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Glucocorticoid Receptor

The glucocorticoid receptor (GR, or GCR) also known as NR3C1 (nuclear receptor subfamily 3, group C, member 1) is the receptor to which cortisol and other glucocorticoids bind. The GR is expressed in almost every cell in the body and regulates genes controlling the development, metabolism, and immune response.
Cat. No. Product name CAS No. Purity Chemical Structure
T37908 Glucocorticoid receptor agonist-1 2166375-82-0 98%
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM extracted from patent WO2017210471A1, compound 41[1].
T34383 Rofleponide 144459-70-1 98%
Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.
TN3910 Ecdysone 3604-87-3 98%
Ecdysone signaling through Ecdysone receptor isoform B1 is required cell autonomously for the muscle death. A nctional Bombyx Ecdysone receptor binds to EcRE-D a...
T1614 Hydrocortisone 50-23-7 98%
Hydrocortisone, a glucocorticoid receptor agonist, promotes protein catabolism, gluconeogenesis, capillary wall stability, renal excretion of calcium, and suppre...
T9022 AZD9977 1850385-64-6 98%
AZD 9977 is a novel, selective modulator of mineralocorticoid receptor .
T2526 Ciclesonide 126544-47-6 98%
Ciclesonide(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.
T0947L Dexamethasone Phosphate disodium 2392-39-4 98%
Dexamethasone disodium phosphate is a water-soluble form of the synthetic glucocorticoid dexamethasone.
T2748 Cortodoxone 152-58-9 98%
Cortodoxone is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.
T1560 Prednisolone 50-24-8 98%
Prednisolone is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
T0820 Triamcinolone acetonide 76-25-5 98%
Triamcinolone acetonide is a Corticosteroid. The mechanism of action of triamcinolone acetonide is as a Corticosteroid Hormone Receptor Agonist. It is an anti-in...
T0354 Canrenone 976-71-6 98%
Canrenone is an aldosterone antagonist with potassium-sparing diuretic activity.
T3962 TPI-1 79756-69-7 98%
TPI-1 is a SHP-1 inhibitor.
T1076 Dexamethasone 50-02-2 98%
Dexamethasone is a glucocorticoid receptor agonist and an IL receptor modulator.Dexamethasone inhibits production of exosomes containing inflammatory microRNA-15...
T1102 Mifepristone 84371-65-3 98%
Mifepristone is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational Hormone Receptor Antagonist.
T0276 Hydrocortisone Valerate 57524-89-7 98%
Hydrocortisone Valerate has anti-inflammatory, antipruritic and vasoconstrictive properties.
T67742 EX-A5386 2452396-89-1 98%
EX-A5386 is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.
T8777 Beclometasone 4419-39-0 98%
BecloMethasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma...
T15246 Esaxerenone 1632006-28-0 98%
Esaxerenone is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor.
T0367 Fluocinolone (Acetonide) 67-73-2 98%
Fluocinolone acetonide is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, gel, lotion, ...
T14301 Apararenone 945966-46-1 98%
Apararenone is a novel antagonist of non-steroidal mineralocorticoid receptor, and for the treatment of diabetic nephropathies and non-alcoholic steatohepatitis....
Glucocorticoid receptor agonist-1
T37908
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM extracted from patent WO2017210471A1, compound 41[1].
Rofleponide
T34383
Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.
Ecdysone
TN3910
Ecdysone signaling through Ecdysone receptor isoform B1 is required cell autonomously for the muscle death. A nctional Bombyx Ecdysone receptor binds to EcRE-D a...
Hydrocortisone
T1614
Hydrocortisone, a glucocorticoid receptor agonist, promotes protein catabolism, gluconeogenesis, capillary wall stability, renal excretion of calcium, and suppre...
AZD9977
T9022
AZD 9977 is a novel, selective modulator of mineralocorticoid receptor .
Ciclesonide
T2526
Ciclesonide(RPR251526) is a glucocorticoid used for the treatment of obstructive airway diseases.
Dexamethasone Phosphate disodium
T0947L
Dexamethasone disodium phosphate is a water-soluble form of the synthetic glucocorticoid dexamethasone.
Cortodoxone
T2748
Cortodoxone is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.
Prednisolone
T1560
Prednisolone is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
Triamcinolone acetonide
T0820
Triamcinolone acetonide is a Corticosteroid. The mechanism of action of triamcinolone acetonide is as a Corticosteroid Hormone Receptor Agonist. It is an anti-in...
Canrenone
T0354
Canrenone is an aldosterone antagonist with potassium-sparing diuretic activity.
TPI-1
T3962
TPI-1 is a SHP-1 inhibitor.
Dexamethasone
T1076
Dexamethasone is a glucocorticoid receptor agonist and an IL receptor modulator.Dexamethasone inhibits production of exosomes containing inflammatory microRNA-15...
Mifepristone
T1102
Mifepristone is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational Hormone Receptor Antagonist.
Hydrocortisone Valerate
T0276
Hydrocortisone Valerate has anti-inflammatory, antipruritic and vasoconstrictive properties.
EX-A5386
T67742
EX-A5386 is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.
Beclometasone
T8777
BecloMethasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma...
Esaxerenone
T15246
Esaxerenone is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor.
Fluocinolone (Acetonide)
T0367
Fluocinolone acetonide is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, gel, lotion, ...
Apararenone
T14301
Apararenone is a novel antagonist of non-steroidal mineralocorticoid receptor, and for the treatment of diabetic nephropathies and non-alcoholic steatohepatitis....
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