Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity. ... | |||
T5159 | Olodaterol hydrochloride | BI-1744 HCl,BI 1744 hydrochloride | Adrenergic Receptor |
Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and activating β2-adrenergic receptors... | |||
T20720 | Norethisterone enanthate | NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,NSC-9564 | Estrogen/progestogen Receptor |
Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects. | |||
T31716 | Etidocaine Hydrochloride | W-19053,Duranest,W19053,W 19053 | Sodium Channel |
Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel. | |||
T0749 | Succinylsulfathiazole | Succinylsulphathiazole | Antibacterial , Antibiotic , Autophagy |
Succinylsulfathiazole (Succinylsulphathiazole) is a sulfonamide. An ultra long-acting drug. | |||
T0364L | Dibucaine hydrochloride | Cinchocaine HCl,Dibucaine HCl,Cinchocaine hydrochloride | Sodium Channel , AChR |
Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia. | |||
T28360 | PF-00489791 | PF-4634817,PF 4634817,PF00489791,PF 00489791,PF4634817 | PDE |
PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy. | |||
T33386 | Milveterol HCl | Milveterol,GSK-159797,GSK 159797,GSK159797 | Adrenergic Receptor |
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD). | |||
T1629 | Rifapentine | MDL473,Rifapentina,Rifapentinum,DL 473,Priftin,Cyclopentylrifampicin | DNA/RNA Synthesis , Antibacterial , Antibiotic |
Rifapentine (Rifapentinum) is a long-acting, cyclopentyl-substituted derivative of rifamycin used to treat mycobacterium infections. | |||
T1239 | Indacaterol maleate | QAB149 | Adrenergic Receptor |
Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist. | |||
T6876 | Liraglutide | Liraglutidum,Victoza,Liraglutida,NN2211 | Glucagon Receptor |
Liraglutide (Liraglutida) is a long-acting GLP-1 receptor agonist. | |||
T11235 | Estradiol 3-sulfamate | ES-J 995,E2MATE,BLE 00084 | Others |
.Estradiol 3-sulfamate inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. Estradiol 3-sulfamate is a potent, long-acting, and orally active steroid sulfatase inhibitor. | |||
T4499 | Mequitazine | Metaplexan,Virginan,Primalan,LM-209 | Histamine Receptor |
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist. | |||
T22508 | 3-CPMT | Chlortropbenzyl hydrochloride,3-[(4-chlorophenyl)-phenylmethoxy]-8-methyl-8-azabicyclo[3.2.1]octane hydrochloride,SL6057,Wy 2149,FC-1 | Dopamine Receptor |
3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent. | |||
T31716L | Etidocaine | Others | |
Etidocaine is an amino acidamide that acts as a local anesthetic with fast onset and long-acting properties. | |||
T1446 | Bambuterol hydrochloride | (±)-Bambuterol hydrochloride,KWD-2183 hydrochloride,Bambuterol HCl | Adrenergic Receptor , AChR |
Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma. | |||
T35048 | Verofylline | CK 0383,Verofilina,CK-0383,Verofyllinum,CK0383 | PDE |
Verofylline (Verofyllinum) is an orally available, long-acting, multiacting, methylxanthine-substituted bronchodilator with inhibitory effects on PDE4 for the treatment of asthma disease research obesity. | |||
T25263 | Clopimozide | R-29764,NSC-335305,NSC 335305,NSC335305,R 29764 | Calcium Channel |
Clopimozide (R-29764) acts as a calcium channel antagonist and inhibits [3H] nilandipine binding.Clopimozide is a novel and orally available long-acting antischizophrenic psychostatic compound. | |||
T20435L | Leuphasyl TFA | Opioid Receptor | |
Leuphasyl TFA is an amid peptide, a δ-opioid receptor agonist, is a degradation resistant long-acting Leu-enkephalin analog used to study the signaling pathway of delta opioid receptors. Leuphasyl TFA is a potent, long-a... | |||
T16433 | Pancopride | LAS 30451 | 5-HT Receptor |
Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-induced vomiting. | |||
T0127 | Glimepiride | Glimperide,HOE-490 | Potassium Channel |
Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity. | |||
T0026 | Sulfalene | Sulfalene(SMPZ),Sulfalen,SMP2,Butadiene sulfone,AS-18908,Sulfametopyrazine,3-Sulfolene | Antibacterial , Antibiotic , Parasite , Autophagy |
Sulfalene (SMP2), a long-acting sulfonamide antibiotic, is used for the therapy of chronic bronchitis, urinary tract infections, and malaria. | |||
T4119 | Octreotide Acetate | SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate) | Somatostatin |
Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone. | |||
T6237 | Trelagliptin | SYR-472 | Proteasome , DPP-4 |
Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor. | |||
T6505 | Formoterol fumarate | Formoterol Hemifumarate,NSC 299587,Eformoterol Hemifumarate,CGP 25827A,Eformoterol,YM 08316 | Adrenergic Receptor |
Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of chronic obstructive pulmonary disease(COPD) and asthma. | |||
T1645 | Ramipril | HOE-498,Tritace,Altace,Carasel | Apoptosis , RAAS |
Ramipril (Altace) is a long-acting angiotensin-converting enzyme inhibitor. It is a prodrug that is transformed in the liver to its active metabolite ramiprilat. | |||
T19858 | Brodimoprim | DHFR , Antibacterial | |
Brodimoprim is an inhibitor of dihydrofolate reductase(DHFR). Brodimoprim is also a long-acting broad-spectrum antibacterial agent characterized by a good pharmacokinetic profile. | |||
T9124 | Laninamivir octanoate | CS-8958 | Influenza Virus |
Laninamivir octanoate (CS-8958) is a long acting influenza neuraminidase (NA) inhibitor which shows superior anti-influenza virus activity. | |||
