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Results for "

atpase activity

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    127
    TargetMol | Inhibitors_Agonists
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    3
    TargetMol | Peptide_Products
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    1
    TargetMol | Dye_Reagents
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    TargetMol | Inhibitors_Agonists
Brefeldin A
Decumbin, Cyanein, BFA, Ascotoxin
T606220350-15-6
Brefeldin A (Cyanein) belongs to the class of macrolide antibiotics and is an ATPase inhibitor (IC50=0.2 μM). Brefeldin A can induce tumor cell differentiation and apoptosis, and also possesses autophagy inhibitory activity.
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Novobiocin Sodium
Cathomycinsodium, Albamycinsodium
T09741476-53-5
Novobiocin Sodium (Albamycinsodium) binds to DNA gyrase and blocks adenosine triphosphatase (ATPase) activity. Novobiocin sodium is an antibiotic compound derived from Streptomyces niveus. It has a chemical structure similar to coumarin.
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Bufalin
T1719465-21-4
Bufalin is an active ingredient and one of the glycosides in the traditional Chinese medicine ChanSu; it is also a bufadienolide toxin originally isolated from the venom of the Chinese toad Bufo gargarizans, with potential cardiotonic and antineoplastic a
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Cinobufagin
Cinobufagine
T3432470-37-1
Cinobufagin (Cinobufagine) is a selective Na+ K+-ATPase inhibitor. The activity of Cinobufagin is same as ouabain.
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Oleandrin
Neriostene, Folinerin, Foliandrin
T5S0890465-16-7
1. Oleandrin (Folinerin), the principal cardiac glycoside component of PBI-524, can quantitatively account for regulation of BDNF at both the protein and transcriptional levels. 2. Oleandrin are known to inhibit the Na, K-ATPase pump, resulting in a consequent increase in calcium influx in heart muscle. 3. Oleandrin has stronger anti-proliferative activity in undifferentiated CaCO-2 cells (IC50, 8.25 nM) , causes an autophagic cell death and altered ERK phosphorylation in undifferentiated.
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Paxilline
T1237357186-25-1
Paxilline is an indole alkaloid mycotoxin from *Penicillium paxilli*, acting as a potent BK channel inhibitor via an almost exclusively closed-channel block mechanism. Paxilline possesses significant anticonvulsant activity.
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7-10 days
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Neriifolin
NSC 123976, NSC123976, 17beta-Neriifolin, 17β-Neriifolin
T124830466-07-9
Neriifolin (17β-Neriifolin), a cardiac glycoside extracted from the unripe fruit of Cerbera manghas, is a Na+K+-ATPase inhibitor with anticancer activity that inhibits cell proliferation by suppressing HOXA9-dependent gene expression and inducing apoptosis in the human acute myeloid cell line, THP-1. Neriifolin induces cell cycle arrest and apoptosis in human hepatocellular carcinoma HepG2 cells and can be used in prostate cancer research.
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7-10 days
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Acerinol
T2361019902-53-5
Acerinol is an active ingredient from traditional Chinese medicinal herbs. It could be used as a cancer multidrug resistance reversal agent. Acerinol can significantly stimulate the activity of ABCB1 ATPase without affecting the expression of ABCB1 on nei
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Mycalolide B
T38609122752-21-0
Mycalolide-B is a marine sponge-derived compound that functions as a selective inhibitor of actomyosin ATPase. It effectively hinders ATP-induced contraction and Mg2+-ATPase activity in the absence of Ca2+.
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Agnuside
chasteberry oil
T386811027-63-7
Agnuside (chasteberry oil) inhibits COX-2 (IC50: 0.026 mg ml) but exhibits less than 10% inhibition of COX-1 at this concentration. It also inhibits 46.3, 66.8, and 82.1% of P-glycoprotein (P-gp) ATPase activity at concentrations of 5, 25, and 100 μM, respectively.
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Wilforine
T6S104911088-09-8
Wilforine, a sesquiterpene pyridine alkaloid, is an important bioactive compound in T. wilfordii plants and is effective in treating idiopathic pulmonary fibrosis. Wilforine exhibits an anti-inflammatory effect, which might be mediated by the down-regulation of inflammatory factors TNF-α, IL-6, and NO. Additionally, it has insecticidal activity by inhibiting the Na+-K+-ATPase in the central nervous system.
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Actein
T719018642-44-9
Actein has a stimulatory effect on osteoblastic bone formation or has potential activity against osteoporosis, it also can prevent oxidative damage to osteoblasts in osteoporotic patients. Actein's ability to pathways involved in lipid disorders and carci
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Norbatzelladine L
T726451187954-93-3
Norbatzelladine L, an inhibitor of both the catalytic and functional activities of the Pdr5p transporter, suppresses Pdr5p ATPase activity with an IC50 of 3.8 µM. Additionally, it exhibits antifungal, antiparasitic, antiviral, antibacterial, and antitumoral properties.
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Licoflavone B
TN186091433-17-9
Licoflavone B has schistosomicidal activity, it showed high S. mansoni ATPase (IC50 of 23.78 μM) and ADPase (IC50 of 31.50 μM) inhibitory activities.
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Echinatine
TN3914480-83-1
Echinatin exerts a protective effect against ischemia reperfusion (I R)-induced myocardial injury on hearts, this effect may be attributed to the antioxidant and anti-inflammatory activities of this compound. Echinatin can inhibit DNP-ATPase activity whil
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HU-331
​Cannabidiol Hydroxy Quinone
TN7359137252-25-6
Cannabidiol hydroxyquinone (HU-331) is potentially an active metabolite of cannabidiol that could play a role in inducing apoptosis. It functions by inhibiting the ATPase activity of topoisomerase IIα through a noncompetitive mechanism.
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Ouabagenin
TN7752508-52-1
Ouabagenin, a naturally occurring LXR ligand with selective agonist activity, functions as an EC 3.6.3.9 (Na(+) K(+)-transport ATPase) inhibitor [1] [2].
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3-Oxo-bufalin
TN81304029-65-6
3-Oxo-bufalin is an active compound isolated from cultured toad liver tissues. It is produced via metabolic pathways as a stereoselectively distinct metabolite of Bufalin, catalyzed by the enzyme 3β-dehydrogenase. Bufalin acts as an inhibitor of Na+ K+-ATPase and possesses antitumor activity.
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cis-3-Indoleacrylic acid
TN840329953-72-8
The compound cis-3-Indoleacrylic acid acts as a nematicidal agent and can be isolated from Streptomyces youssoufiensis YMF3.862. It functions as a V-ATPase inhibitor, reducing both the expression and enzymatic activity of V-ATPase. Additionally, cis-3-Indoleacrylic acid causes swelling in Meloidogyne incognita larvae and notable cracking on the cuticle surface [LC50: 16.31 μg mL]. It also inhibits the accumulation of H+ within nematodes.
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Acremorin E
TN9022
Acremorin E (Compound 7) is a terpene compound with antifungal properties. It exhibits activity against C. gattii (MIC: 8 μg mL) by enhancing ribosome biosynthesis and RNA-binding gene expression, while inhibiting RNA, nucleic acid metabolism, and ATPase activity.
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Chebulinic acid
TQ018418942-26-2
Chebulinic acid is a potent inhibitor of M. tuberculosis DNA gyrase. It also can inhibit SMAD-3 phosphorylation and H+ K+-ATPase activity.
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