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Cat No. | Product Name | Synonyms | Targets |
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T8435 | YM90K | YM90K hydrochloride,6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)- | GluR , iGluR |
YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride is an antagonist of AMPA receptor. | |||
T4278 | AM966 | LPA Receptor , LPL Receptor | |
AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release. | |||
T7954 | YM976 | PDE | |
YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM) | |||
T10593 | BPR1M97 | Opioid Receptor | |
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.8 nM for MOP and 4.2 nM for NOP.BPR1M97 exhibits anti-injuri... | |||
T40165 | OM99-2 TFA | OM99-2 TFA | |
OM99-2 TFA is an eight-residue peptidomimetic compound, functioning as a tight-binding inhibitor of human brain memapsin 2. It exhibits a high affinity for the target with a Ki value of 9.58 nM, making it a promising can... | |||
T79272 | BDM91514 | ||
BDM91514 enhances antibiotic efficacy by inhibiting AcrB, effectively curbing the proliferation of E. coli BW25113 with an EC90 of 8 μM when coupled with 8 μg/mL Pyridomycin. Additionally, BDM91514 exhibits favorable pla... | |||
T70194 | AM92016 | ||
AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity. | |||
T78200 | BDM91270 | ||
BDM91270 (compound 29) serves as an inhibitor of the E. coli AcrAB-TolC efflux pump, displaying an EC90 value of 0.6 μM against wild-type E. coli AcrB. It has applications in research on Escherichia coli drug resistance ... | |||
T15768 | LM985 | Others | |
LM985 is one of a series of compounds based on the flavone ring structure. It has anti-tumor activities. | |||
T24663 | YM928 | YM-928,YM 928 | |
YM928 is an orally active antagonist of the AMPA receptor. | |||
T70868 | HM90822 | ||
HM90822 is a novel antagonist to the inhibitors of apoptosis (IAPs), potentiating cell death in EGFR-overexpressing non-small-cell lung cancer cells. | |||
T69733 | LM9 | ||
LM9 is a MyD88 inhibitor which prevents atherosclerosis by regulating inflammatory responses and oxidative stress in macrophages. | |||
T40393 | OM99-2 | OM99-2 | |
OM99-2 is an eight-residue peptidomimetic with a high affinity for human brain memapsin 2, exhibiting a Ki value of 9.58 nM. This compound represents a significant advancement in the development of BACE1 inhibitors and h... | |||
T10294 | AM9405 | 5-HT Receptor | |
AM9405 is a novel peripherally active cannabinoid type 1 (CB1) and serotonin type 3 receptor agonist. AM9405 inhibits twitch contraction of the ileum and the colon with IC 50 s of 45.71 and 0.076 nM, respectively. AM9405... |
Cat No. | Product Name | Species | Expression System |
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TMPY-03343 | EIF3K Protein, Human, Recombinant (His & GST) | Human | Baculovirus Insect Cells |
EIF3K is a member of the eIF3 subunit K family. It is a component of the eukaryotic translation initiation factor 3 (eIF-3) complex, which is required for several steps in the initiation of protein synthesis. The eIF-... | |||
TMPK-00553 | ADAM9 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
A disintegrin and metalloproteinase 9 (ADAM9) is a member of the transmembrane ADAM family. It is expressed in different types of solid cancer and promotes tumor invasiveness. ADAM9 may be a prognostic marker for vestibu... | |||
TMPH-01272 | TRIM9 Protein, Human, Recombinant (His & SUMO) | Human | E. coli |
E3 ubiquitin-protein ligase which ubiquitinates itself in cooperation with an E2 enzyme UBE2D2/UBC4 and serves as a targeting signal for proteasomal degradation. May play a role in regulation of neuronal functions and ma... | |||
TMPY-02404 | ADAM9 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
ADAM9 (A disintegrin and metallopeptidase domain 9, MDC9, meltrin gamma), is a type 1 transmembrane protein that has been associated with cancer development and metastases. ADAM9 is consistently overexpressed in various ... |