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Glucocorticoid receptor agonist-1

🥰Excellent
Catalog No. T37908Cas No. 2166375-82-0

Glucocorticoid receptor agonist-1, a potent glucocorticoid receptor agonist, has an IC50 of 2.8 nM[1].

Glucocorticoid receptor agonist-1

Glucocorticoid receptor agonist-1

🥰Excellent
Purity: 99.16%
Catalog No. T37908Cas No. 2166375-82-0
Glucocorticoid receptor agonist-1, a potent glucocorticoid receptor agonist, has an IC50 of 2.8 nM[1].
Pack SizePriceAvailabilityQuantity
1 mg$89In Stock
5 mg$182In Stock
10 mg$293In Stock
25 mg$583In Stock
50 mg$932In Stock
100 mg$1,490In Stock
200 mg$1,970In Stock
1 mL x 10 mM (in DMSO)$229In Stock
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This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.
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Batch Information

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Purity:99.16%
ee:100%
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COA CSFC HNMR LCMS

Product Introduction

Bioactivity
Description
Glucocorticoid receptor agonist-1, a potent glucocorticoid receptor agonist, has an IC50 of 2.8 nM[1].
Targets&IC50
GR:2.8 nM (IC50)
In vitro
Glucocorticoid receptor agonist-1 (Compound 41) is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM.[1]
Chemical Properties
Molecular Weight569.69
FormulaC35H39NO6
Cas No.2166375-82-0
Smiles[H][C@]1(O[C@]2([H])C[C@@]3([H])[C@]4([H])CCC5=CC(=O)C=C[C@]5(C)[C@@]4([H])[C@@H](O)C[C@]3(C)[C@@]2(O1)C(=O)CO)c1ccc(Cc2cccc(N)c2)cc1
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 50 mg/mL (87.77 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.7553 mL8.7767 mL17.5534 mL87.7670 mL
5 mM0.3511 mL1.7553 mL3.5107 mL17.5534 mL
10 mM0.1755 mL0.8777 mL1.7553 mL8.7767 mL
20 mM0.0878 mL0.4388 mL0.8777 mL4.3884 mL
50 mM0.0351 mL0.1755 mL0.3511 mL1.7553 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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μL
2 Enter the in vivo formulation:
% DMSO
%
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% Saline/PBS/ddH2O

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

GlucocorticoidReceptorGlucocorticoid receptor agonist-1Glucocorticoid receptor agonist1Glucocorticoid receptor agonist 1Glucocorticoid ReceptorADCCytotoxinADC Cytotoxin
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