T8748 | Exendin-4 acetate | Glucagon Receptor | |
Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM). | |||
T16952 | Sulfabrom | Sulfabromomethazine,N 3517 | Anti-infection , Antibacterial |
Sulfabrom (Sulfabromomethazine) is a long-acting sulfonamide medicine for the treatment of coccidiosis and various bacterial infections in poultry, pigs, and cattle. | |||
T4102 | Goserelin acetate | Fertilan,ICI-118630 acetate,Zoladex | Apoptosis , GNRH Receptor |
Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer. | |||
T0748 | Sulfameter | 5-Methoxysulfadiazine,Sulfametoxydiazine | DHFR , Antibacterial , Antibiotic |
Sulfameter (Sulfametoxydiazine) is a long-acting sulfonamide antibacterial agent used to treat urinary tract infections and leprosy. | |||
T15301 | Fluspirilene | Redeptin,R 6218 | Calcium Channel |
Fluspirilene (R 6218) is a non-competitive L-type calcium channel antagonist (IC50: 0.03 μM).Fluspirilene is a long-acting antipsychotic compound used in the treatment of schizophrenia. | |||
TP1796 | Albiglutide TFA (782500-75-8 free base) | Albiglutide TFA | Glucagon Receptor |
Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM). | |||
T0706 | Lisinopril dihydrate | Lisinopril,Renacor,MK-521 (dihydrate) | RAAS , MRP |
Lisinopril dihydrate (MK-521) is an orally bioavailable, long-acting angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity. | |||
T1909 | L-701324 | L701324 | NMDAR , iGluR |
L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant. | |||
T6566 | Levobupivacaine hydrochloride | Levobupivacaine HCl,(S)-(-)-Bupivacaine HCl,(S)-(-)-Bupivacaine monohydrochloride | Sodium Channel |
Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, which is the pure S(-)-enantiomer of bupivacaine. It was utilized as a long-acting local anesthetic... | |||
T4991 | Ertapenem sodium | MK-826,L-749345 | Antibacterial , Antibiotic |
Ertapenem sodium (MK-826) is a new long-acting 1-β-methyl carbapenem antibiotic with a broad antibacterial spectrum including common aerobic and anaerobic bacteria and organisms with extended-spectrum β-lactamases. | |||
T0699 | Sulfamonomethoxine | Antibacterial , Antibiotic | |
Sulfamonomethoxine is a long-acting sulfonamide antibacterial agent, blocks the synthesis of folic acid by inhibiting synthetase of dihydropteroate. | |||
T6098 | Cabotegravir | GSK744,GSK-1265744,S/GSK1265744 | HIV Protease |
Cabotegravir (S/GSK1265744) (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor and inhibits the HIV-1 integrase catalyzed strand transfer reaction (IC50: 3.0 nM). | |||
T1423 | 3-Methylsalicylic acid | Hydroxytoluic acid,o-Cresotic acid | COX |
3-Methylsalicylic acid (o-Cresotic acid) is a long-acting salicylate derivative with antilipidemic properties. Hydroxytoluic acid has been shown to lower plasma free fatty acid and cholesterol levels. | |||
T16759 | Ritanserin | R 55667 | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor |
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors. | |||
T6457 | CTEP | mGluR5 inhibitor,RO 4956371 | GluR |
CTEP (RO 4956371) (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold selectivity over other mGlu receptors. | |||
T13106 | TD-5471 hydrochloride | Adrenergic Receptor | |
TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (COPD). | |||
T12829 | Salmeterol | GR33343X | Adrenergic Receptor |
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma. |
Cat No. | Product Name | Synonyms | Targets |
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T1261 | Medroxyprogesterone Acetate | Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,Farlutin,Medroxyprogesterone (acetate) | Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , Androgen Receptor , Endogenous Metabolite |
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally or by intramuscular injection and has also been... | |||
T0086 | Galanthamine hydrobromide | Galantamine hydrobromide,Galanthamine HBr | AChR , AChE |
Galanthamine hydrobromide (Galantamine hydrobromide), a long-acting and centrally active AChE inhibitor (IC50:410 nM), is an allosteric potentiator at neuronal nicotinic ACh receptors. | |||
T3S2007 | MRE-269 | MRE 269,ACT-333679,MRE269 | Prostaglandin Receptor |
MRE-269 (ACT-333679) is an orally available and long-acting prostacyclin receptor agonist prodrug. MRE-269(ACT-333679) is used for the treatment of pulmonary arterial hypertension. MRE-269(ACT-333679) is an active metabo... | |||
T0012 | Cinchonine | LA40221,(8R,9S)-Cinchonine | Apoptosis , P-gp , Parasite |
Cinchonine (LA40221), a local anesthetic of the amide type, now generally used for surface anesthesia. It is one of the most potent and toxic of the long-acting local narcotics and its parenteral use is restricted to spi... | |||
T2520 | Desloratadine | Sch34117,NSC 675447 | Endogenous Metabolite , Histamine Receptor |
Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typical histaminergic effects on H1-receptors in bronchial smoot... |
Cat No. | Product Name | Species | Expression System |
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TMPY-01816 | Pentraxin 3 Protein, Human, Recombinant (His) | Human | HEK293 |
Pentraxin-related protein PTX3, also known as Tumor necrosis factor alpha-induced protein 5, Tumor necrosis factor-inducible gene 14 protein, TSG-14, PTX3 and TNFAIP5, is a secreted protein that contains one pentaxin dom... |